TC-G 1003

Cat. No. 5080

TC-G 1003 C26H25ClN2O2 [1021912-42-4]

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Chemical Name: 3-[4-(3-Aminopropoxy)-7-chloro-3-(3,5-dimethylphenyl)-6-quinolinyl]phenol

Biological Activity

High affinity somatostatin sst2 receptor agonist (Ki = 0.025 nM). Inhibits growth hormone secretion and attenuates laser-induced ocular neovascular lesion size in rats.

Technical Data

M.Wt:
432.94
Formula:
C26H25ClN2O2
Solubility:
Soluble to 100 mM in DMSO and to 100 mM in ethanol
Purity:
>98 %
Storage:
Store at -20°C
CAS No:
1021912-42-4

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.

Certificate of Analysis / Product Datasheet / Safety Datasheet

References are publications that support the products' biological activity.

Wolkenberg et al (2011) Design, synthesis, and evaluation of novel 3,6-diaryl-4-aminoalkoxyquinolines as selective agonists of somatostatin receptor subtype 2. J.Med.Chem. 54 2351. PMID: 21395312.

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Keywords: TC-G 1003, supplier, TC-G1003, high, affinity, somatostatin, sst2, receptors, agonists, Tocris Bioscience, Somatostatin (sst) Receptor Agonist products

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