Cat. No. 3588

Estropipate C18H22O5S.C4H10N2 [7280-37-7]

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Chemical Name: Piperazine estrone sulfate

Biological Activity

Estrogen receptor agonist. Also inhibits organic anion transporting polypeptide 1B1 (OATP1B1) (IC50= 70 nM).

Technical Data

Soluble to 5 mM in water and to 100 mM in DMSO
>97 %
Store at RT

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.

Certificate of Analysis / Safety Data Sheet

Certificate of Analysis: View current batch
Safety Data Sheet: View Safety Data Sheet

Obaidat et al (2009) A cell-based high-throughput assay to identify inhibitors of organic anion transporting polypeptides 1B1 and 1B3. FASEB J. 23 748.

Williams et al (2004) Estrogen regulation of the cytochrome P450 3A subfamily in humans. J.Pharmacol.Exp.Ther. 311 728. PMID: 15282264.

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Keywords: Estropipate, supplier, Estrogen, receptor, agonists, OATP1B, inhibitors, inhibits, Tocris Bioscience, Estrogen and Related Receptor Agonist products

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