SDM25N hydrochloride

Cat. No. 1410

SDM25N hydrochloride C26H26N2O3.HCl [342884-71-3]

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Chemical Name: (4bS,8R,8aS,14bR)-5,6,7,8,14,14b-Hexahydro-7-(2-methyl-2-propenyl)-4,8-methanobenzofuro[2,3-a]pyrido[4,3-b]carbazole-1,8a(9H)-diol hydrochloride

Biological Activity

Potent and highly selective non-peptide δ receptor antagonist (Ki values are 4.7, 3800 and 7900 nM for δ, κ and μ receptors respectively). More selective than naltrindole (Cat. No. 0740).

Technical Data

M.Wt:
450.96
Formula:
C26H26N2O3.HCl
Solubility:
Soluble to 10 mM in water and to 100 mM in DMSO
Purity:
>99 %
Storage:
Store at +4°C
CAS No:
342884-71-3

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.

Certificate of Analysis / Safety Data Sheet

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McLamore et al (2001) Effect of N-alkyl and N-alkenyl substituents in noroxymorphindole, 17-substituted-6,7-dehydro-4,5α-epoxy-3,14-dihydroxy-6,7:2 ',3 '-indolomorphinans, on opioid receptor affinity, selectivity, and efficacy. J.Med.Chem. 44 1471. PMID: 11311071.

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Keywords: SDM25N hydrochloride, supplier, Potent, selective, non-peptide, δ-opioid, delta-opioid, antagonist, DOP, Receptors, OP1, Tocris Bioscience, δ Opioid Receptor Antagonist products

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