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Displaying products by catalog number (4200 - 4299)

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Cat.No.
Product Name / Activity
4200C 646

Selective p300/CBP inhibitor

4202Adenine

Adenine receptor agonist

4204BTZO 1

MIF binder

4205MDA 19

CB2 agonist

4206Valdecoxib

Selective and potent COX-2 inhibitor

4207SB 277011A dihydrochloride

Selective D3 antagonist

4208MS 245 oxalate

High affinity 5-HT6 antagonist

4209EMDT oxalate

Selective 5-HT6 agonist

4210Ascomycin

Calcineurin phosphatase inhibitor; analog of FK 506 (Cat. No. 3631)

4212PIR 3.5

Negative control of IPA 3 (Cat. No. 3622)

4213SB 297006

Potent and selective CCR3 antagonist

4214Prostaglandin F2α

Naturally-occurring prostanoid; potent vasoconstrictor

42154E1RCat

Protein translation inhibitor; blocks eIF4F subunit interaction

4216Valsartan

High affinity, selective AT1 antagonist

4218Travaprost

Potent and selective FP prostaglandin receptor agonist

4219Banoxantrone dihydrochloride

Prodrug topoisomerase II inhibitor

4220XCC

Adenosine receptor antagonist

4221TCS 21311

Potent JAK3 inhibitor. Also inhibits GSK-3β and PKC

4222Dynole 34-2

Dynamin I inhibitor

4224MitMAB

Dynamin inhibitor

4225OctMAB

Dynamin inhibitor

4227RWJ 50271

Inhibitor of LFA-1/ICAM mediated cell adhesion

4228A 286982

Potent inhibitor of the LFA-1/ICAM-1 interaction

4230NPEC-caged-D-AP5

Caged D-AP5 (Cat.No. 0106)

4231Nateglinide

Kir6 (KATP) blocker; displays high affinity for SUR1/Kir6.2 channels

4232A 839977

Potent P2X7 antagonist

4233TQS

Positive allosteric modulator of α7 nAChRs

42344BP-TQS

Allosteric agonist at α7 nAChR

4236CP 945598 hydrochloride

CB1 receptor antagonist

4237PD 184352

Selective MEK inhibitor

4238PF 184

Potent and selective IKKβ inhibitor

4239PF 04217903 mesylate

Highly selective MET inhibitor

4240SCH 529074

Restores mutant p53 activity

4241Olopatadine hydrochloride

H1 antagonist; ocular antiallergic agent

4242GW 803430

MCH1 antagonist

4243Kisspeptin 10 (rat)

Endogenous ligand for kisspeptin receptor

4244TCS 3035

GPR35 agonist

4245Meclizine dihydrochloride

Human pregnane X receptor agonist; H1 antagonist

4246CID 2858522

Selectively inhibits PKC-induced NF-κB activation

4247Torin 1

Potent and selective mTOR inhibitor

4248Torin 2

Potent and selective mTOR inhibitor

4249A 887826

Potent voltage-dependent NaV1.8 channel blocker

4250Mitoxantrone dihydrochloride

Topoisomerase II inhibitor; immunosuppressive and antineoplastic agent

4252PF 4981517

Selective CYP3A4 inhibitor

4253TMPyP4 tosylate

Inhibitor of human telomerase

4254TAK 715

Potent p38 MAPK inhibitor; anti-inflammatory

4255TC-O 9311

Potent and selective GPR139 agonist

4256Tiagabine hydrochloride

GABA uptake inhibitor; anticonvulsant

4257PP 242

Dual mTORC1/mTORC2 inhibitor

4259TCN 238

Positive allosteric modulator of mGlu4

4260MRS 2957 triethylammonium salt

Potent and selective P2Y6 agonist

4261MRS 4062 triethylammonium salt

Selective P2Y4 receptor agonist

4264TG 100713

PI 3-kinase inhibitor

4266ML 141

Selective inhibitor of Cdc42 Rho family GTPase

4268Ro 1138452 hydrochloride

Selective prostacyclin IP receptor antagonist

4270TC-H 106

Class I histone deacetylase inhibitor

4272[D-Trp8]-γ-MSH

Selective MC3 receptor agonist

4273LRRK2-IN-1

Potent and selective LRRK2 inhibitor

4274AP 24534

Potent multi-kinase and pan-Bcr-Abl inhibitor

4276ERB 041

Potent ERβ agonist

4277PF 477736

Selective Chk1 inhibitor

4278PF 431396

Dual FAK/PYK2 inhibitor

4279PF 3644022

Potent MK2 inhibitor

4281PF 4800567 hydrochloride

Selective casein kinase 1ε inhibitor

4282WYE 687 dihydrochloride

Potent and selective mTOR inhibitor

4283Begacestat

γ-secretase inhibitor; lowers Aβ40 and Aβ42 levels

4285HBX 41108

Selective USP7 inhibitor

4286UA 62784

Inhibits microtubule polymerization

4287Poly(I:C)

TLR3 agonist

4288ISO 1

Macrophage migration inhibitory factor (MIF) inhibitor

4289RP 001 hydrochloride

Potent S1P1 agonist

4291CCT 137690

Potent pan-Aurora kinase inhibitor

4292SBE 13 hydrochloride

Potent and selective PLK1 inhibitor

4293CID 2745687

GPR35 antagonist

4294LB 42708

Selective farnesyltransferase (FTase) inhibitor

4295VU 0357017 hydrochloride

Positive allosteric modulator of M1 receptors

4297SMER 28

Positive regulator of autophagy

4298Pamoic acid disodium salt

GPR35 agonist

4299iCRT 14

Inhibits β-catenin-responsive transcription (CRT)

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