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Displaying products by catalog number (5900 - 5999)

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Cat.No.
Product Name / Activity
5900c-Di-GMP sodium salt

Endogenous STING and DDX41 agonist; activates STING-dependent signaling

5901c-Di-AMP sodium salt

Endogenous STING and DDX41 agonist; activates STING-dependent signaling

5902Tiotropium bromide

Potent muscarinic receptor antagonist

5903CATPB

FFA2 antagonist/inverse agonist

5904Montelukast sodium

CysLT1 and GPR17 antagonist

5905Neurosensor 521

Selective noradrenalin and dopamine fluorescent indicator

5906Imatinib mesylate

Potent and selective v-Abl tyrosine kinase inhibitor; also inhibits PDGFR and c-kit

5907VX 680

High affinity and selective Aurora kinase inhibitor

5908Bis-ANS

Fluorescent probe for nonpolar cavities in proteins; used to detect Aβ fibres

5909RMM 46

MSK/RSK family kinase inhibitor

5911FFN 200 dihydrochloride

Selective fluorescent VMAT2 substrate

5913Ro 6842262

Potent LPA1 antagonist

5915PF 04449613

Potent PDE9 inhibitor; brain penetrant

5916Canertinib dihydrochloride

Potent EGFR kinase inhibitor

5917PF 9184

Potent microsomal prostaglandin E synthase 1 (mPGES-1) inhibitor

5918TPPU

Potent soluble epoxide hydrolase inhibitor; orally bioavailable and brain penetrant

5919PI 3065

Potent and selective PI 3-kinase p110δ inhibitor

5921D9

Potent thioredoxin reductase (TxrR) inhibitor

5928RS 09

TLR4 peptide agonist; acts as an adjuvant in vivo

5929BeKm 1

Potent and selective KV11.1 (hERG) channel blocker

5930PBIT

JARID1 (Jumonji AT-Rich Interactive Domain 1) inhibitor

5931PF 05089771

Potent and selective Nav1.7 channel blocker

5932Tocriscreen Library of FDA-Approved Compounds

A library of 160 FDA-approved compounds (250 μL 10 mM DMSO solutions)

5933Tocriscreen Kinase Inhibitor Toolbox I

A library of 80 kinase inhibitor compounds (250 μL 10 mM DMSO solutions)

5934NCT 501 hydrochloride

Potent and selective ALDH1A1 inhibitor

5935H2DCFDA

Fluorescent ROS indicator; cell permeable

5937A 779

Selective Mas receptor (Ang-(1-7) receptor) antagonist

5938Mambalgin 1

Selective ASIC1a inhibitor; analgesic

5939PF 6274484

High affinity and potent covalent EGFR kinase inhibitor

5940AdTx1

Selective, high affinity, non-competitive α1A adrenoceptor antagonist

5941OD1

Potent hNav1.4, rNav1.6 and rNav1.7 channel activator

5943ML 339

Potent and selective hCXCR6 antagonist

5944G10

Activator of STING-dependent signaling

59452',3'-cGAMP sodium salt

Endogenous high affinity STING agonist

59463',3'-cGAMP sodium salt

STING agonist

5951WAY 252623

Potent LXR agonist

5952PDD 00017273

Potent and selective poly (ADP ribose) glycohydrolase (PARG) inhibitor; cell permeable

5953Adaptaquin

HIF-prolyl hydroxylase-2 (PHD2) inhibitor; antioxidant

5954MSG 606

Potent human MC1 receptor antagonist; also MC3 and MC5 partial agonist

5955eCF 309

Potent mTOR inhibitor

5958Desloratadine

High affinity H1 antagonist; anti-inflammatory.

5959Autocamtide-2-related inhibitory peptide, myristoylated

CaM kinase II inhibitor; enhanced cell permeable derivative of Autocamtide-2-related inhibitory peptide

5960TMI 1

Adam 17 (TACE) and MMP inhibitor; orally bioavailable

5961HIOC

Selective TrkB receptor agonist; neuroprotectant

59623-AP

Ribonucleotide reductase inhibitor; also an iron chelator

5963CMPI hydrochloride

Potent positive allosteric modulator of α4β2 nAChRs; also inhibitor of (α4)2(β2)3, muscle-type and Torpedo nAChRs

5964SI-2 hydrochloride

Steroid receptor coactivator 3 (SRC-3) inhibitor

5965ISAM 140

High affinity A2B receptor antagonist

5966ML 233

Non-peptide apelin receptor agonist

5968Ro 3280

Potent and selective PLK1 inhibitor

5970BAY 299

Potent and selective BRD1 and TAF1 inhibitor

5973CP 724714

Potent and selective ErbB2 inhibitor

5976Ned K

NAADP signaling inhibitor

5978WL 47 - dimer

High affinity caveolin-1 ligand

5979Eicosapentaenoic Acid

Endogenous polyunsaturated fatty acid; stimulates ERK1/2 phosphorylation

5981Itraconazole

SMO antagonist; acts at different binding site to cyclopamine (Cat No. 1623)

5982cis-6-Hydroxynorketamine hydrochloride

Enhances AMPA currents: antidepressant

5983BMS 986187

Potent δ-opioid receptor positive allosteric modulator

5986NAV 2729

Selective ARF6 inhibitor

5987(±)-ML 209

RORγt inverse agonist; suppresses Th17 cell differentiation

5989BIRB 796

High affinity and selective p38 kinase inhibitor

5992MM 54

Potent apelin receptor antagonist

5993CP 673451

Potent and selective PDGFR inhibitor

5994Enzastaurin

Potent PKCβ inhibitor

5995AMG 517

Potent TRPV1 antagonist

5996(R)-Norketamine hydrochloride

NMDA receptor modulator; analgesic

5999TP 472N

Negative control for TP 472 (Cat. No. 6000).

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