COR 170

Cat. No. 4756

COR 170  [1048039-15-1]

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Chemical Name: N-(Adamant-1-yl)-4-oxo-1-pentyl-6-phenyl-1,4-dihydroquinoline-3-carboxamide

Biological Activity

Selective inverse agonist of CB2 receptors (Ki values are 3.8 and >10,000 nM for CB2 and CB1, respectively).

Technical Data

M.Wt:
468.63
Formula:
C31H36N2O2
Solubility:
Soluble to 100 mM in ethanol and to 20 mM in DMSO
Purity:
>99 %
Storage:
Store at RT
CAS No:
1048039-15-1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.

Certificate of Analysis / Product Datasheet / Safety Data Sheet

Contartese et al (2012) A novel CB2 agonist, COR167, potently protects rat brain cortical slices against OGD and reperfusion injury. Pharmacol.Res. 66 555. PMID: 23036353.

Pasquini et al (2008) Investigations on the 4-quinolone-3-carboxylic acid motif. 2. Synthesis and structure-activity relationship of potent and selective cannabinoid-2 receptor agonists endowed with analgesic activity in vivo. J.Med.Chem. 51 5075. PMID: 18680276.

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Keywords: COR 170, supplier, COR170, CB2, receptors, C2BR, inverse, agonists, selective, cannabinoids, Tocris Bioscience, CB2 Receptor Antagonist products

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