Zolantidine dimaleate

Cat. No. 1070

Zolantidine dimaleate C22H27N3OS.2C4H4O4 [104076-39-3]

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Chemical Name: N-[3-[3-(1-Piperidinylmethyl)phenoxy]propyl]-2-benzothiazolamine dimaleate

Biological Activity

A potent, selective and brain penetrating H2 receptor antagonist.

Licensing Information

Sold with the permission of GlaxoSmithKline

Technical Data

Soluble to 100 mM in water
Desiccate at +4°C

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.

Certificate of Analysis / Product Datasheet / Safety Datasheet

References are publications that support the products' biological activity.

Coruzzi et al (1996) Cardiac and gastric effects of histamine H2 receptor antagonists: no evidence for a correlation between lipophilicity and receptor affinity. Br.J.Pharmacol. 118 1813. PMID: 8842448.

Coruzzi et al (1994) Activity of the new histamine H2-receptor antagonist zolantidine at cardiac and gastric H2 receptors. Pharmacology 48 69. PMID: 7907797.

Calcutt et al (1988) Zolantidine (SK&F 95282) is a potent selective brain penetrating histamine H2-receptor antagonist. Br.J.Pharmacol. 93 69. PMID: 2894879.

If you know of a relevant reference for Zolantidine dimaleate please let us know.

Citations are publications that use Tocris products. Selected citations for Zolantidine dimaleate include:

Porter et al (2005) Fenobam: a clinically validated nonbenzodiazepine anxiolytic is a potent, selective, and noncompetitive mGlu5 receptor antagonist with inverse agonist activity. J Pharmacol Exp Ther 315 711. PMID: 16040814.

Do you know of a great paper that uses Zolantidine dimaleate from Tocris? If so please let us know.

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Keywords: Zolantidine dimaleate, supplier, Potent, centrally, active, H2, antagonists, Receptors, Histamine, histaminergic, GlaxoSmithKline, GSK, Tocris Bioscience, Histamine H2 Receptor Antagonist products

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