Cat. No. 3247
Alternative Name: Phentanyl citrate
Chemical Name: N-Phenyl-N-[1-(2-phenylethyl)-4-pip
Biological ActivityPotent and selective μ-opioid receptor agonist (Ki values are 7.0, 151 and 470 nM for μ-, δ- and κ-opioid receptors respectively). Displays antinociceptive activity in vivo.
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Certificate of Analysis / Product Datasheet / Safety Datasheet
References are publications that support the products' biological activity.
Liu et al (2003) Opioid activity of C8813, a novel and potent opioid analgesic. Life Sci. 73 233. PMID: 12738037.
Stevenson et al (2003) Opioid interactions in rhesus monkeys: effects of δ + μ and δ + κ agonists on schedule-controlled responding and thermal nociception. J.Pharmacol.Exp.Ther. 307 1054. PMID: 14557380.
Zernig et al (1995) Receptor reserve and affinity of mu-opioid agonists in mouse antinociception: correlation with receptor binding. Life Sci. 57 2113. PMID: 7475964.
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Keywords: Fentanyl citrate, supplier, Potent, selective, μ-opioid, mu-opioid, agonists, MOP, Receptors, OP3, Tocris Bioscience, μ Opioid Receptor Agonist products
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August 20 - 24, 2017
Paris , France