Cat. No. 3021
Chemical Name: 2-[(2E)-3,7-Dimethyl-2,6-octadienyl
Biological ActivityPartial agonist of CB2 and CB1 receptors (Ki values are 337 and 440 nM respectively). Also exhibits α2-adrenoceptor agonist activity (EC50 = 0.2 nM in mouse brain membranes).
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Certificate of Analysis / Product Datasheet / Safety Datasheet
References are publications that support the products' biological activity.
Cascio et al (2010) Evidence that the plant cannabinoid cannabigerol is a highly potent α2-adrenoceptor agonist and moderately potent 5HT1A receptor antagonist. Br.J.Pharmacol. 159 129. PMID: 20002104.
Gauson et al (2007) Cannabigerol behaves as a partial agonist at both CB1 and CB2 receptors. Symposium on the Cannabinoids 206.
Pertwee The diverse CB1 and CB2 receptor pharmacology of three plant cannabinoids: Δ9-tetrahydrocannabinol, cannabidiol and Δ9-tetrahydrocannabivarin. Br.J.Pharmacol. 153 199. PMID: 17828291.
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Citations are publications that use Tocris products.
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Keywords: Cannabigerol, supplier, phytocannabinoids, cbg, cannabigerol, cb1, cb2, partial, agonists, alpha2, α2, a2-adrenoceptors, adrenergics, receptors, agonists, Tocris Bioscience, Non-selective Cannabinoid Agonist products