Cat. No. 3116
Chemical Name: 7-Nitro-5-(trifluoromethyl)-2-benzo
Biological ActivitySelective, ATP-competitive polo-like kinase 1 (PLK1) inhibitor (IC50 = 500 nM).
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Certificate of Analysis / Product Datasheet / Safety Data Sheet
Taylor et al (2008) Ligand discovery and virtual screening using the program LIDAEUS. Br.J.Pharmacol. 153 S55. PMID: 18037921.
McInnes et al (2006) Inhibitors of polo-like kinase reveal roles in spindle pole maintenance. Nature Chem.Biol. 2 608.
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Citations are publications that use Tocris products. Selected citations for Cyclapolin 9 include:
Cozzoli et al (2012) Nucleus accumbens mGluR5-associated signaling regulates binge alcohol drinking under drinking-in-the-dark procedures. Proc Natl Acad Sci U S A 36 1623. PMID: 22432643.
Do you know of a great paper that uses Cyclapolin 9 from Tocris? If so please let us know.
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Keywords: Cyclapolin 9, supplier, Selective, ATP-competitive, PLK1, inhibitors, inhibits, Polo-like, Kinase, Kinases, Cyclapolin9, Tocris Bioscience, Polo-like Kinase Inhibitor products
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