CYM 50769

Cat. No. 4948

CYM 50769 C24H17ClN2O3 [1421365-63-0]

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Alternative Name: ML250

Chemical Name: 5-Chloro-2-(9H-fluoren-9-yl)-4-(4-methoxyphenoxy)-3(2H)-pyridazinone

Biological Activity

Novel non-peptide antagonist of neuropeptide W/B receptor 1 (NPBWR1, GPR7) (IC50 = 0.12 μM).

Technical Data

M.Wt:
416.86
Formula:
C24H17ClN2O3
Solubility:
Soluble to 100 mM in DMSO
Purity:
>98 %
Storage:
Store at +4°C
CAS No:
1421365-63-0

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.

Certificate of Analysis / Product Datasheet / Safety Datasheet

References are publications that support the products' biological activity.

Guerrero et al (2013) SAR analysis of novel non-peptidic NPBWR1 (GPR7) antagonists. Bioorg.Med.Chem.Lett. 23 614. PMID: 23287738.

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Citations are publications that use Tocris products.

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Keywords: CYM 50769, supplier, NPBWR1, antagonists, neuropeptide, B, W, receptor, 1, CYM50769, ML250, GPR7, Tocris Bioscience, Other Peptide Receptor products

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