Cat. No. 3199
Chemical Name: 8-[4-[4-(4-Chlorobenzyl)piperazide-
Biological ActivityPotent and selective adenosine A2B receptor antagonist (IC50 = 3.64 nM at human A2B receptors). Displays > 100-fold selectivity over hA1, hA2A and hA3 receptors.
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Certificate of Analysis / Product Datasheet / Safety Datasheet
References are publications that support the products' biological activity.
Borrmann et al (2009) 1-alkyl-8-(piperazine-1-sulfonyl)phenylxanthines: development and characterization of adenosine A2B receptor antagonists and a new radioligand with subnanomolar affinity and subtype specificity. J.Med.Chem. 52 3994. PMID: 19569717.
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Keywords: PSB 0788, supplier, Selective, A2B, antagonists, Receptors, adenosines, PSB0788, Tocris Bioscience, Adenosine A2B Receptor Antagonist products
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