Perlapine

Cat. No. 5549

Perlapine C19H21N3 [1977-11-3]

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Chemical Name: 6-(4-Methyl-1-piperazinyl)-11H-dibenz[b,e]azepine

Biological Activity

Potent and selective hM3Dq DREADD agonist (EC50 = 2.8 nM). Exhibits >10,000-fold selectivity for hM3Dq over hM3.

Technical Data

M.Wt:
291.39
Formula:
C19H21N3
Solubility:
Soluble to 50 mM in DMSO and to 5 mM in water with gentle warming
Purity:
>99 %
Storage:
Store at RT
CAS No:
1977-11-3

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.

Certificate of Analysis / Product Datasheet / Safety Datasheet

References are publications that support the products' biological activity.

Chen et al (2015) The first structure-activity relationship studies for designer receptors exclusively activated by designer drugs. ACS Chem.Neurosci. 6 476. PMID: 25587888.

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Citations are publications that use Tocris products.

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