Cat. No. 5080
Chemical Name: 3-[4-(3-Aminopropoxy)-7-chloro-3-(3
Biological ActivityHigh affinity somatostatin sst2 receptor agonist (Ki = 0.025 nM). Inhibits growth hormone secretion and attenuates laser-induced ocular neovascular lesion size in rats.
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Certificate of Analysis / Product Datasheet / Safety Data Sheet
Wolkenberg et al (2011) Design, synthesis, and evaluation of novel 3,6-diaryl-4-aminoalkoxyquinolines as selective agonists of somatostatin receptor subtype 2. J.Med.Chem. 54 2351. PMID: 21395312.
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Keywords: TC-G 1003, supplier, TC-G1003, high, affinity, somatostatin, sst2, receptors, agonists, Tocris Bioscience, Somatostatin (sst) Receptor Agonist products
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