Fentanyl citrate

Cat. No. 3247

Fentanyl citrate C22H28N2O.C6H8O7 [990-73-8]

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Alternative Name: Phentanyl citrate

Chemical Name: N-Phenyl-N-[1-(2-phenylethyl)-4-piperidinyl]propanamide citrate

Biological Activity

Potent and selective μ-opioid receptor agonist (Ki values are 7.0, 151 and 470 nM for μ-, δ- and κ-opioid receptors respectively). Displays antinociceptive activity in vivo.

Technical Data

M.Wt:
528.59
Formula:
C22H28N2O.C6H8O7
Solubility:
Soluble to 40 mM in water
Purity:
>99 %
Storage:
Store at RT
CAS No:
990-73-8

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.

Certificate of Analysis / Safety Data Sheet

Certificate of Analysis: View current batch
Safety Data Sheet: View Safety Data Sheet

Liu et al (2003) Opioid activity of C8813, a novel and potent opioid analgesic. Life Sci. 73 233. PMID: 12738037.

Stevenson et al (2003) Opioid interactions in rhesus monkeys: effects of δ + μ and δ + κ agonists on schedule-controlled responding and thermal nociception. J.Pharmacol.Exp.Ther. 307 1054. PMID: 14557380.

Zernig et al (1995) Receptor reserve and affinity of mu-opioid agonists in mouse antinociception: correlation with receptor binding. Life Sci. 57 2113. PMID: 7475964.

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Keywords: Fentanyl citrate, supplier, Potent, selective, μ-opioid, mu-opioid, agonists, MOP, Receptors, OP3, Tocris Bioscience, μ Opioid Receptor Agonist products

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