ROS 234 dioxalate
Cat. No. 2034
Chemical Name: N-[3-(1H-Imidazol-4-yl)propyl]-1H-b
Biological ActivityPotent H3 antagonist (pKB at guinea-pig ileum H3-receptor = 9.46). Limited blood brain barrier permeability (ED50 = 19.12 mg/kg i.p.).
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Certificate of Analysis / Product Datasheet / Safety Datasheet
References are publications that support the products' biological activity.
Mor et al (2004) Synthesis, biological activity, QSAR and QSPR study of 2-aminobenzimidazole derivatives as potent H3-antagonists. Bioorg.Med.Chem.Lett. 12 663.
Ballabeni et al (2002) CNS access of selected H3-antagonists: ex vivo binding study in rats. Inflamm.Res. 51 (Suppl 1) S55. PMID: 12013409.
If you know of a relevant reference for ROS 234 dioxalate please let us know.
Citations are publications that use Tocris products.
Do you know of a great paper that uses ROS 234 dioxalate from Tocris? If so please let us know.
View Related Products by Product Action
Keywords: ROS 234 dioxalate, supplier, Potent, H3, antagonists, Receptors, Histamine, histaminergic, ROS234, dioxalate, Tocris Bioscience, Histamine H3 Receptor Antagonist products
Find multiple products by catalog number
Follow @Tocris on Twitter
Tocris is now actively tweeting. For regular updates on news, events and special offers, follow @Tocris on Twitter.