WAY 207024 dihydrochloride

Cat. No. 3890

WAY 207024 dihydrochloride C30H32N6.2HCl [872002-73-8]

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Chemical Name: 6-[[4-[2-[4-(1,1-Dimethylethyl)phenyl]-1H-benzimidazol-7-yl]-i-piperazinyl]methyl]-quinoxaline dihydrochloride

Biological Activity

Gonadotropin releasing hormone receptor (GnRH-R) antagonist. Exhibits potent affinity (IC50 values are 12 and 71 nM for human and rat GnRH receptors respectively). Lowers plasma leuteinizing hormone levels in the rat. Orally active.

Licensing Information

Sold for research purposes under agreement from Pfizer Inc.

Technical Data

M.Wt:
549.54
Formula:
C30H32N6.2HCl
Solubility:
Soluble to 85 mM in DMSO
Purity:
>99 %
Storage:
Desiccate at RT
CAS No:
872002-73-8

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.

Certificate of Analysis / Product Datasheet / Safety Datasheet

References are publications that support the products' biological activity.

Pelletier et al (2009) Discovery of 6-({4-[2-(4-tert-butylphenyl)-1H-benzimidazol-4-yl]piperazin-1-yl}methyl)quinoxaline (WAY-207024): an orally active antagonist of the gonadotropin releasing hormone receptor (GnRH-R). J.Med.Chem. 52 214. PMID: 19072222.

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Keywords: WAY 207024 dihydrochloride, supplier, WAY207024, dihydrochloride, GnRH, antagonists, gonadtrophin, releasing, hormone, antagonist, gonadotropin, Tocris Bioscience, Gonadotropin-Releasing Hormone Receptor Antagonist products

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