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Displaying products by catalog number (4300 - 4399)

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Product Name / Activity
4300TC 14012

CXCR4 antagonist; ACKR3 (CXCR7) agonist

4301TC-DAPK 6

Potent and selective inhibitor of DAPK1

4302Perindopril erbumine

Angiotensin-converting enzyme (ACE) inhibitor

4303PPQ 102

Potent, voltage-independent CFTR chloride channel inhibitor

4305ICA 069673

KV7.2/KV7.3 channel opener

4306INCB 3284 dimesylate

Selective CCR2 antagonist

4307YC 1

Soluble guanylyl cyclase (sGC) activator; induces G1 cell cycle arrest

4308Rasagiline mesylate

Selective, irreversible MAO-B inhibitor


Cell-permeable Zn2+ chelator

4310ML 7 hydrochloride

Selective inhibitor of myosin light chain kinase

4311GW 542573X

Selective activator of KCa2.1 channels

4312Nigericin sodium salt

Selective K+ ionophore

4314SB 268262

Selective non-peptide CGRP1 antagonist

4315NGD 98-2 hydrochloride

High affinity CRF1 antagonist


Immunomodulatory and antitumor compound

4317JNJ 10397049

Selective OX2 receptor antagonist

4318BX 795

PDPK1 (PDK1) inhibitor

4319A 784168

Potent and selective TRPV1 antagonist

4320FC 131

CXCR4 antagonist

4322JH 295

Irreversible Nek2 inhibitor

4323VU 0360172 hydrochloride

Positive allosteric modulator at mGlu5


HIF-1α inhibitor; down-regulates HIF-1α protein synthesis

4325Phosphocreatine disodium salt

Phosphate reservoir

4326PhiKan 083

p53 stabilizing agent

4327JW 480

Potent and selective inhibitor of serine hydrolase KIAA1363 (AADACL1)

4330AMG 21629

Potent and selective TRPV1 antagonist

4333PSB 1114

Potent, selective P2Y2 agonist

4334PSB 0777 ammonium salt

Potent adenosine A2A agonist

4335AR-M 1000390 hydrochloride

Low-internalizing δ agonist

4336TG 003

Potent inhibitor of Clk-family kinases; also inhibits DYRK1A/B

4337ST 1936 oxalate

Selective, high affinity 5-HT6 agonist

4338NSC 33994

JAK2 inhibitor

4339Tertiapin LQ

Selective Kir1.1 blocker; derivative of tertiapin-Q (Cat. No. 1316)

4341A 582941

Partial agonist at α7 nAChR

4342UNC 0646

Potent and selective G9a and GLP inhibitor

4343UNC 0638

Selective G9a and GLP inhibitor

4344FH 535

Inhibitor of Wnt/β-catenin signaling

4345TC-C 14G

Potent, high affinity CB1 receptor inverse agonist

4346Ro 67-7476

Positive allosteric modulator of mGlu1

4347Ro 67-4853

Positive allosteric modulator of group I mGlu receptors

4348Ro 01-6128

Positive allosteric modulator of mGlu1


5-HT2A/D2 antagonist; atypical antipsychotic


Potent VEGFR-1, -2 and -3 inhibitor

4351JHW 007 hydrochloride

High affinity dopamine uptake inhibitor

4352Talsupram hydrochloride

Selective inhibitor of noradrenalin transporters

4353TC-G 24

Potent and selective GSK-3β inhibitor

4354ML 130

Inhibits NOD1-induced NF-κB activation

4355TC-F 2

Potent, reversible and selective FAAH inhibitor

4357Bicifadine hydrochloride

Noradrenalin, 5-HT and dopamine re-uptake inhibitor

4358Dapoxetine hydrochloride

Selective serotonin reuptake inhibitor


MGMT inhibitor


Dual Src-Abl inhibitor; antiproliferative

4362PF 5081090

Potent LpxC inhibitor

4363TC-SP 14

Potent S1P1 receptor agonist

4365TC-MCH 7c

Selective melanin-concentrating hormone receptor 1 (MCH1R) antagonist


Potent Smoothened receptor agonist; activates the Hedgehog signaling pathway

4367Psora 4

Potent KV1.3 channel blocker


Potent c-MET/ALK inhibitor

4370TC-N 22A

Potent, selective mGlu4 positive allosteric modulator

4371VU 0364439

Positive allosteric modulator at mGlu4

4372BC 11 hydrobromide

Selective urokinase (uPA) inhibitor


Positive allosteric modulator of GluR2 receptors

4374BIMU 8

Potent 5-HT4 receptor full agonist

4375SMER 3

Selective inhibitor of E3 ubiquitin ligase

43765-OMe-UDP trisodium salt

Potent P2Y6 agonist


LRH-1 agonist; regulates bile acid metabolism

4379(S)-(+)-Ketamine hydrochloride

NMDA receptor antagonist; enantiomer of ketamine hydrochloride (Cat. No. 3131); neuroprotective.

4380WAY 100635 maleate

Potent, 5-HT1A silent antagonist. Also D4 agonist

4381VU 0285683

Negative allosteric modulator at mGlu5


Potent, reversible non-steroidal aromatase inhibitor

4385Donepezil hydrochloride

Potent AChE inhibitor

4386TC-P 262

Selective P2X3, P2X2/3 antagonist

4387Calhex 231 hydrochloride

Negative allosteric modulator of the calcium-sensing receptor

4388MNI 137

Selective negative allosteric modulator of group II mGlu receptors

4390Thiamet G

Potent O-GlcNAcase inhibitor

4391Ro 51

Potent P2X3, P2X2/3 antagonist


Potent and selective tryptophan 2,3-dioxygenase (TDO) inhibitor


Tryptophan catabolite; endogenous aryl hydrocarbon receptor ligand

4394VU 0360223

Negative allosteric modulator at mGlu5


Reversible MAO-A inhibitor


Induces apoptosis; increases p53 and ROS levels in cancer cells

4397AV 412

Potent inhibitor of EGFR, ErbB2 and Abl receptor tyrosine kinases

4398SC 66

Allosteric Akt inhibitor

4399GNF 2

Selective allosteric inhibitor of Bcr-Abl tyrosine kinase activity

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Careers at Tocris

Tocris Bioscience currently has opportunities for a Product Manager.

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Bio-Techne Events

26th ISN-ESN Biennal Meeting

26th ISN-ESN Biennial Meeting

August 20 - 24, 2017

Paris , France

Booth: 11