Cat. No. 3921
Chemical Name: N-(Piperidin-1-yl)-5-(4-methoxyphen
Biological ActivityHigh affinity CB1 receptor antagonist (Ki = 4.1 nM). Exhibits significantly reduced lipophilicity compared to other CB1 antagonists.
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Certificate of Analysis / Product Datasheet / Safety Datasheet
Miller et al (2007) Analogs of SR-141716A (Rimonabant) alter d-amphetamine-evoked [3H] dopamine overflow from preloaded striatal slices and amphetamine-induced hyperactivity. Life Sci. 81 63. PMID: 17532007.
Katoch-Rouse et al (2003) Synthesis, structure-activity relationship and evaluation of SR141716 analogues: development of central cannabinoid receptor ligands with lower lipophilicity. J.Med.Chem. 46 642. PMID: 12570386.
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Citations are publications that use Tocris products. Selected citations for NIDA 41020 include:
Buznikov et al (2010) A putative 'pre-nervous' endocannabinoid system in early echinoderm development. Dev Neurosci 32 1. PMID: 19907129.
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Keywords: NIDA 41020, supplier, NIDA41020, cannabinoid, receptors, antagonists, CB1, selective, Tocris Bioscience, CB1 Receptor Antagonist products
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April 22 - 26, 2017
Chicago, IL, USA