ARC 239 dihydrochloride
Cat. No. 0928
Chemical Name: 2-[2-(4-(2-Methoxyphenyl)piperazin-
Biological ActivitySelective α2B adrenoceptor antagonist (pKD values are 8.8, 6.7 and 6.4 at α2B, α2A, and α2D receptors respectively). Also available as part of the α2-Adrenoceptor Tocriset™.
Licensing InformationSold with the permission of Boehringer Ingelheim GmbH
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Certificate of Analysis / Product Datasheet / Safety Data Sheet
Fuder and Selback (1993) Characterisation of sensory neurotransmission and its inhibition via α2B-adrenoceptors and via non-α2 adrenoceptors in rabbit iris. Naunyn Schmiedebergs Arch.Pharmacol. 347 394. PMID: 7685502.
Bylund et al (1988) Alpha-2A and alpha-2B adrenergic subtypes: antagonist binding in tissues and cell lines containing only one subtype. J.Pharmacol.Exp.Ther. 245 600. PMID: 2835476.
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