All Products

Displaying products by catalog number (4200 - 4299)

0100 0200 0300 0400 0500 0600 0700 0800 0900 1000
1100 1200 1300 1400 1500 1600 1700 1800 1900 2000
2100 2200 2300 2400 2500 2600 2700 2800 2900 3000
3100 3200 3300 3400 3500 3600 3700 3800 3900 4000
4100 4200 4300 4400 4500 4600 4700 4800 4900 5000
5100 5200 5300 5400 5500 5600 5700 5800 5900 6000
6100 6200
Product Name / Activity
4200C 646

Selective p300/CBP inhibitor


Adenine receptor agonist

4204BTZO 1

MIF binder

4205MDA 19

CB2 agonist


Selective and potent COX-2 inhibitor

4207SB 277011A dihydrochloride

Selective D3 antagonist

4208MS 245 oxalate

High affinity 5-HT6 antagonist

4209EMDT oxalate

Selective 5-HT6 agonist


Calcineurin phosphatase inhibitor; analog of FK 506 (Cat. No. 3631)

4212PIR 3.5

Negative control of IPA 3 (Cat. No. 3622)

4213SB 297006

Potent and selective CCR3 antagonist

4214Prostaglandin F2α

Naturally-occurring prostanoid; potent vasoconstrictor


Protein translation inhibitor; blocks eIF4F subunit interaction


High affinity, selective AT1 antagonist


Potent and selective FP prostaglandin receptor agonist

4219Banoxantrone dihydrochloride

Prodrug topoisomerase II inhibitor


Adenosine receptor antagonist

4221TCS 21311

Potent JAK3 inhibitor. Also inhibits GSK-3β and PKC

4222Dynole 34-2

Dynamin I inhibitor


Dynamin inhibitor


Dynamin inhibitor

4227RWJ 50271

Inhibitor of LFA-1/ICAM mediated cell adhesion

4228A 286982

Potent inhibitor of the LFA-1/ICAM-1 interaction


Caged D-AP5 (Cat.No. 0106)


Kir6 (KATP) blocker; displays high affinity for SUR1/Kir6.2 channels

4232A 839977

Potent P2X7 antagonist


Positive allosteric modulator of α7 nAChRs


Allosteric agonist at α7 nAChR

4236CP 945598 hydrochloride

CB1 receptor antagonist

4237PD 184352

Selective MEK inhibitor

4238PF 184

Potent and selective IKKβ inhibitor

4239PF 04217903 mesylate

Highly selective MET inhibitor

4240SCH 529074

Restores mutant p53 activity

4241Olopatadine hydrochloride

H1 antagonist; ocular antiallergic agent

4242GW 803430

MCH1 antagonist

4243Kisspeptin 10 (rat)

Endogenous ligand for kisspeptin receptor

4244TCS 3035

GPR35 agonist

4245Meclizine dihydrochloride

Human pregnane X receptor agonist; H1 antagonist

4246CID 2858522

Selectively inhibits PKC-induced NF-κB activation

4247Torin 1

Potent and selective mTOR inhibitor

4248Torin 2

Potent and selective mTOR inhibitor

4249A 887826

Potent voltage-dependent NaV1.8 channel blocker

4250Mitoxantrone dihydrochloride

Topoisomerase II inhibitor; immunosuppressive and antineoplastic agent

4252PF 4981517

Selective CYP3A4 inhibitor

4253TMPyP4 tosylate

Inhibitor of human telomerase

4254TAK 715

Potent p38 MAPK inhibitor; anti-inflammatory

4255TC-O 9311

Potent and selective GPR139 agonist

4256Tiagabine hydrochloride

GABA uptake inhibitor; anticonvulsant

4257PP 242

Dual mTORC1/mTORC2 inhibitor

4259TCN 238

Positive allosteric modulator of mGlu4

4260MRS 2957 triethylammonium salt

Potent and selective P2Y6 agonist

4261MRS 4062 triethylammonium salt

Selective P2Y4 receptor agonist

4264TG 100713

PI 3-kinase inhibitor

4266ML 141

Selective inhibitor of Cdc42 Rho family GTPase

4268Ro 1138452 hydrochloride

Selective prostacyclin IP receptor antagonist

4270TC-H 106

Class I histone deacetylase inhibitor


Selective MC3 receptor agonist


Potent and selective LRRK2 inhibitor

4274AP 24534

Potent multi-kinase and pan-Bcr-Abl inhibitor

4276ERB 041

Potent ERβ agonist

4277PF 477736

Selective Chk1 inhibitor

4278PF 431396

Dual FAK/PYK2 inhibitor

4279PF 3644022

Potent MK2 inhibitor

4281PF 4800567 hydrochloride

Selective casein kinase 1ε inhibitor

4282WYE 687 dihydrochloride

Potent and selective mTOR inhibitor


γ-secretase inhibitor; lowers Aβ40 and Aβ42 levels

4285HBX 41108

Selective USP7 inhibitor

4286UA 62784

Inhibits microtubule polymerization


TLR3 agonist

4288ISO 1

Macrophage migration inhibitory factor (MIF) inhibitor

4289RP 001 hydrochloride

Potent S1P1 agonist

4291CCT 137690

Potent pan-Aurora kinase inhibitor

4292SBE 13 hydrochloride

Potent and selective PLK1 inhibitor

4293CID 2745687

GPR35 antagonist

4294LB 42708

Selective farnesyltransferase (FTase) inhibitor

4295VU 0357017 hydrochloride

Positive allosteric modulator of M1 receptors

4297SMER 28

Positive regulator of autophagy

4298Pamoic acid disodium salt

GPR35 agonist

4299iCRT 14

Inhibits β-catenin-responsive transcription (CRT)

Products Alphabetically by Name



Quick Order

Find multiple products by catalog number

divider line

Careers at Tocris

Careers at Tocris

Tocris Bioscience currently has opportunities for a Product Manager.

If you would like to be considered for any positions not currently advertised, we welcome your speculative application.

divider line

Bio-Techne Events

WCI 2017

13th World Congress on Inflammation

July 8 - 12, 2017

London, UK