Cat. No. 3752
Chemical Name: N-[2-Methyl-5-(1-piperidinylsulfony
Biological ActivityEndothelial lipase and lipoprotein lipase inhibitor (IC50 values are 0.13 and 0.10 μM respectively).
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Certificate of Analysis / Safety Data Sheet
Goodman et al (2009) Discovery of potent, selective sulfonylfuran urea endothelial lipase inhibitors. Bioorg.Med.Chem.Letts. 19 27.
Keller et al (2008) A high-throughput screen for the endothelial lipase using HDL as substrate. J.Biomol.Screen. 13 468. PMID: 18566479.
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Keywords: GSK 264220A, supplier, GSK264220A, endothelial, lipase, lipoprotein, lipases, inhibitors, Tocris Bioscience, Lipase Inhibitor products
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Selective endothelial lipase inhibitor; orally bioavailable
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