BRL 52537 hydrochloride
Cat. No. 0699
Chemical Name: (±)-1-(3,4-Dichlorophenyl)acetyl-2-(
Biological ActivityThe most κ/μ-selective and among the most potent κ ligands known (25 times more potent than morphine in vivo).
Licensing InformationSold with the permission of GlaxoSmithKline
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Certificate of Analysis / Product Datasheet / Safety Data Sheet
Vecchietti et al (1991) (2S)-1-(Arylacetyl)-2-(aminomethyl)piperidine derivatives: novel, highly selective κ opioid analgesics. J.Med.Chem. 34 397. PMID: 1846921.
If you know of a relevant reference for this product please let us know.
Citations are publications that use Tocris products.
Do you know of a great paper that uses BRL 52537 hydrochloride from Tocris? If so please let us know.
View Related Products by Target
View Related Products by Product Action
Keywords: BRL 52537 hydrochloride, supplier, Potent, selective, κ-opioid, kappa-opioid, agonist, agonists, KOP, Receptors, OP2, BRL52537, hydrochloride, GlaxoSmithKline, GSK, Tocris Bioscience, κ Opioid Receptor Agonist products
Find multiple products by catalog number
New Products in this Area
Fluorescent opioid antagonist; fluorescent-derivative of naloxone (Cat. No. 0599)BMS 986187
Potent δ-opioid receptor positive allosteric modulator
April 10 - 13, 2017