BRL 52537 hydrochloride
Cat. No. 0699
Chemical Name: (±)-1-(3,4-Dichlorophenyl)acetyl-2-(
Biological ActivityThe most κ/μ-selective and among the most potent κ ligands known (25 times more potent than morphine in vivo).
Licensing InformationSold with the permission of GlaxoSmithKline
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Certificate of Analysis / Product Datasheet / Safety Data Sheet
Vecchietti et al (1991) (2S)-1-(Arylacetyl)-2-(aminomethyl)piperidine derivatives: novel, highly selective κ opioid analgesics. J.Med.Chem. 34 397. PMID: 1846921.
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