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Displaying products by catalog number (1100 - 1199)

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Product Name / Activity

DNA topoisomerase inhibitor

1101Cyclosporin A

Calcineurin inhibitor

1102Procaterol hydrochloride

Potent β2 agonist


Cytochrome P450c17 inhibitor


Highly selective A3 agonist

1105AF-DX 116

Selective M2 antagonist


Selective, potent GluR5 agonist


EGFR kinase inhibitor. Also estrogen and PPARγ ligand


Group III mGlu agonist


Competitive mGlu receptor antagonist

1114CGP 37157

Antagonist of mitochondrial Na+/Ca2+ exchange

1115AM 281

Potent, selective CB1 antagonist/inverse agonist

1116AM 404

Anandamide transport inhibitor

1117AM 251

Potent CB1 antagonist; also GPR55 agonist

1118Nocistatin (bovine)

Opposes action of nociceptin


Orphan neuropeptide

1120AM 630

CB2 selective antagonist/inverse agonist


Potent and selective CB1 agonist

1122Telenzepine dihydrochloride

Potent, selective M1 antagonist

1123(S)-(+)-Niguldipine hydrochloride

α1 antagonist, L-type Ca2+ channel blocker

1124(R)-(-)-Niguldipine hydrochloride

α1 antagonist, L-type Ca2+ channel blocker. Less active enantiomer of Niguldipine hydrochloride (Cat. No. 1123)


Non-selective PI 3-kinase inhibitor


Anti-inflammatory glucocorticoid

1127Yohimbine hydrochloride

Selective α2 antagonist


GABAA receptor antagonist

1129BRL 54443

Potent 5-ht1E/F agonist

1130LY 294002 hydrochloride

Prototypical PI 3-kinase inhibitor; also inhibits other kinases


Antagonist of pancreatic imidazoline receptor


Putative endogenous imidazoline ligand. Also MAO inhibitor

1133BRL 44408 maleate

Selective α2A antagonist

1134CGP 12177 hydrochloride

β3 partial agonist. β1/β2 antagonist.

1135Spermine NONOate

Slow NO releasing agent

1136Okadaic acid

Protein phosphatase 1 and 2A inhibitor


Potent vanilloid receptor agonist


Potent inhibitor of SERCA ATPase

1139L-NIL hydrochloride

Selective iNOS inhibitor

11408-Bromo-cAMP, sodium salt

Cell-permeable cAMP analog

1141Dibutyryl-cAMP, sodium salt

Cell-permeable cAMP analog

1142Oxymetazoline hydrochloride

α1A agonist


Potent, selective inhibitor of MEK1 and 2

1145L-733,060 hydrochloride

Potent NK1 antagonist

1146MDL 28170

Potent, selective calpain and cathepsin B inhibitor

1147SKF 96365 hydrochloride

TRPC channel blocker; also inhibits store-operated Ca2+ entry


PDE3 inhibitor


Involved in gastrointestinal tract function

1150CCK Octapeptide, non-sulfated

Non-sulfated form of CCK octapeptide

1151CRF (human, rat)

Stimulates ACTH release

1152Neurokinin A (porcine)

Endogenous tachykinin peptide

1153Neuropeptide Y (human, rat)

Influences feeding and sexual behavior

1154Pancreatic Polypeptide (human)

NPY Y4 agonist; involved in gastrointestinal tract function


Tyrosine kinase substrate peptide

1156Substance P

Sensory neuropeptide; inflammatory mediator


Influences growth hormone release

1158Angiotensin II

Potent vasoconstrictor peptide

1159Calcitonin (salmon)

Affects bone formation and resorption

1160Endothelin 1 (human, porcine)

Potent vasoconstrictor peptide

1161CGRP (rat)

Potent vasodilator

1162Endothelin 3 (human, rat)

Potent vasoconstrictor


Non-selective angiotensin II antagonist

1164Endothelin 2 (human)

ETA/ETB agonist

1165Somatostatin 1-28

sst receptor agonist

1166CCK Octapeptide, sulfated

C-terminal octapeptide of CCK

1167Leupeptin hemisulfate

Inhibits trypsin-like/cysteine proteases

1168[Leu31,Pro34]-Neuropeptide Y (porcine)

NPY Y1 receptor agonist

1169CGRP 8-37 (rat)

CGRP1 receptor antagonist


Selective μ agonist

1172[Ac-Tyr1,D-Phe2]GRF 1-29, amide (human)

VIP receptor antagonist

1173Neuropeptide Y (porcine)

Influences feeding and sexual behavior

1174Sarafotoxin S6b

Endothelin receptor agonist; non-selective

1175Sarafotoxin S6c

Selective ETB agonist

1176[Leu31,Pro34]-Neuropeptide Y (human, rat)

NPY Y1 receptor agonist

1177Neuropeptide Y 13-36 (porcine)

NPY Y2 receptor agonist

1178[Sar9,Met(O2)11]-Substance P

Potent, selective NK1 agonist

1179Galanin (1-30) (human)

Endogenous galanin receptor agonist

1180[D-Ala2]-Deltorphin II

Selective δ agonist peptide

1181CGRP 8-37 (human)

CGRP1 receptor antagonist

1182VIP (guinea pig)

Involved in neurotransmission and smooth muscle relaxation

1183PACAP 1-27

Potent stimulator of adenylyl cyclase

1184α-helical CRF 9-41

CRF receptor antagonist

1185Thrombin Receptor Agonist Peptide

Causes platelet aggregation and secretion

1186PACAP 1-38

Potent stimulator of adenylyl cyclase


Selective ETA antagonist


Selective ETB agonist

1190Pepstatin A

Aspartic protease inhibitor

1191Amyloid β-Peptide (1-40) (human)

Amyloid β-protein fragment


Activates Gi and Go


Inhibits Gs and stimulates Gi activity

1194MDL 29,913

Selective NK2 antagonist


ETB antagonist


Highly selective ETB agonist


Selective ETB agonist

1198Nocistatin (human)

Human putative counterpart of nocistatin

1199NF 279

Potent and selective P2X1 antagonist

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