Cat. No. 3500
Chemical Name: rel-5-(1,1-Dimethylheptyl)-2-[(1R,3
Biological ActivityPotent CB1 receptor agonist (Ki = 2.2 nM). Exhibits analgesic, motor depressant, anticonvulsant and hypothermic effects in vivo.
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Certificate of Analysis / Safety Data Sheet
Huffman et al (2008) Synthesis and pharmacology of 1-deoxy analogs of CP-47,497 and CP-55,940. Bioorg.Med.Chem. 16 322. PMID: 17919913.
Melvin et al (1993) Structure-activity relationships for cannabinoid receptor-binding and analgesic activity: studies of bicyclic cannabinoid analogs. Mol.Pharmacol. 44 1008. PMID: 8246904.
Weissman et al (1982) Cannabimimetic activity from CP-47,497, a derivative of 3-phenylcyclohexanol. J.Pharmacol.Exp.Ther. 223 516. PMID: 6290642.
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Keywords: (±)-CP 47497, supplier, Potent, CB1, agonists, cannabinoids, Receptors, (±)-CP47497, cb1r, Tocris Bioscience, CB1 Receptor Agonist products