All Products

Displaying products alphabetically by name (U)

Product Name / Activity
4540U 104

Potent carbonic anhydrase (CA) IX and XII inhibitor

1638U 18666A

Inhibitor of Hedgehog (Hh) signaling. Also inhibits cholesterol synthesis

1932U 46619

Potent, stable thromboxane A2 (TP) receptor agonist

1268U 73122

Phospholipase C inhibitor

4133U 73343

Analog of U 73122 (Cat. No. 1268)

2734U 89843A

Positive allosteric modulator of GABAA receptors

2733U 90042

GABAA receptor ligand

2745U 93631

GABAA receptor antagonist

1357U 99194 maleate

Potent, selective D3 antagonist


Inactive analog of U0126 (Cat. No. 1144)


Potent, selective inhibitor of MEK1 and 2

0496(-)-U-50488 hydrochloride

Standard selective κ agonist. More active enantiomer of (±)-U-50488 (Cat. No. 0495)

0471(+)-U-50488 hydrochloride

Standard selective κ agonist. Less active enantiomer of (±)-U-50488 (Cat. No. 0495)

0495(±)-U-50488 hydrochloride

Standard selective κ agonist

0498U-54494A hydrochloride

κ agonist

4286UA 62784

Inhibits microtubule polymerization

4954UAMC 00039 dihydrochloride

Dipeptidyl peptidase II (DPP-II) inhibitor

1348UB 165 fumarate

Subunit selective nAChR agonist

1765UBP 282

AMPA/kainate antagonist; distinguishes between motoneuron and dorsal root kainate receptors

2078UBP 296

Selective, potent kainate antagonist; selective for GluR5-containing receptors

1766UBP 301

Kainate receptor antagonist

2079UBP 302

Potent and selective kainate antagonist; active enantiomer of UBP 296 (Cat. No. 2078)

3621UBP 310

GLUK5 antagonist


Group III mGlu antagonist

5251UC 112

IAP and XIAP inhibitor; antitumor

2757UCB 35625

Potent CCR1 and CCR3 antagonist

1310UCL 1684

Highly potent blocker of KCa2

2661UCL 2077

Slow afterhyperpolarization (sAHP) channel blocker; sub-type selective Kv channel effects

1966UCM 707

Potent anandamide transport inhibitor

3490UCPH 101

Selective non-substrate EAAT1 inhibitor

3111UDP disodium salt

Endogenous ligand; competitive antagonist at P2Y14 receptors

5588UF 010

Class I HDAC inhibitor

2529UFP 803

Urotensin-II (UT) antagonist


Potent, selective silent antagonist for NOP

0775(+)-UH 232 maleate

D2 autoreceptor antagonist. Also D3 partial agonist

0425UK 14,304

α2 agonist

2466UK 14,304 tartrate

α2 agonist. Water-soluble form of UK 14,304 (Cat. No. 0425)

4187UK 356618

Potent and selective MMP-3 inhibitor

2900UK 370106

Highly selective MMP-3 and MMP-12 inhibitor

4188UK 383367

Potent and selective BMP-1 (PCP) inhibitor

4186UK 5099

MCT inhibitor; also inhibits of pyruvate transport

3829UK 78282 hydrochloride

Blocker of KV1.3 and KV1.4 channels

5518UMB 68

GHB receptor ligand

3861UNC 0224

Potent G9a and GLP inhibitor

4343UNC 0638

Selective G9a and GLP inhibitor

5132UNC 0642

Potent and selective G9a and GLP inhibitor

4342UNC 0646

Potent and selective G9a and GLP inhibitor

4666UNC 1215

Potent inhibitor of L3MBTL3 Kme reader domain; cell permeable

4904UNC 1999

Potent and selective EZH2/EZH1 inhibitor

5057UNC 2327

Allosteric inhibitor of PRMT3

4930UNC 2399

Biotinylated UNC 1999 (Cat.No. 4904)

4905UNC 2400

Negative control of UNC 1999 (Cat. No. 4904)

5271UNC 3230

Potent and selective PIP5K1C inhibitor; antinociceptive

4516UNC 926 hydrochloride

L3MBTL1 domain inhibitor

3736UPF 1069

PARP-2 inhibitor

4926UPF 648

Potent kynurenine 3-monooxygenase (KMO) inhibitor


Selective and competitive urotensin II receptor antagonist

1772Urapidil hydrochloride

α1 antagonist. Also 5-HT1A receptor agonist

4612URB 597

Potent and selective FAAH inhibitor

6020URB 602

Non-competitive MAGL inhibitor


Used to solubilize and denature proteins

1604Urocortin (human)

Endogenous CRF agonist

1605Urocortin (rat)

Endogenous CRF agonist

1642Urotensin II (human)

Endogenous vasoactive agonist for the UT receptor


Urotensin-II (UT) receptor antagonist

3279UTPγS trisodium salt

Selective P2Y2/4 agonist

3303UVI 3003

RXR antagonist

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