Cat. No. 3588
Chemical Name: Piperazine estrone sulfate
Biological ActivityEstrogen receptor agonist. Also inhibits organic anion transporting polypeptide 1B1 (OATP1B1) (IC50= 70 nM).
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Certificate of Analysis / Product Datasheet / Safety Datasheet
Obaidat et al (2009) A cell-based high-throughput assay to identify inhibitors of organic anion transporting polypeptides 1B1 and 1B3. FASEB J. 23 748.
Williams et al (2004) Estrogen regulation of the cytochrome P450 3A subfamily in humans. J.Pharmacol.Exp.Ther. 311 728. PMID: 15282264.
If you know of a relevant reference for this product please let us know.
Citations are publications that use Tocris products.
Do you know of a great paper that uses Estropipate from Tocris? If so please let us know.
View Related Products by Product Action
Keywords: Estropipate, supplier, Estrogen, receptor, agonists, OATP1B, inhibitors, inhibits, Tocris Bioscience, Estrogen and Related Receptor Agonist products