BAY-u 9773

Cat. No. 3138

BAY-u 9773 C27H36O5S [154978-38-8]

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Chemical Name: 4-[[(1R,2E,4E,6Z,9Z)-1-[(1S)-4-Carboxy-1-hydroxybutyl]-2,4,6,9-pentadecatetraen-1-yl]thio]benzoic acid

Biological Activity

Cysteinyl leukotriene receptor antagonist with equal affinity at both CysLT1 and CysLT2 receptors (pKB values are 6.8 and 6.5 respectively). Competitive antagonist of LTC4- and LTE4-induced contractions of the guinea pig trachea.

Technical Data

M.Wt:
472.64
Formula:
C27H36O5S
Solubility:
Soluble in ethanol (supplied pre-dissolved in Ethanol, 0.1mg/ml)
Storage:
Store at -80°C
CAS No:
154978-38-8

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.

Certificate of Analysis / Product Datasheet / Safety Datasheet

Back (2002) Functional characteristics of cysteinyl-leukotriene receptor subtypes. Life Sci. 71 611. PMID: 12072150.

Goranne et al (1996) Cysteinyl leukotriene receptors in the human lung: what's new? TiPS 17 342. PMID: 8979767.

Labat et al (1992) A second cysteinyl leukotriene receptor in human lung. J.Pharmacol.Exp.Ther. 263 800. PMID: 1331415.

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Keywords: BAY-u 9773, supplier, Dual, CysLT1, CysLT2, antagonists, Receptors, leukotrienes, eicosanoids, BAY-u9773, Tocris Bioscience, Leukotriene and Related Receptor Antagonist products

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