5-Iodo-A-85380, 5-trimethylstannyl N-BOC derivative
Cat. No. 1527
Chemical Name: (2S)-2-[[[5-(Trimethylstannyl)-3-py
Biological ActivityPrecursor to the highly potent and selective ligand for the α4β2 nicotinic receptor, 5-Iodo-A-85380 (Cat. No.1518). Suitable for radioiodination.
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Certificate of Analysis / Product Datasheet / Safety Datasheet
References are publications that support the products' biological activity.
Mukhin et al (2000) 5-Iodo-A-85380, an α4β2 subtype-selective ligand for nicotinic acetylcholine receptors. Mol.Pharmacol. 57 642. PMID: 10692507.
Koren et al (1998) 2-, 5-, and 6-Halo-3-(2(S)-azetidinylmethoxy)pyridines: synthesis, affinity for nicotinic acetylcholine receptors, and molecular modeling. J.Med.Chem. 41 3690. PMID: 9733494.
If you know of a relevant reference for 5-Iodo-A-85380, 5-trimethylstannyl N-BOC derivative please let us know.
Citations are publications that use Tocris products.
Do you know of a great paper that uses 5-Iodo-A-85380, 5-trimethylstannyl N-BOC derivative from Tocris? If so please let us know.
View Related Products by Target
View Related Products by Product Action
Keywords: 5-Iodo-A-85380, 5-trimethylstannyl N-BOC derivative, supplier, Precursor, α4β2, a4b2, Nicotinic, Receptors, Acetylcholine, nAChR, Non-Selective, Subtypes, Other, 5-Iodo-A-853805-trimethylstannyl, N-BOC, derivative, Tocris Bioscience, Nicotinic (α4β2) Receptor Agonist products
Find multiple products by catalog number
New Products in this Area
Potent positive allosteric modulator of α4β2 nAChRs; also inhibitor of (α4)2(β2)3, muscle-type and Torpedo nAChRs
Follow Tocris on LinkedIn
Visit our LinkedIn page for the latest Tocris news, events and updates.