TC-O 9311

Cat. No. 4255

TC-O 9311 C20H19N3O4 [444932-31-4]

Price and Availability

For TC-O 9311 pricing & availability please select your country from the drop down menu:
Submit
By clicking submit you agree to accept a cookie from Tocris Bioscience. For details, please read our privacy and cookie policy.

Chemical Name: 3,5-Dimethoxybenzoic acid 2-[(1-naphthalenylamino)carbonyl]hydrazide

Biological Activity

Potent GPR139 agonist (EC50 = 39 nM in CHO-K1 cells expressing human GPR139). Displays no activity against a range of 90 diverse targets.

Technical Data

M.Wt:
365.38
Formula:
C20H19N3O4
Solubility:
Soluble to 50 mM in DMSO
Purity:
>98 %
Storage:
Store at +4°C
CAS No:
444932-31-4

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.

Certificate of Analysis / Product Datasheet / Safety Datasheet

References are publications that support the products' biological activity.

Shi et al (2011) Discovery and SAR of a series of agonists at orphan G protein-coupled receptor 139. ACS Med.Chem.Lett. 2 303.

If you know of a relevant reference for TC-O 9311 please let us know.

Citations are publications that use Tocris products.

Do you know of a great paper that uses TC-O 9311 from Tocris? If so please let us know.

View Related Products by Target

View Related Products by Product Action

Keywords: TC-O 9311, supplier, TCO9311, gpr139, receptors, orphan, potent, selective, agonists, Tocris Bioscience, Orphan 7-TM Receptor Agonist products

Quick Order

Find multiple products by catalog number

divider line

GPCR Product Listing

GPCR Product Listing

Highlights over 450 products for GPCRs. Request copy or view PDF today.

divider line

New Products in this Area

Prasugrel

Irreversible P2Y12 antagonist; antiplatelet and orally active

BigLEN (rat)

Potent GPR171 agonist

BigLEN (mouse)

GPR171 agonist

BPTU

P2Y1 allosteric antagonist

AC 265347

CaSR biased allosteric modulator

7α,25-Dihydroxycholesterol

Highly potent GPR183 (EBI2) agonist

AR-C 69931 tetrasodium salt

Highly potent P2Y12 antagonist

FTY 720

Potent S1P receptor agonist; also immunosuppressant

Cinacalcet hydrochloride

Calcium-sensing receptor (CaSR) allosteric agonist; also CYP2D2 inhibitor and Ca2+ channel blocker; orally bioavailable

AMG 837 hemicalcium salt

Potent free fatty acid receptor 1 (FFA1/GPR40) partial agonist

UMB 68

GHB receptor ligand

Sign-up for new product e-alerts
divider line

Twitter Updates

Follow @Tocris on Twitter

Follow us on Twitter!

Tocris is now actively tweeting. For regular updates on news, events and special offers, follow @Tocris on Twitter.