Cat. No. 4756
Chemical Name: N-(Adamant-1-yl)-4-oxo-1-pentyl-6-p
Biological ActivitySelective inverse agonist of CB2 receptors (Ki values are 3.8 and >10,000 nM for CB2 and CB1, respectively).
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Certificate of Analysis / Product Datasheet / Safety Datasheet
References are publications that support the products' biological activity.
Contartese et al (2012) A novel CB2 agonist, COR167, potently protects rat brain cortical slices against OGD and reperfusion injury. Pharmacol.Res. 66 555. PMID: 23036353.
Pasquini et al (2008) Investigations on the 4-quinolone-3-carboxylic acid motif. 2. Synthesis and structure-activity relationship of potent and selective cannabinoid-2 receptor agonists endowed with analgesic activity in vivo. J.Med.Chem. 51 5075. PMID: 18680276.
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Citations are publications that use Tocris products.
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Keywords: COR 170, supplier, COR170, CB2, receptors, C2BR, inverse, agonists, selective, cannabinoids, Tocris Bioscience, CB2 Receptor Antagonist products
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Potent and selective CB2 partial agonist; orally biovailable
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