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Displaying products by catalog number (4700 - 4799)

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Cat.No.
Product Name / Activity
4700PU 02

Negative allosteric modulator of 5-HT3

4701EC 144

High affinity, potent and selective Hsp90 inhibitor

4702ETP 45658

Potent PI 3-kinase inhibitor; also inhibits DNA-PK and mTOR

47033-Deazaneplanocin A hydrochloride

EZH2 histone methyltransferase inhibitor

4704LP 20 hydrochloride

Selective 5-HT7 ligand

4705Chetomin

Blocks interaction of HIF-1α, HIF-2α and STAT2 with CBP/p300

4706Borrelidin

Antiangiogenic; inhibits threonyl-tRNA synthetase

4707MI 2 dihydrochloride

Menin-MLL interaction inhibitor

4708TC LPA5 4

LPA5 receptor antagonist

4709RuBi GABA trimethylphosphine

Caged GABA; inhibits neural activity

4710PF 06465469

Potent ITK inhibitor; also inhibits BTK

4711Hexa-D-arginine

Furin inhibitor

4712Salmeterol xinafoate

Long-acting β2 agonist; bronchodilator

4713IQ 1

Enables Wnt/β-catenin-driven expansion of ESCs; prevents spontaneous differentiation

4715JZL 195

Dual FAAH and MAGL inhibitor

4716A 967079

Selective TRPA1 channel blocker

4717Jervine

Inhibitor of Hedgehog (Hh) signaling; binds directly to Smo

4718Huwentoxin IV

Selective NaV1.7 channel blocker

4719VU 0463271

Potent and selective KCC2 inhibitor

4720Entacapone

Potent COMT inhibitor; blocks α-synuclein aggregation

4722Decynium 22

PMAT inhibitor

4723T2AA

PCNA inhibitor

4724BTT 3033

Selective inhibitor of integrin α2β1

4725Eptifibatide

Glycoprotein IIb/IIIa inhibitor; inhibits platelet aggregation

4726CTA 056

ITK inhibitor

4727GS 6201

Selective A2B antagonist

4729α-Spinasterol

TRPV1 antagonist; active in vivo

4730PPY A

Potent inhibitor of Abl T315l mutant and wild-type Abl kinases

4731KY 02111

Inhibits canonical Wnt signaling. Promotes differentiation of human ESCs and iPSCs into cardiomyocytes

4732ML 204

Selective TRPC4 blocker

4733P005091

USP7 inhibitor

4734TRC 051384

Inducer of heat shock protein Hsp70

4735Quetiapine hemifumarate

5-HT2/D2 antagonist; atypical antipsychotic

4736WIN 18446

ALDH1a2 inhibitor

4737CDDO Im

Nrf2 signaling activator

4738LY 333531 hydrochloride

Protein kinase C inhibitor; selective for β isozymes

4739Cesium chloride

Potassium channel blocker; neuroprotective

4740Lithium carbonate

Mood stabilizer; inhibits Na+/K+ ATPase pump activity

4741Gadolinium chloride

Stretch-activated calcium channel blocker; calcium-sensing receptor agonist

4742Gue 1654

Selective inhibitor of OXE-R Gβγ signaling

4744P11

Potent antagonist of αvβ3-vitronectin interaction; antiangiogenic

4745LIMKi 3

Potent LIM kinase inhibitor; antitumor

4746ML SA1

Activator of TRPML channels

4747TC-G 1006

Potent and selective sphingosine-1-phosphate receptor 1 (S1P1) agonist

4748ML 221

Apelin receptor (APJ) antagonist

4749Strontium chloride

Calcium sensing receptor (CaSR) agonist

4750TC Mps1 12

Potent and selective Mps1 kinase inhibitor

4751FSLLRY-NH2

PAR2 peptide antagonist

4752SA 57

Potent FAAH inhibitor

4753AL 8697

Potent and selective p38α inhibitor

4754AK 7

Selective SIRT2 inhibitor; brain penetrant

4755Q94 hydrochloride

Negative allosteric modulator at PAR1 receptor

4756COR 170

Selective CB2 receptor inverse agonist

4757Latanoprost

FP prostaglandin receptor agonist; also exhibits agonist activity at EP1 and EP3 receptors

4758Bromosporine

Broad spectrum bromodomain inhibitor

4759G-36

Selective GPER antagonist

4761Plumbagin

Induces G2/M cell cycle arrest; anticancer

4762MIM1

Mcl-1 inhibitor; proapoptotic

4763Pyridostatin pentahydrochloride

Stabilizes G-quadruplexes; induces DNA damage and cell cycle arrest

4764SIB 1553A hydrochloride

Subunit selective nAChR agonist

4766SIB 1508Y maleate

Potent agonist of α4β2, α2β4, α4β4 and α3β4 nACh receptors

4767WAY 316606 hydrochloride

Secreted Frizzled-related protein-1 (sFRP-1) inhibitor; increases Wnt signaling

4769VUF 10460

Selective H4 agonist

4773ESI 09

EPAC inhibitor

4774BMS 536924

Dual IR/IGF1R inhibitor

4775SD 2590 hydrochloride

Potent MMP inhibitor

4776BIRT 377

Potent negative allosteric modulator of LFA-1

4777ML 277

Selective Kv7.1 (KCNQ1) potassium channel activator; augments IKs current

4778BETP

Positive allosteric modulator of GLP-1 receptors

4779GRI 977143

Selective LPA2 receptor non-lipid agonist

4780VUF 11207 fumarate

Potent ACKR3 (CXCR7) agonist

4781ANA 12

TrkB receptor antagonist

4782Org 25543 hydrochloride

Potent and selective GlyT2 inhibitor

4783Lu AA 47070

Prodrug of a potent and selective adenosine A2A receptor antagonist

4784Edaglitazone

Potent and selective PPARγ agonist; antidiabetic

4785SA 47

Selective FAAH inhibitor

4786PD 0332991 isethionate

Potent, selective Cdk4/6 inhibitor; brain penetrant

4787CPPHA

Positive allosteric modulator at mGlu1 and mGlu5

4788NS 11021

Activator of BKCa (KCa1.1) channels

4791Candesartan

AT1 receptor antagonist

4792Candesartan cilexetil

Prodrug of candesartan (Cat. No. 4791), an AT1 receptor antagonist

4793CE3F4

Uncompetitive Epac1 inhibitor

4794ZCL 278

Cdc42 inhibitor

4795Galloflavin

Lactate dehydrogenase inhibitor; impairs aerobic glycolysis

4796Escitalopram oxalate

Selective serotonin reuptake inhibitor (SSRI)

4797Org 37684

5-HT2 agonist

4798(S)-Duloxetine hydrochloride

Potent 5-HT and NA reuptake inhibitor; also blocks dopamine reuptake

4799Capecitabine

Prodrug of 5-Fluorouracil (Cat. No. 3257). Inhibits DNA synthesis

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