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Displaying products by catalog number (5600 - 5699)

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Product Name / Activity
5600BA 1

Potent BRS-3 agonist; also NMBR and GRPR agonist


mSTING agonist; induces antitumor immunological responses


CD40-TRAF6 interaction inhibitor


Inactive control for (+)-JQ1 (Cat. No. 4499)

5604MI 14

Potent and selective PI 4-kinase IIIβ inhibitor

5605CINPA 1

Potent CAR antagonist


High affinity protein disulfide isomerase (PDI) modulator

5607GNF 7

Ras signaling inhibitor; inhibits Ack1 and GCK

5608BS 181 dihydrochloride

Selective cdk7 inhibitor


Mimic of GFP fluorophore for imaging RNA in living cells

5610DFHBI 1T

Mimic of GFP fluorophore for imaging RNA in living cells

5611Salvinorin B

Activates the κ-opioid DREADD (KORD)


HIV cell entry blocker

5613AZD 9272

Potent and selective mGlu5 antagonist; brain penetrant

5614AZD 2066

mGlu5 antagonist; orally bioavailable and brain penetrant

5615AZD 3147

Potent and selective dual mTORC1 and 2 inhibitor; orally bioavailable

5617AZD 1480

Potent and selective JAK2 inhibitor; antiangiogenic

5619N-Acetylcysteine amide

Glutathione (GSH) precursor; neuroprotective

5620BDY FL-X, SE

Fluorescent reagent for the labeling of amines

5621GLPG 0974

Potent FFA2 antagonist

5622HTH 01-015

Potent and selective NUAK1 inhibitor

5625ML 334

Inhibitor of Keap1- Nrf2 interaction

5626SR 7826

Potent and selective LIMK inhibitor; antitumor

5627HFI 142

Insulin-regulated aminopeptidase (IRAP) inhibitor

5629Dolasetron mesylate

Potent and selective 5-HT3 antagonist

5630(Z-LL)2 ketone

Putative inhibitor of signal peptide peptidase

5631LDN 193188

Inhibitor of phosphatidylcholine transfer protein (PC-TP)

5632AZ Dyrk1B 33

Potent and selective Dyrk1B kinase inhibitor

5633MRS 2905

Potent and selective P2Y14 receptor agonist

5635GSK 2801

Selective BAZ2A and BAZ2B inhibitor

5636GS 143

β-TrCP1 ligase inhibitor


Oct3/4 inducer

5640PF 06463922

High affinity and selective ALK and ROS1 inhibitor

5641MSC 2032964A

Potent and selective ASK1 inhibitor; orally bioavailable


Potent and selective GRK2/3 inhibitor


OX2 receptor antagonist; orally bioavailable

5646EML 425

Reversible and non-competitive p300/CBP inhibitor

5647MI 192

Potent and selective HDAC2/3 inhibitor

5648Hydroxychloroquine sulfate

Autophagy inhibitor; also TLR9 inhibitor

5650SAR 216471 hydrochloride

Potent P2Y12 antagonist; orally available

5651ONO 6818

High affinity and selective human neutrophil elastase 1 (HNE1) inhibitor; orally active

5653JW 74

Wnt pathway inhibitor

5654BMS 265246

Potent cdk1/2 inhibitor

5655GN 44028

Potent HIF-1α inhibitor

5656DY 268

Potent FXR antagonist


KV4 channel blocker

5660NVP CXCR2 20

Potent and selective CXCR2 antagonist


Potent and selective CREB inhibitor


Oct3/4 inducer; induces expression of pluripotent-associated genes

5665IRAK1/4 Inhibitor I

IRAK4 and IRAK1 inhibitor

5666JNJ 63533054

Potent and selective GPR139 agonist

5667YK 3-237

SIRT1 activator

5668VUF 11222

High affinity non-peptide CXCR3 agonist

5671SB 332235

Potent CXCR2 antagonist

5672GSK 319347A

Potent and selective IKKε inhibitor

5673GW 2580

Selective cFMS kinase inhibitor; orally bioavailable

5674GW 501516

Potent and selective PPARδ agonist

5675AZ PFKFB3 26

Potent and selective PFKFB3 inhibitor

5676Guangxitoxin 1E

Potent Kv2.1 and Kv2.2 channel blocker

5677RFRP-1 (human)

Potent NPFF receptor agonist

5678RN 9893 hydrochloride

Potent and selective TRPV4 antagonist


Downregulates SnoN and Ski protein expression; promotes TGF-β signaling

5680Vatalanib succinate

Potent VEGFR inhibitor; also aromatase inhibitor


Activator of SUMO-activating enzyme, E1 ligase

5682OSU 03012

PDPK1 (PDK1) inhibitor; inhibits Akt signaling


Potent dolastatin 10 analog; antitumor

5684Naloxone 3-glucuronide carbonic acid salt

Naloxone conjugate

5685MS049 oxalate salt

Potent and selective PRMT4 and PRMT6 inhibitor


High affinity and selective PLK4 inhibitor

5690Centrinone B

High affinity and selective PLK4 inhibitor

5692ITH 12575

Mitochondrial Na+/Ca2+ exchange (mNCX) inhibitor.

5693VU 0409551

Selective mGlu5 positive allosteric modulator; brain penetrant and orally bioavailable

5694GSK 2033

Potent LXR antagonist


Potent and selective PDE4 inhibitor; suppresses hedgehog signaling

5697PMX 53c

Negative control for PMX 53 (Cat. No. 5473)


Indoleamine 2,3-dioxygenase (IDO) inhibitor


Potent Nurr1 activator

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