E4CPG

Cat. No. 1009

E4CPG C11H13NO4 [170846-89-6]

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Chemical Name: (RS)-α-Ethyl-4-carboxyphenylglycine

Biological Activity

Novel group I/group II metabotropic glutamate receptor antagonist, more potent than (RS)-MCPG (Cat. No. 0336).

Technical Data

M.Wt:
223.23
Formula:
C11H13NO4
Solubility:
Soluble to 100 mM in 1.1eq. NaOH
Purity:
>99 %
Storage:
Store at RT
CAS No:
170846-89-6

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.

Certificate of Analysis / Safety Data Sheet

Certificate of Analysis: View current batch
Safety Data Sheet: View Safety Data Sheet

Sekiyama et al (1996) Structure-activity relationships of new agonists and antagonists of different metabotropic glutamate receptor subtypes. Br.J.Pharmacol. 117 1493. PMID: 8730745.

Bedingfield et al (1995) Structure-activity relationships for a series of phenylglycine derivatives acting at metabotropic glutamate receptors (mGluRs). Br.J.Pharmacol. 116 3323. PMID: 8719814.

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Citations are publications that use Tocris products.

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Keywords: E4CPG, supplier, Group, II, group, I, mGlur, antagonists, Receptors, mGlu2, mGlu3, mGluR2, mGluR3, Glutamate, Metabotropic, mGlu1, mGlu5, mGluR1, mGluR5, Tocris Bioscience, Glutamate (Metabotropic) Group I Receptor Antagonist products

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