Cat. No. 5549
Chemical Name: 6-(4-Methyl-1-piperazinyl)-11H-dibe
Biological ActivityPotent and selective hM3Dq DREADD agonist (EC50 = 2.8 nM). Exhibits >10,000-fold selectivity for hM3Dq over hM3.
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Certificate of Analysis / Product Datasheet / Safety Data Sheet
Chen et al (2015) The first structure-activity relationship studies for designer receptors exclusively activated by designer drugs. ACS Chem.Neurosci. 6 476. PMID: 25587888.
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One Day Symposium
March 1, 2017
Amsterdam, The Netherlands