Cat. No. 3752
Chemical Name: N-[2-Methyl-5-(1-piperidinylsulfony
Biological ActivityEndothelial lipase and lipoprotein lipase inhibitor (IC50 values are 0.13 and 0.10 μM respectively).
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Certificate of Analysis / Product Datasheet / Safety Datasheet
References are publications that support the products' biological activity.
Goodman et al (2009) Discovery of potent, selective sulfonylfuran urea endothelial lipase inhibitors. Bioorg.Med.Chem.Letts. 19 27.
Keller et al (2008) A high-throughput screen for the endothelial lipase using HDL as substrate. J.Biomol.Screen. 13 468. PMID: 18566479.
If you know of a relevant reference for GSK 264220A please let us know.
Citations are publications that use Tocris products.
Do you know of a great paper that uses GSK 264220A from Tocris? If so please let us know.
View Related Products by Product Action
Keywords: GSK 264220A, supplier, GSK264220A, endothelial, lipase, lipoprotein, lipases, inhibitors, inhibits, Tocris Bioscience, Lipase Inhibitor products