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Displaying products by catalog number (4500 - 4599)

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Cat.No.
Product Name / Activity
4500Cercosporamide

Potent Mnk2 inhibitor

4501Ribavirin

Antiviral guanosine analog; blocks eIF4E activity

4502DIM

Activates Chk2; induces G2/M cell cycle arrest

4503CC 0651

Allosteric inhibitor of hCdc34

4504Chaetocin

SUV39H1 inhibitor

4505ICG 001

Inhibits TCF/β-catenin-mediated transcription

4506TAME hydrochloride

Ubiquitin ligase APC/C inhibitor; promotes Cdc20 autoubiquitination

4507ML 218 hydrochloride

Ca2+ channel blocker (T-type)

4508S 32212 hydrochloride

5-HT2C inverse agonist; α2 antagonist

4509STF 083010

Inhibits IRE1α endonuclease activity

4510SHA 68

Selective neuropeptide S receptor antagonist

4511MMF

Activator of Nrf2 pathway; primary metabolite of DMF (Cat. No. 4512)

4512DMF

Nrf2 pathway activator; neuroprotective

4513Kartogenin

Potently induces chondrogenesis in MSCs

4514JW 55

Tankyrase inhibitor

45152-Deoxy-D-glucose

Non-metabolizable glucose analog; hexokinase substrate

4516UNC 926 hydrochloride

L3MBTL1 domain inhibitor

4517NS 2028

Potent soluble guanylyl cyclase (sGC) inhibitor

4518EPPTB

Trace amine 1 (TA1) receptor antagonist/inverse agonist

4519ML 213

KV7.2 and KV7.4 channel opener

4520Cytarabine

Nucleoside analog; inhibits DNA replication

4521TAS 301

Inhibitor of smooth muscle cell migration and proliferation

4522Flufenamic acid

Activates TRPC6; NSAID

4523DIDS

Chloride channel blocker; TRPV1 modulator; RAD51 recombinase inhibitor

4524EGCG

Inhibits formation of amyloid fibrils

4525Piclamilast

Potent and selective PDE4 inhibitor

4527TC-I 15

Potent α2β1 inhibitor; displays antithrombotic activity in vivo

4528(±)-NBI 74330

Potent and selective CXCR3 antagonist

4529Ciliobrevin A

Hedgehog (Hh) pathway antagonist, inhibits ciliogenesis; also inhibits dynein

4530ONO 2506

Inhibits S-100β synthesis; neuroprotective

4531NCX 4040

NO-donating aspirin; anti-inflammatory and antitumor

4532VUF 10166

High affinity 5-HT3 receptor antagonist

4533PTAC oxalate

Muscarinic receptor ligand; exhibits partial agonist and antagonist activity at different subtypes

4534CZC 54252 hydrochloride

Potent LRRK2 inhibitor; neuroprotective

4535Phalloidin

Promotes actin polymerization

4536Resiquimod

Toll-like receptor 7 (TLR7) agonist

4537NCX 466

Cyclooxygenase-inhibiting nitric oxide donor

4538T16Ainh - A01

Ca2+-activated Cl- channel transmembrane protein 16A (TMEM16A) inhibitor

4539(R)-(+)-Etomoxir sodium salt

Carnitine palmitoyltransferase I (CPT1) inhibitor

4540U 104

Potent carbonic anhydrase (CA) IX and XII inhibitor

4541SGC 0946

Highly potent and selective DOT1L inhibitor; cell permeable

4542(+)-Fluprostenol

High affinity FP prostaglandin receptor agonist

4543CS 2100

Selective S1P1 agonist

4544YM 244769

Na+/Ca2+ exchange inhibitor (reverse mode); neuroprotective

4545E 64d

Cathepsin inhibitor; interferes with autolysosomal digestion

4546rac-CCT 250863

Potent Nek2 inhibitor

4547ACHP

Selective IKKα and IKKβ inhibitor

4549ML 133 hydrochloride

Kir2 channel blocker

4550IQ 3

Selective JNK3 inhibitor

4551Purmorphamine

Smo receptor agonist

4552A 412997 dihydrochloride

Selective D4 agonist

4553Azilsartan

Potent AT1 receptor inverse agonist; antihypertensive

4554GC 1

High affinity thyroid receptor α (TRα) and TRβ agonist; thyromimetic

4555HI TOPK 032

Selective T-LAK-cell-originated protein kinase (TOPK) inhibitor

4556CP 690550 citrate

Potent JAK inhibitor

4557GTS 21 dihydrochloride

Partial agonist at α7 nAChR

4558EMPA

Highly potent and selective OX2 antagonist; brain penetrant

4559GNF 5837

Potent Trk inhibitor; inhibits TrkA, TrkB and TrkC

4561BIBN 4096

Potent and selective CGRP receptor antagonist

4562Topotecan hydrochloride

DNA topoisomerase I inhibitor; Camptothecin (Cat. No. 1100) analog

4564JTV 519 fumarate

Ryanodine receptor (RyR) inhibitor

4565ML 228

HIF pathway activator

4566NSC 687852

Inhibitor of UCHL5 and USP14

4567CCG 50014

Potent and selective inhibitor of regulator of G-protein signaling 4 (RGS4) protein

4568CPYPP

DOCK2-Rac1 interaction inhibitor

4569PS 1145 dihydrochloride

Selective IKK inhibitor; orally active

4570ML 161

Inhibits PAR1-mediated platelet activation

4571A 867744

Positive allosteric modulator of α7 nAChR

4572TC-E 5005

Potent and selective PDE10A inhibitor

4574ARN 272

FAAH-like anandamide transporter (FLAT) inhibitor

4575TC HSD 21

Potent and selective 17β-hydroxysteroid dehydrogenase type 3 inhibitor

4577LDV FITC

Fluorescent ligand for α4β1 (VLA-4)

4578Phenobarbital sodium salt

Enhances GABAergic activity

4579Pentobarbital sodium salt

Enhances GABAergic activity

4580Atiprimod dihydrochloride

JAK2 inhibitor

4581Grifolic acid

Selective partial FFA4 (GPR120) agonist

4582MLR 1023

Selective allosteric activator of Lyn kinase

4583Digoxin

Na+/K+ ATPase inhibitor

4584SNS 314 mesylate

Potent pan-Aurora kinase inhibitor

4585MRT 10

Smoothened (Smo) antagonist

4586ML 3403

p38 inhibitor

45888MDP

Potent equilibrative nucleoside transporter (ENT) inhibitor

4590Honokiol

Blocks NF-κB activation; also anti-inflammatory and antioxidant

4591Deltorphin I

Potent δ agonist

4592R8-T198wt

Pim-1 kinase inhibitor

4593GSK J1

Potent JMJD3/UTX inhibitor

4594GSK J4

Histone KDM inhibitor; cell permeable

4596IT1t dihydrochloride

Potent CXCR4 antagonist

4597NS 8593 hydrochloride

Selective KCa2 (SK) channel negative modulator; inhibits SK currents

4598PHT 427

Dual Akt and PDK1 inhibitor; antitumor

45993,5-DHBA

Selective HCA1 agonist

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