Cat. No. 3912
Chemical Name: 4-(7,8,9,10-Tetrahydro-5,7,7,10.10-
Biological ActivityPotent RXR antagonist (IC50 = 18 nM).
Licensing InformationSold under licence.
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Certificate of Analysis / Safety Data Sheet
Suzuki et al (2009) Docosahexaenoic acid induces adipose differentiation-related protein through activation of retinoid X receptor in human choriocarcinoma BeWo cells. Biol.Pharm.Bull. 32 1177. PMID: 19571381.
Alique et al (2006) Vitamin A active metabolite, all-trans retinoic acid, induces spinal cord sensitization. II. Effects after intrathecal administration. Br.J.Pharmacol. 149 65. PMID: 16847438.
Ebisawa et al (1999) Retinoid X receptor-antagonistic diazepinylbenzoic acids. Chem.Pharm.Bull. 47 1778. PMID: 10748721.
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Keywords: HX 531, supplier, HX531, rxrs, retinoids, x, receptors, antagonists, potent, Tocris Bioscience, Retinoid X Receptor Antagonist products
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