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Displaying products by catalog number (5300 - 5399)

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Cat.No.
Product Name / Activity
5301BPTES

Selective allosteric glutaminase (GLS1) inhibitor

5303GSK 2194069

Potent human fatty acid synthase (hFASN) inhibitor

5304FICZ

High affinity aryl hydrocarbon receptor (AhR) agonist

5305Verteporfin

YAP inhibitor; disrupts YAP-TEAD interactions

5306KJ Pyr 9

High affinity Myc inhibitor

5307MM 102

WDR5/MLL interaction inhibitor

5308ASP 2535

Potent and selective GlyT1 inhibitor

5309SP 100030

NF-κB and AP-1 dual inhibitor

5310ASP 3026

Potent anaplastic lymphoma kinase (ALK) inhibitor; also potent ACK inhibitor

5311RHPS 4 methosulfate

Telomerase inhibitor

5313LY 315920

Selective secreted phospholipase A2 (sPLA2) inhibitor

5314SMBA 1

High affinity and selective activator of Bax

5315Rostafuroxin

Na+/K+ ATPase modulator; antihypertensive agent

5316Elinogrel

P2Y12 antagonist

5317WWL 123

α/β-hydrolase domain 6 (ABHD6) inhibitor; antiepileptic

5318AEE 788

Potent EGFR and VEGFR inhibitor

5319ACT 462206

Potent, dual orexin receptor antagonist

5320CORM 3

Water-soluble carbon monoxide-releasing molecule

5321PSNCBAM-1

CB1 receptor negative allosteric modulator

5322VU 0409106

Potent and selective negative allosteric modulator at mGlu5

5323WDR5 0103

WDR5 antagonist

5324M8 B hydrochloride

Potent and selective TRPM8 channel blocker

5325Rosiglitazone

Potent and selective PPARγ agonist; antidiabetic agent.

5326CHR 6494 trifluoroacetate

Potent and selective haspin inhibitor

5327BGC 20-1531 hydrochloride

High affinity and selective EP4 antagonist

5328TY 52156

S1P3 receptor antagonist

5329CKI 7 dihydrochloride

CK1 inhibitor

5330AEG 40730 dihydrochloride

IAP antagonist; induces apoptosis

5331CPI 203

BET bromodomain inhibitor; arrests cell cycle at G1 phase

5332SP 141

High affinity MDM2 inhibitor

5335Angiotensin A

Potent endogenous vasoconstrictor peptide - derivative of angiotensin II (Cat. No. 1158)

5336BRD 7116

Inhibitor of leukemia stem cell activity

5337ML 365

Potent and selective TASK-1 channel blocker

5338PK-THPP

Potent TASK-3 channel blocker

5339PFK 15

Selective PFKFB3 inhibitor

5340NSC 617145

Werner syndrome helicase (WRN) inhibitor

5342SCR7 pyrazine

Enhances HDR efficiency

5344ML 349

Selective and reversible lysophospholipase 2 (LYPLA2) inhibitor

5345ML 348

Selective and reversible lysophospholipase 1 (LYPLA1) inhibitor

5347Kisspeptin 10 (dog)

Endogenous ligand for canine kisspeptin receptor

5348CPI 613

PDH and KGDH inhibitor

5349Treprostinil

Potent prostacyclin (PGI2) analog

5351PQ 69

Potent and selective A1 antagonist/inverse agonist

5353Gap19

Cx43 hemichannel blocker

5355TC-G 1008

Potent and selective GPR39 agonist

5356SGX 523

Selective and potent c-MET kinase inhibitor

5357DC 260126

FFA1 (GPR40) antagonist

5358Cariporide

Selective NHE1 inhibitor; cardioprotective and antitumor

5359Rifaximin

Pregnane X receptor agonist; antibiotic

5361GSK LSD 1 dihydrochloride

Potent and selective LSD1 inhibitor

5363NHI 2

LDHA inhibitor

5364Hydroxy Dynasore

Dynamin inhibitor; analog of dynasore (Cat. No. 2897)

5365LLY 507

Potent SMYD2 inhibitor

5367SGC 707

Potent and selective allosteric inhibitor of PRMT3

5368Maritoclax

Mcl-1 inhibitor; proapoptotic

5369Norleual

Highly potent HGF/c-MET inhibitor; also AT4 antagonist

5371Clemizole hydrochloride

TRPC5 blocker; also H1 antagonist

5373C34

TLR4 inhibitor

5374GLP-1 (7-37)

Endogenous bioactive GLP-1 receptor ligand

5375BIX

BiP (Hsp70-5) ER chaperone inducer

5376Pregnenolone sulfate sodium salt

NMDA Potentiator

5377VU 0483605

Positive allosteric modulator at mGlu1

5378VU 0422288

Selective group III mGlu positive allosteric modulator

5379VU 0469650 hydrochloride

Potent and selective negative allosteric modulator of mGlu1

5380ML 297

Selective Kir3.1/3.2 (GIRK1/2) channel activator

5382C16

PKR inhibitor

5383TA 01

Induces cardiomyocyte differentiation from hESCs

5384TA 02

Induces cardiomyocyte differentiation from hESCs

5385GSK 5959

Potent and selective BRPF1 inhibitor

5387ML 354

Selective PAR4 antagonist

5388RQ 00203078

Potent and selective TRPM8 antagonist; orally active

5389Ro 48-8071 fumarate

2,3-Oxidosqualene cyclase (OSC) inhibitor; blocks cholesterol synthesis

5390Tobramycin

Aminoglycoside antibiotic

5391SPP 86

Potent RET inhibitor

5393ERK5-IN-1

Potent and selective ERK5 inhibitor

5395Virodhamine trifluoroacetate

TFA salt of virodhamine, an endogenous cannabinoid receptor mixed agonist/antagonist

5397A01

High affinity Smurf1 inhibitor; enhances BMP signaling

5398NQTrp

Potent inhibitor of Aβ oligomer and fibril formation

5399BTB1

Selective and ATP-competitive Kif18A inhibitor

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