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Displaying products by catalog number (5100 - 5199)

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Product Name / Activity
5100TC-T 6000

Potent equilibrative nucleoside transporter 4 (ENT4) inhibitor

5101PD 90780

Inhibits NGF binding to p75NTR

5102PLX 647 dihydrochloride

Potent dual Fms/KIT inhibitor


Selective p300 inhibitor

5106GSK 2193874

Potent and selective TRPV4 antagonist; orally active

5107GSK 2606414

Potent and selective PERK inhibitor; orally bioavailable

5108TFC 007

Potent hematopoietic prostaglandin D synthase (H-PGDS) inhibitor

5109SB 743921 hydrochloride

Potent kinesin spindle protein (KSP) inhibitor

5110GSK 1562590 hydrochloride

High affinity, selective urotensin II (UT) receptor antagonist

5111GSK 1838705

Potent IR and IGF1R inhibitor; also inhibits anaplastic lymphoma kinase (ALK)

5112NS 9283

Positive allosteric modulator of α4β2


Photo-crosslinking probe

5115OXA (17-33)

Potent and selective peptide OX1 agonist

5116PACMA 31

Irreversible protein disulfide isomerase (PDI) inhibitor

5117Hoechst 33342

Fluorescent dye for labeling DNA

5118SynaptoRedTM C2

Fluorescent dye; stains synaptic vesicles

5119Calcein AM

Cell permeable compound; hydrolyzed to become fluorescent in living cells


PFKFB3 inhibitor


Potent and selective fluorescent adenosine A1 agonist

5124PD 404182

High affinity inhibitor of KDO 8-P synthase; also DDAH1 inhibitor

5125CKD 602

Topoisomerase I inhibitor


Suppressor of MDK expression; inhibits PI 3-K signaling


Protein disulfide isomerase (PDI) inhibitor

5128C 21

Selective PRMT1 inhibitor

5129TC-G 1005

Potent and selective GPBA receptor (TGR5) agonist

5130CTCE 9908

CXCR4 antagonist; antitumor

5131NAB 2

Protects against α-synuclein toxicity; promotes Rsp5/Nedd4-dependent endosomal transport

5132UNC 0642

Potent and selective G9a and GLP inhibitor

5133GKA 50

Glucokinase activator

5134MRT 67307 dihydrochloride

Salt inducible kinase (SIK) inhibitor

5135Propidium iodide

Red-fluorescent DNA stain; membrane impermeant to live cells

5136Rizatriptan benzoate

Potent 5-HT1B/1D agonist

5138RSVA 405

AMPK activator; also STAT3 inhibitor


AT1 antagonist; PPARγ partial agonist

5140GSK 2830371

Potent and selective allosteric inhibitor of Wip1 phosphatase

5141AZD 5582 dihydrochloride

Dimeric Smac mimetic; potent IAP inhibitor

5142Mps1-IN-1 dihydrochloride

Selective Mps1 kinase inhibitor


TRPM3 blocker

5144CFM 4

CARP-1 mimetic; proapoptotic


ARE activator; induces Nrf2-ARE-dependent transcription

5146Sulforhodamine 101

Fluorescent dye; selective astrocyte marker


Potent and selective adenosine A2A receptor antagonist


Highly potent PORCN inhibitor

5149CX 614

AMPAkine; positive allosteric modulator of AMPA

5150NCL 00017509

Potent and reversible NIMA related kinase 2 (Nek2) inhibitor

5151Prosaptide TX14(A)

Potent GPR37 and GPR37L1 agonist

5153ML 240

ATP-competitive inhibitor of p97 ATPase


Humanin analog; increases insulin sensitivity

5155SGI 1027

DNA methyltransferase inhibitor

5156Ivermectin B1a-d2

Deuterated ivermectin B1a (Cat. No. 1260)

5157DMNPE-caged ATP diammonium salt

Caged ATP

5158Morphine hydrochloride

Narcotic opioid analgesic

5160Medetomidine hydrochloride

Potent, highly selective α2 agonist

5161ML 154

Potent neuropeptide S receptor (NPSR) antagonist

5163A 366

Potent and selective G9a/GLP inhibitor

5164CVT 10216

Potent and selective ALDH2 inhibitor

5166Perhexiline maleate

Carnitine palmitoyltransferase 1 and 2 (CPT1/2) inhibitor

5167Congo Red

Amyloid fibril binding dye; also a VGlut inhibitor

5168Rose Bengal

Potent VGlut and VMAT inhibitor; cell permeable

5169Noradrenaline bitartrate

Endogenous adrenergic hormone and neurotransmitter

5171NBOH-2C-CN hydrochloride

High affinity, selective 5-HT2A agonist

5172FLI 06

Inhibitor of Notch signaling

5173MS 436

Potent and selective BRD4(1) inhibitor


Broad spectrum, irreversible inhibitor of serine proteases

5176JNJ 27141491

Potent and selective human CCR2 antagonist

5177WZ 4003

Potent and selective NUAK1/2 inhibitor

5178ASP 7663

Selective TRPA1 activator


Selective ubiquitin C-terminal hydrolase-L3 (UCH-L3) inhibitor

5180Ferrostatin 1

Selective inhibitor of erastin induced ferroptosis


Potent and selective vasopressin V2 receptor antagonist; renoprotective and orally active

5182OXA 06 dihydrochloride

Potent ROCK inhibitor

5183ETP 45835 dihydrochloride

Mnk1 and Mnk2 inhibitor

5184BDS I

Potent and reversible Kv3.4 potassium channel blocker; neuroprotective

5185JTE 607 dihydrochloride

Cytokine release inhibitor; anti-inflammatory


Selective inducer of neuronal differentiation in hippocampal neural progenitors

5188S 07662

Inverse agonist of the constitutive androstane receptor (CAR)

5189GSK 2837808A

Potent, selective LDHA inhibitor

5190FRAX 486

Potent PAK inhibitor; brain penetrant and orally bioavailable

5191PTC 209

Bmi-1 inhibitor; antitumor

5192NBI 31772

High affinity insulin-like growth factor-I binding protein IGFBP inhibitor


N-acetyltransferase 10 (NAT10) inhibitor

5195Agitoxin 2

Potent Shaker K+ channel blocker

5196PMX 205

Potent C5a receptor peptide antagonist

5197Spautin 1

USP10 and USP13 inhibitor; inhibits autophagy

5198AZ 20

Potent and selective ATR kinase inhibitor; antitumor

5199AZD 7762 hydrochloride

Potent and selective ATP-competitive inhibitor of Chk1 and Chk2

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