CID 2011756

Cat. No. 4644

CID 2011756 C22H21ClN2O3 [638156-11-3]

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Chemical Name: 5-(3-Chlorophenyl)-N-[4-(4-morpholinylmethyl)phenyl]-2-furancarboxamide

Biological Activity

Protein kinase D (PKD) inhibitor (IC50 values are 0.6, 0.7 and 3.2 μM for PKD2, PKD3 and PKD1 respectively). Cell permeable (EC50 = 10 μM for PKD1 inhibition). ATP-competitive.

Technical Data

M.Wt:
396.87
Formula:
C22H21ClN2O3
Solubility:
Soluble to 50 mM in DMSO
Purity:
>99 %
Storage:
Store at RT
CAS No:
638156-11-3

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.

Certificate of Analysis / Product Datasheet / Safety Datasheet

References are publications that support the products' biological activity.

Sharlow et al (2011) Discovery of diverse small molecule chemotypes with cell-based PKD1 inhibitory activity. PLoS One 6 e25134. PMID: 21998636.

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Keywords: CID 2011756, supplier, CID2011756, pan, protein, kinase, D, PKD, inhibits, inhibitors, cell, permeable, ATP, competitive, Tocris Bioscience, Protein Kinase D Inhibitor products

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