Diprenorphine

Cat. No. 2965

Diprenorphine C26H35NO4 [14357-78-9]

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Chemical Name: 17-(Cyclopropylmethyl)-4,5-epoxy-18,19-dihydro-3-hydroxy-6-methoxy-α,α-dimethyl-6,14-ethenomorphinan-7-methanol

Biological Activity

Non-selective opioid receptor antagonist (Ki values are 0.017, 0.072 and 0.23 nM for κ-, μ- and δ-opioid receptors).

Technical Data

M.Wt:
425.56
Formula:
C26H35NO4
Solubility:
Soluble to 20 mM in DMSO and to 25 mM in ethanol
Purity:
>99 %
Storage:
Store at RT
CAS No:
14357-78-9

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.

Certificate of Analysis / Safety Data Sheet

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Iwasaki et al (1994) The effect of the nonselective opioid antagonist diprenorphine vasopressin secretion in the rat. Endocrinology 134 48. PMID: 8275962.

Raynor et al (1994) Pharmacological characterization of the cloned κ-, δ-, and μ-opioid receptors. Mol.Pharmacol. 45 330. PMID: 8114680.

Paterson et al (1983) Classification of opioid receptors. Br.Med.Bull. 39 31. PMID: 6301606.

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Keywords: Diprenorphine, supplier, Non-Selective, opioids, antagonists, Receptors, Tocris Bioscience, Miscellaneous Opioid Antagonist products

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