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Displaying products by catalog number (2400 - 2499)

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Product Name / Activity
2400FK 888

High affinity NK1 receptor antagonist

2402MRS 2211

Competitive P2Y13 antagonist

2403MRS 3777 hemioxalate

High affinity, selective A3 antagonist

2404Ambroxol hydrochloride

Na+ channel blocker

2407FTI 277

Prodrug form of FTI 276 (Cat. No. 2406)

2408Ro 90-7501

Inhibitor of Aβ42 fibril formation


Potent and selective H3 receptor antagonist


Potent and selective oxytocin receptor antagonist


Potent and selective CCK1 agonist; suppresses feeding

2412BIBO 3304 trifluoroacetate

Highly selective NPY Y1 receptor antagonist

2414H 1152 dihydrochloride

Selective Rho-kinase (ROCK) inhibitor

2415HA 1100 hydrochloride

Cell-permeable, selective Rho-kinase inhibitor

2416BIBX 1382 dihydrochloride

Highly selective EGFR-kinase inhibitor

2417BIBU 1361 dihydrochloride

Selective inhibitor of EGFR-kinase

2418LY 303511

Negative control of LY 294002 (Cat. No. 1130)

2419GT 2016

Selective H3 antagonist


Potent peptide agonist for APJ receptor


Histone deacetylase inhibitor


Akt/PKB substrate (synthetic)


Chemokine receptor 5 (CCR5) antagonist

2424Amyloid β-peptide (1-40) (rat)

Amyloid β-protein fragment

2425Amyloid β-peptide (1-42) (rat)

Predominant amyloid β-protein fragment

2426Apelin-36 (human)

Endogenous APJ receptor agonist

2427Apelin-36 (rat, mouse)

Endogenous APJ receptor agonist

2429Fexofenadine hydrochloride

H1 receptor antagonist; non-sedating antiallergic agent

2430GGTI 298

Geranylgeranyltransferase I (GGTase I) inhibitor

2432Anagrelide hydrochloride

Potent PDE3 inhibitor


High affinity, selective CB2 agonist


Highly selective CB2 agonist

2435CCT 018159

Hsp90 inhibitor

2436AC 55649

Selective RARβ2 agonist

2438TMPH hydrochloride

Neuronal nicotinic receptor antagonist

2440NNC 26-9100

Selective sst4 agonist

2441JNJ 10191584 maleate

Selective H4 receptor antagonist; orally active

2442CGP 53353

Selective inhibitor of PKCβII


MDM2-p53 interaction inhibitor


Potent and selective sst2 agonist

2445Obestatin (rat)

Endogenous reported anorexigenic peptide

2446AS 101

Immunomodulator; inhibits IL-10 synthesis and potentiates IL-1α, IL-2 and TNF-α release

2447Desmethyl-YM 298198

Derivative of mGlu1 antagonist YM 298198 (Cat. No. 2448)

2448YM 298198 hydrochloride

Highly potent, selective non-competitive mGlu1 antagonist

2450NF 157

Selective P2Y11/P2X1 antagonist

2451LY 344864 hydrochloride

Potent, selective 5-HT1F agonist

2452LY 2183240

Novel, potent anandamide uptake inhibitor; inhibits FAAH

2453LY 379268

Highly selective group II mGlu agonist

2454CH 275

Potent and selective sst1 receptor agonist

2456Co 101244 hydrochloride

Highly selective NR2B antagonist

2457Arcyriaflavin A

Potent cdk4/cyclin D1 and CaM Kinase II inhibitor. Antiviral agent (anti-HCMV)

2458ZM 447439

Inhibits Aurora kinase B

2459Tropisetron hydrochloride

Potent 5-HT3 receptor antagonist; also partial agonist of α7 nAChR

2460Lazabemide hydrochloride

Selective MAO-B inhibitor

2463SCH 442416

Very selective, high affinity A2A antagonist

2464TNP-ATP triethylammonium salt

Potent, selective P2X antagonist

2465SDZ WAG 994

Potent, selective A1 agonist

2466UK 14,304 tartrate

α2 agonist. Water-soluble form of UK 14,304 (Cat. No. 0425)

2467CGS 20625

Selective central benzodiazepine receptor partial agonist

2469IBC 293

Selective agonist for the GPR109B (HM74) receptor. Antilipolytic


Cyclooxygenase-2 (COX-2) inhibitor

2471ER 27319 maleate

Selective Syk kinase inhibitor

2472Triacsin C

Inhibitor of acyl-CoA synthetase

2473GW 4064

Selective farnesoid X receptor (FXR) agonist

2474GW 3965 hydrochloride

Orally active liver X receptor (LXR) agonist

2475ZM 323881 hydrochloride

Potent, selective inhibitor of VEGFR-2

2476SR 11302

AP-1 inhibitor; antitumor agent

2477Proxyfan oxalate

High affinity H3 ligand

24782-Pyridylethylamine dihydrochloride

H1 receptor agonist

2479JTE 907

Selective CB2 receptor antagonist/inverse agonist

2481JTC 801

Selective NOP antagonist


Inhibitor of human telomerase activity

2484(±)-AC 7954 hydrochloride

Non-peptide UT receptor agonist

2485Glycyl-H 1152 dihydrochloride

Selective Rho-kinase (ROCK) inhibitor. More selective analog of H 1152 dihydrochloride (Cat. No. 2414)

2489C 75

Potent fatty acid synthase inhibitor; proapoptotic

2490(±)-Clopidogrel hydrochloride

Selective P2Y12 antagonist

2491Xaliproden hydrochloride

Orally active, high affinity 5-HT1A agonist


Novel, non-toxic immunosuppressive agent

2493VUF 5681 dihydrobromide

Potent H3 receptor silent antagonist

2494VUF 8430 dihydrobromide

Potent, high affinity H4 agonist

2495Melperone hydrochloride

5-HT2A/D2 receptor antagonist; neuroleptic

2496DR 2313

PARP-1 and PARP-2 inhibitor

2498PNU 120596

Positive allosteric modulator of α7 nAChR; active in vivo

2499ZM 306416 hydrochloride

Inhibitor of VEGF receptor tyrosine kinase

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