Cat. No. 3247
Alternative Name: Phentanyl citrate
Chemical Name: N-Phenyl-N-[1-(2-phenylethyl)-4-pip
Biological ActivityPotent and selective μ-opioid receptor agonist (Ki values are 7.0, 151 and 470 nM for μ-, δ- and κ-opioid receptors respectively). Displays antinociceptive activity in vivo.
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Certificate of Analysis / Safety Data Sheet
Liu et al (2003) Opioid activity of C8813, a novel and potent opioid analgesic. Life Sci. 73 233. PMID: 12738037.
Stevenson et al (2003) Opioid interactions in rhesus monkeys: effects of δ + μ and δ + κ agonists on schedule-controlled responding and thermal nociception. J.Pharmacol.Exp.Ther. 307 1054. PMID: 14557380.
Zernig et al (1995) Receptor reserve and affinity of mu-opioid agonists in mouse antinociception: correlation with receptor binding. Life Sci. 57 2113. PMID: 7475964.
If you know of a relevant reference for this product please let us know.
Citations are publications that use Tocris products.
Do you know of a great paper that uses Fentanyl citrate from Tocris? If so please let us know.
View Related Products by Target
View Related Products by Product Action
Keywords: Fentanyl citrate, supplier, Potent, selective, μ-opioid, mu-opioid, agonists, MOP, Receptors, OP3, Tocris Bioscience, μ Opioid Receptor Agonist products
Find multiple products by catalog number
Follow @Tocris on Twitter
Tocris is now actively tweeting. For regular updates on news, events and special offers, follow @Tocris on Twitter.