Cat. No. 5549
Chemical Name: 6-(4-Methyl-1-piperazinyl)-11H-dibe
Biological ActivityPotent and selective hM3Dq DREADD agonist (EC50 = 2.8 nM). Exhibits >10,000-fold selectivity for hM3Dq over hM3.
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Certificate of Analysis / Product Datasheet / Safety Datasheet
Chen et al (2015) The first structure-activity relationship studies for designer receptors exclusively activated by designer drugs. ACS Chem.Neurosci. 6 476. PMID: 25587888.
If you know of a relevant reference for this product please let us know.
Citations are publications that use Tocris products.
Do you know of a great paper that uses Perlapine from Tocris? If so please let us know.
View Related Products by Product Action
Keywords: Perlapine, supplier, Perlapine, potent, selective, hM3Dq, DREADD, agonists, antagonism, designer, receptors, drugs, muscarinic, receptors, activators, Tocris Bioscience, DREADD Ligand Activator products