Cat. No. 4824
Chemical Name: N-[5-[3,4-Difluoro-2-[(2-fluoro-4-i
Biological ActivityInhibitor of MEK1. Analog of PD 184352 (Cat. No. 4237).
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Certificate of Analysis / Product Datasheet / Safety Datasheet
References are publications that support the products' biological activity.
Zhang et al (2009) Targeting cancer with small molecule kinase inhibitors. Nat.Rev.Cancer 9 28. PMID: 19104514.
Ohren et al (2004) Structures of human MAP kinase kinase 1 (MEK1) and MEK2 describe novel competitive kinase inhibition. Nat.Struct.Mol.Biol. 11 1192. PMID: 15543157.
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Citations are publications that use Tocris products.
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Keywords: PD 334581, supplier, PD334581, MEK1, kinase, inhibitors, inhibits, mitogen, activated, protein, kinase, 1, Tocris Bioscience, MEK Inhibitor products
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August 20 - 24, 2017
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