Cat. No. 3199
Chemical Name: 8-[4-[4-(4-Chlorobenzyl)piperazide-
Biological ActivityPotent and selective adenosine A2B receptor antagonist (IC50 = 3.64 nM at human A2B receptors). Displays > 100-fold selectivity over hA1, hA2A and hA3 receptors.
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Certificate of Analysis / Safety Data Sheet
Borrmann et al (2009) 1-alkyl-8-(piperazine-1-sulfonyl)phenylxanthines: development and characterization of adenosine A2B receptor antagonists and a new radioligand with subnanomolar affinity and subtype specificity. J.Med.Chem. 52 3994. PMID: 19569717.
If you know of a relevant reference for this product please let us know.
Citations are publications that use Tocris products.
Do you know of a great paper that uses PSB 0788 from Tocris? If so please let us know.
View Related Products by Target
View Related Products by Product Action
Keywords: PSB 0788, supplier, Selective, A2B, antagonists, Receptors, adenosines, PSB0788, Tocris Bioscience, A2B Receptor Antagonist products
Find multiple products by catalog number
New Products in this Area
Potent and selective A1 antagonist/inverse agonist
Follow @Tocris on Twitter
Tocris is now actively tweeting. For regular updates on news, events and special offers, follow @Tocris on Twitter.