Cat. No. 4948
Alternative Name: ML250
Chemical Name: 5-Chloro-2-(9H-fluoren-9-yl)-4-(4-m
Biological ActivityNovel non-peptide antagonist of neuropeptide W/B receptor 1 (NPBWR1, GPR7) (IC50 = 0.12 μM).
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Certificate of Analysis / Product Datasheet / Safety Datasheet
References are publications that support the products' biological activity.
Guerrero et al (2013) SAR analysis of novel non-peptidic NPBWR1 (GPR7) antagonists. Bioorg.Med.Chem.Lett. 23 614. PMID: 23287738.
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Citations are publications that use Tocris products.
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Keywords: CYM 50769, supplier, NPBWR1, antagonists, neuropeptide, B, W, receptor, 1, CYM50769, ML250, GPR7, Tocris Bioscience, Other Peptide Receptor products
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