Cat. No. 2965
Chemical Name: 17-(Cyclopropylmethyl)-4,5-epoxy-18
Biological ActivityNon-selective opioid receptor antagonist (Ki values are 0.017, 0.072 and 0.23 nM for κ-, μ- and δ-opioid receptors).
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Certificate of Analysis / Product Datasheet / Safety Datasheet
References are publications that support the products' biological activity.
Iwasaki et al (1994) The effect of the nonselective opioid antagonist diprenorphine vasopressin secretion in the rat. Endocrinology 134 48. PMID: 8275962.
Raynor et al (1994) Pharmacological characterization of the cloned κ-, δ-, and μ-opioid receptors. Mol.Pharmacol. 45 330. PMID: 8114680.
Paterson et al (1983) Classification of opioid receptors. Br.Med.Bull. 39 31. PMID: 6301606.
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Citations are publications that use Tocris products.
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Keywords: Diprenorphine, supplier, Non-Selective, opioids, antagonists, Receptors, Tocris Bioscience, Miscellaneous Opioid Antagonist products