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Displaying products by catalog number (1000 - 1099)

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Product Name / Activity
1000ZD 7288

Inhibits pacemaker (If) current

1001Chlorisondamine diiodide

Nicotinic antagonist; slow offset

1002L-745,870 trihydrochloride

Highly selective D4 antagonist


High affinity D2 antagonist

1004L-741,742 hydrochloride

Highly selective D4 antagonist

1006BMY 7378 dihydrochloride

Selective α1D antagonist


5-HT2C antagonist


Group I/group II mGlu antagonist

1014QX 314 bromide

Na+ channel blocker

1015RS 16566 dihydrochloride

5-HT3 ligand. Also shows affinity for zacopride binding site

1017Anandamide (in Tocrisolve™ 100)

Endogenous CB receptor agonist (in water-soluble emulsion)

1018LY 225910

Potent CCK2 antagonist

1019LY 235959

Competitive NMDA antagonist

1024CGP 20712 dihydrochloride

Highly potent and selective β1 antagonist

1025Nisoxetine hydrochloride

Noradrenalin re-uptake inhibitor


Potent group I mGlu antagonist


Selective non-competitive mGlu1 receptor antagonist

1029Methyllycaconitine citrate

α7 neuronal nicotinic receptor antagonist

1030Guanfacine hydrochloride

α2A agonist

1031Piribedil dihydrochloride

Dopamine agonist

1032CP 93129 dihydrochloride

5-HT1B agonist

1033Fluvoxamine maleate

5-HT re-uptake inhibitor


MT2 antagonist


Melatonin agonist

1036ZM 241385

Potent, highly selective A2A antagonist

1037PD 153035 hydrochloride

EGFR-kinase inhibitor

1038WIN 55,212-2 mesylate

Highly potent cannabinoid receptor agonist


Selective GABAA-ρ antagonist


Activator of epithelial KCa channels

1042N-Methyllidocaine iodide

Enhances biosynthesis of phosphatidylinositol

1043QX 222

Na+ channel blocker

1044NBQX disodium salt

Potent AMPA antagonist. More water soluble form of NBQX (Cat. No. 0373)

1045CNQX disodium salt

Potent AMPA/kainate antagonist. More water soluble form of CNQX (Cat. No. 0190)


PDE3/4 inhibitor

1047ICI 182,780

Estrogen receptor antagonist


Modulates AMPA-mediated responses


mGlu5 selective agonist

1050RS 102221 hydrochloride

Selective 5-HT2C antagonist

1051Zinterol hydrochloride

Selective β2 agonist

1052A 61603 hydrobromide

α1A agonist

1053RJR 2403 oxalate

α4β2 selective nicotinic agonist

1054GR 55562 dihydrochloride

5-HT1B antagonist


Potent and selective μ agonist


Potent and selective μ agonist

1057WIN 64338 hydrochloride

Bradykinin B2 antagonist

1059BW 723C86 hydrochloride

5-HT2B agonist


β3 partial agonist. More active enantiomer of pindolol (Cat. No. 0994)

1061(-)-Quinpirole hydrochloride

Selective D2-like agonist

10622-Methylthioadenosine triphosphate tetrasodium salt

P2 purinergic agonist

1063CGS 21680 hydrochloride

A2A agonist

1064Methysergide maleate

5-HT1/5-HT2 antagonist

1065PD 168077 maleate

High affinity, selective D4 agonist


A3 selective agonist

1067Oxotremorine M

Muscarinic agonist


Tachykinin NK3 agonist

1069Tetrodotoxin citrate

Na+ channel blocker; citrate salt of tetrodotoxin (Cat. No. 1078)

1070Zolantidine dimaleate

Potent, centrally active H2 antagonist

1071Pirenzepine dihydrochloride

Selective M1 muscarinic antagonist

1072AGN 192403 hydrochloride

I1 selective ligand


Selective group II antagonist

1074(RS)-AMPA hydrobromide

Selective AMPA agonist. More water soluble form of (RS)-AMPA (Cat. No. 0169)


Ca2+ channel blocker (L-type)


Na+/K+ ATPase inhibitor

1077(-)-Lobeline hydrochloride

Nicotinic partial agonist


Na+ channel blocker

1079(+)-SK&F 10047 hydrochloride

σ1 selective agonist

1080(R)-(+)-8-Hydroxy-DPAT hydrobromide

Selective 5-HT1A agonist. Enantiomer of 8-Hydroxy-DPAT hydrobromide (Cat. No. 0529)

1081SKF 89976A hydrochloride

Potent GABA uptake inhibitor. Penetrates blood brain barrier


Non-competitive AMPA antagonist

1084ω-Conotoxin MVIIC

Ca2+ channel blocker (N, P and Q-type)

1085ω-Conotoxin GVIA

Ca2+ channel blocker (N-type)


KCa channel blocker (big conductance)


KCa channel blocker (big conductance)

1088CGP 54626 hydrochloride

Potent, selective GABAB antagonist

10898-Bromo-cGMP, sodium salt

cGMP analog; activates PKG

1091BU 226 hydrochloride

Potent, highly selective I2 ligand


Selective nociceptin receptor agonist


Antifibrotic agent; regulates cytokine levels in vivo


Benzodiazepine agonist

1095(R)-(-)-Deprenyl hydrochloride

MAO-B inhibitor


Promotes assembly and inhibits disassembly of microtubules


Antiallergic; inhibits inflammatory mediator release from mast cells


Adenylyl cyclase activator

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