G Protein (Heterotrimeric) Inhibitors

Cat No Product Name / Activity
2974 CCG 2046
Inhibitor of regulator of G-protein signaling 4 (RGS4)
4567 CCG 50014
Potent and selective inhibitor of regulator of G-protein signaling 4 (RGS4) protein
4028 CCG 63802
Inhibitor of regulator of G-protein signaling 4 (RGS4) protein
5642 CMPD101
Potent and selective GRK2/3 inhibitor
4773 ESI 09
EPAC inhibitor
1931 G-Protein antagonist peptide
Inhibits G protein activation by GPCRs
3090 Gallein
Inhibitor of βγ signaling
3594 GRK2i
GRK2 inhibitory polypeptide. Gβγ antagonist
4742 Gue 1654
Selective inhibitor of OXE-R Gβγ signaling
1240 NF 023
Inhibitor of Go/i α-subunits; also P2X1 purinoceptor antagonist
1400 SCH 202676 hydrobromide
Inhibitor of ligand binding to G-protein-coupled receptors
1884 [D-Trp7,9,10]-Substance P
Inhibits M1 ACh receptor activation of Gq/11