Cat. No. 5549
Chemical Name: 6-(4-Methyl-1-piperazinyl)-11H-dibe
Biological ActivityPotent and selective hM3Dq DREADD agonist (EC50 = 2.8 nM). Exhibits >10,000-fold selectivity for hM3Dq over hM3.
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Certificate of Analysis / Safety Data Sheet
Chen et al (2015) The first structure-activity relationship studies for designer receptors exclusively activated by designer drugs. ACS Chem.Neurosci. 6 476. PMID: 25587888.
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November 12 - 16, 2016
San Diego, CA, USA