BML-190

Cat. No. 1383

BML-190 C23H23ClN2O4 [2854-32-2]

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Alternative Names: Indomethacin morpholinylamide, IMMA

Chemical Name: 1-(4-Chlorobenzoyl)-5-methoxy-2-methyl-1-[2-(4-morpholinyl)-2-oxoethyl]-1H-indole

Biological Activity

Potent and selective CB2 receptor ligand (Ki values are 435 nM and > 2 μM for CB2 and CB1 respectively).

Technical Data

M.Wt:
426.9
Formula:
C23H23ClN2O4
Solubility:
Soluble to 100 mM in DMSO with gentle warming
Purity:
>99 %
Storage:
Store at RT
CAS No:
2854-32-2

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.

Certificate of Analysis / Safety Data Sheet

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Melck et al (2000) Suppression of nerve growth factor Trk receptors and prolactin receptors by endocannabinoids leads to inhibition of human breast and prostate cancer cell proliferation. Endocrinology 141 118. PMID: 10614630.

Gallant et al (1996) New class of potent ligands for the human peripheral cannabinoid receptor. Bioorg.Med.Chem.Lett. 6 2263.

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Keywords: BML-190, supplier, Potent, selective, CB2, ligands, Cannabinoid, Receptors, cb2r, Tocris Bioscience, CB2 Receptor products

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