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Displaying products by catalog number (4900 - 4999)

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Cat.No.
Product Name / Activity
4900PF 4778574

Positive allosteric modulator of AMPA receptors

4901Optovin

Reversible photoactive TRPA1 activator

4902NSC 405020

Inhibitor of MT1-MMP; antitumor

4903NU 9056

Inhibitor of KAT5 (Tip60)

4904UNC 1999

Potent and selective EZH2/EZH1 inhibitor

4905UNC 2400

Negative control of UNC 1999 (Cat. No. 4904)

4906JW 642

MAGL inhibitor

4907SN 2

Selective TRPML3 channel activator

4908GNF 5

Selective allosteric inhibitor of Bcr-Abl; analog of GNF 2 (Cat. No. 4399)

4911GaTx2

High affinity, selective ClC-2 blocker; inhibits slow-gating

4912GsMTx4

TRPC1 and TRPC6 blocker; inhibits mechanosensitive ion channels

4913Jingzhaotoxin III

Selective NaV1.5 channel blocker

4914Phrixotoxin 3

Potent blocker of NaV1.2, NaV1.3 and NaV1.5 channels

4916PF 04885614

Potent and selective NaV1.8 channel blocker; active in vivo

4917M 25

Potent Smoothened (Smo) receptor antagonist

4918GSA 10

Smo receptor agonist

4919PG 106

Selective MC3 receptor antagonist

4920Methoxy-X04

Fluorescent amyloid β detector; brain penetrant

4921Leukadherin 1

Allosteric activator of CD11b/CD18

4922Purotoxin 1

Potent P2X3 modulator

4923Shz 1

Activator of early cardiac genes in pluripotent stem cells; induces differentiation in M-PBMCs

4924CEP 1347

Inhibitor of JNK signaling

4926UPF 648

Potent kynurenine 3-monooxygenase (KMO) inhibitor

4927AS 1892802

Potent ROCK inhibitor; orally bioavailable

4928OXF BD 02

Selective BRD4(1) inhibitor

4931EG 00229

Neuropilin 1 (NRP1) receptor antagonist; inhibits VEGFA binding to NRP1

4932RuBi-Dopa

Caged dopamine; exhibits two-photon sensitivity

4934MA 2029

Potent and selective, competitive motilin receptor antagonist; orally active

4935Sulfasalazine

Inhibitor of NF-κB activation; also inhibits SXC

4936Clozapine N-oxide

Activator of muscarinic DREAADs

4941PKI 166 hydrochloride

Potent EGFR-kinase inhibitor

4942Pitavastatin calcium

HMG-CoA reductase inhibitor

4943Sulfidefluor 7 AM

H2S fluorescent probe

4944Peroxy Orange 1

Fluorescent hydrogen peroxide indicator

4945ML 347

Potent and selective ALK1 and ALK2 inhibitor

4946AIM 100

Potent and selective Ack1 (TNK2) inhibitor

4948CYM 50769

Novel non-peptide NPBWR1 antagonist

4949MaxiPost

Potassium channel modulator; exerts subtype-specific effects

4950ICA 110381

KV7.2/7.3 activator; displays anticonvulsant properties

4951SA 4503 dihydrochloride

Selective σ1 receptor agonist

4952TRAM 39

Potent KCa3.1 blocker

4953CHIR 99021 trihydrochloride

Hydrochloride salt of CHIR 99021 (Cat. No. 4423); selective GSK-3 inhibitor

4954UAMC 00039 dihydrochloride

Dipeptidyl peptidase II (DPP-II) inhibitor

4957ML 179

Selective liver receptor homolog 1 (LRH1) inverse agonist

4958Eplivanserin hemifumarate

Potent and selective 5-HT2A antagonist

4959CID 16020046

Selective GPR55 antagonist

4960AR-C155858

MCT1 and MCT2 inhibitor; inhibits glycolysis in cancer cells

4961TC-S 7001

Potent and highly selective ROCK inhibitor; orally active

4962SB 204990

ATP citrate lyase (ACLY) inhibitor

4963SC 144 hydrochloride

gp130 inhibitor; blocks cytokine-triggered gp130 signaling

4964R 1485 dihydrochloride

Selective and high affinity 5-HT6 antagonist

4965PD 180970

p210Bcr/Abl kinase inhibitor; also inhibits c-Src and KIT

4968CCT 241533 dihydrochloride

Potent Chk2 inhibitor

4969LY 2389575 hydrochloride

Selective negative allosteric modulator of mGlu3

4972JIB 04

Pan Jumonji inhibitor; active in vivo

4975CRT 0066101

Potent protein kinase D (PKD) inhibitor

4976ML 289

Selective negative allosteric modulator of mGlu3

4977RN 1 dihydrochloride

LSD1 inhibitor

4978Pyrintegrin

Enhances survival of human ESCs following enzymatic dissociation

4979Methylmalonate

Succinate dehydrogenase inhibitor

4981Cystamine dihydrochloride

Transglutaminase inhibitor; neuroprotective

4982ML 337

Selective negative allosteric modulator of mGlu3

4983ACT 335827

Potent and selective OX1 antagonist

4984CK 869

Arp2/3 inhibitor; inhibits actin polymerization

4985Miglitol

α-glucosidase inhibitor

4986K 02288

Type 1 BMP receptor inhibitor

4987Ethacrynic acid - d5

Deuterated ethacrynic acid

4988Vialinin A

Inhibitor of USP4 and USP5/IsoT

4989Salirasib

Ras inhibitor; also induces autophagy

4990Stavudine

Nucleoside analog; antiviral

4992IWP L6

Potent PORCN inhibitor

4993NSC 624206

Ubiquitin-activating enzyme (E1) inhibitor

4994PYZD 4409

Ubiquitin-activating enzyme (E1) inhibitor

4995Phortress

Prodrug of the antitumor agent 5F 203

4996PMX 464

Putative inhibitor of the Trx-TrxR system; antiproliferative

4997INDY

DYRK1A/B inhibitor

4998ProINDY

DYRK1A/B inhibitor; prodrug of INDY (Cat. No. 4997)

49999-Phenanthrol

Selective TRPM4 blocker

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