Cat. No. 1122
Chemical Name: 4,9-Dihydro-3-methyl-4-[(4-methyl-1
Biological ActivitySelective high affinity muscarinic M1 receptor antagonist (Ki = 0.94 nM). Inhibits gastric acid secretion.
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Certificate of Analysis / Product Datasheet / Safety Datasheet
References are publications that support the products' biological activity.
Christofi et al (1991) Neuropharmacology of the muscarinic antagonist telenzepine in myenteric ganglia of the guinea-pig small intestine. Eur.J.Pharmacol. 195 333. PMID: 1868879.
Galvan et al (1989) Interaction of telenzepine with muscarinic receptors in mammalian sympathetic ganglia. Eur.J.Pharmacol. 167 1. PMID: 2776837.
Eltze et al (1985) Pharmacological evidence for selective inhibition of gastric acid secretion by telenzepine, a new antimuscarinic drug. Eur.J.Pharmacol. 112 211. PMID: 4029260.
If you know of a relevant reference for Telenzepine dihydrochloride please let us know.
Citations are publications that use Tocris products. Selected citations for Telenzepine dihydrochloride include:
Pediani et al (2016) Dynamic regulation of quaternary organization of the M1 muscarinic receptor by subtype-selective antagonist drugs. J.Biol.Chem. 291 13132. PMID: 27080256.
Do you know of a great paper that uses Telenzepine dihydrochloride from Tocris? If so please let us know.
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Keywords: Telenzepine dihydrochloride, supplier, Potent, selective, M1, antagonists, Muscarinic, Receptors, Acetylcholine, ACh, Tocris Bioscience, M1 Receptor Antagonist products
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May 17 - 19, 2017