Cat. No. 3588
Chemical Name: Piperazine estrone sulfate
Biological ActivityEstrogen receptor agonist. Also inhibits organic anion transporting polypeptide 1B1 (OATP1B1) (IC50= 70 nM).
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All Tocris products are intended for laboratory research use only.
Certificate of Analysis / Product Datasheet / Safety Data Sheet
Obaidat et al (2009) A cell-based high-throughput assay to identify inhibitors of organic anion transporting polypeptides 1B1 and 1B3. FASEB J. 23 748.
Williams et al (2004) Estrogen regulation of the cytochrome P450 3A subfamily in humans. J.Pharmacol.Exp.Ther. 311 728. PMID: 15282264.
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Keywords: Estropipate, supplier, Estrogen, receptor, agonists, OATP1B, inhibitors, inhibits, Tocris Bioscience, Estrogen and Related Receptor Agonist products