Cat. No. 4677
Chemical Name: 2-Chloro-3-[2-(2,4-dichlorophenoxy)
Biological ActivityPotent sphingosine-1-phosphate receptor 4 (S1P4) agonist (EC50 = 45 nM). Displays no activity at other S1P receptor subtypes (S1P1-3 and S1P5) at concentrations up to 25 μM.
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Certificate of Analysis / Product Datasheet / Safety Data Sheet
Guerrero et al (2011) Discovery, design and synthesis of novel potent and selective sphingosine-1-phosphate 4 receptor (S1P4-R) agonists. Bioorg.Med.Chem.Lett. 22 537. PMID: 22119461.
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Keywords: CYM 50260, supplier, CYM50260, sphingosine-1-phosphate, receptors, S1P4, agonists, potent, selective, Tocris Bioscience, Sphingosine-1-Phosphate Receptor Agonist products
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