Cat. No. 5418
Chemical Name: 1-[2-[2,5-Dimethyl-1-(phenylmethyl)
Biological ActivitySelective S1P2 allosteric agonist (EC50 = 0.48 μM). Selective for S1P2 receptors over a panel of 29 other receptors and transporters.
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Certificate of Analysis / Product Datasheet / Safety Datasheet
References are publications that support the products' biological activity.
Satsu et al (2013) A sphingosine 1-phosphate receptor 2 selective allosteric agonist. Bioorg.Med.Chem. 21 5373. PMID: 23849205.
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Keywords: CYM 5520, supplier, selective, allosteric, agonists, sphingosine-1-phosphate, receptor, 2, S1P2, S1PR2, agonism, CYM5520, Tocris Bioscience, Sphingosine-1-Phosphate Receptor Agonist products
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