All Products

Displaying products alphabetically by name (T)

Product Name / Activity
1676T 0156 hydrochloride

Highly potent, selective PDE5 inhibitor

2373T 0901317

Potent liver X receptor (LXR) agonist; also CAR inverse agonist

5269T 5601640

Selective LIMK2 inhibitor; antitumor

2519T 98475

GnRH receptor antagonist

2301T 0070907

Highly potent and selective PPARγ antagonist

4538T16Ainh - A01

Ca2+-activated Cl- channel transmembrane protein 16A (TMEM16A) inhibitor


PCNA inhibitor

5383TA 01

Induces cardiomyocyte differentiation from hESCs

5384TA 02

Induces cardiomyocyte differentiation from hESCs

2308Tabimorelin hemifumarate

Potent, orally active ghrelin receptor agonist


GABAA agonist. Also GABA-T substrate and GABA uptake inhibitor


Synthetic vitamin D3 (Cat. No. 4156) analog

0965Tacrine hydrochloride

Cholinesterase inhibitor


Potent and highly selective PDE5 inhibitor; orally bioavailable

3599TAK 165

Potent and selective ErbB2 inhibitor

5209TAK 21d

Potent FAAH inhibitor

4254TAK 715

Potent p38 MAPK inhibitor; anti-inflammatory

5403TAK 960 hydrochloride

Potent and selective PLK1 inhibitor


Non-competitive AMPA/kainate antagonist


CaCC blocker and Cl-/HCO3- exchange inhibitor

3145Talopram hydrochloride

Potent, selective inhibitor of noradrenalin transporters

4352Talsupram hydrochloride

Selective inhibitor of noradrenalin transporters


Synthetic thyrotropin-releasing hormone analog

4506TAME hydrochloride

Ubiquitin ligase APC/C inhibitor; promotes Cdc20 autoubiquitination

0999Tamoxifen citrate

Estrogen receptor partial agonist/antagonist

54415-TAMRA SE

Fluorescent reagent for the labeling of amines

3050Tamsulosin hydrochloride

Selective α1A antagonist

2854Tandospirone hydrochloride

Selective 5-HT1A partial agonist

4426Tanshinone IIA

Inhibits NF-κB and AP-1 DNA binding. Displays antioxidant properties

5757Tariquidar dihydrochloride

Potent P-glycoprotein (P-gp) inhibitor

4521TAS 301

Inhibitor of smooth muscle cell migration and proliferation

5729TASP 0390325

Potent and selective V1B receptor antagonist; orally bioavailable

5362TASP 0433864

Selective mGlu2 receptor positive allosteric modulator

4811TAT 14

Nrf2 pathway activator; blocks Nrf2/Keap1 interaction


Cx43 hemichannel blocker


Non-selective, endogenous glycine receptor partial agonist


Selective PP1 inhibitor


Promotes assembly and inhibits disassembly of microtubules


Receptor-selective retinoid; binds RAR-β and -γ

2905TB 21007

α5-selective GABAA inverse agonist


Selective cell-permeable CK2 inhibitor


Selective CK2 inhibitor


Selective non-transportable inhibitor of EAATs

2669TC 1

High affinity σ1 ligand

4300TC 14012

CXCR4 antagonist; ACKR3 (CXCR7) agonist

2518TC 1698 dihydrochloride

α7-selective agonist

2737TC 2559 difumarate

Selective partial agonist at α4β2 receptors

6105TC AC 28

High affinity BET bromodomain ligand

5412TC AQP1 1

Aquaporin 1 (AQP1) channel blocker

4825TC ASK 10

Potent and selective ASK1 inhibitor; orally bioavailable

4575TC HSD 21

Potent and selective 17β-hydroxysteroid dehydrogenase type 3 inhibitor

4708TC LPA5 4

LPA5 receptor antagonist

4750TC Mps1 12

Potent and selective Mps1 kinase inhibitor

5087TC NTR1 17

Selective non-peptide NTS1 agonist

4625TC OT 39

Potent non-peptide oxytocin receptor partial agonist; also V1a receptor antagonist

4066TC-A 2317 hydrochloride

Potent, selective Aurora kinase A inhibitor


Potent, high affinity 5-HT2A agonist

4345TC-C 14G

Potent, high affinity CB1 receptor inverse agonist

4301TC-DAPK 6

Potent and selective inhibitor of DAPK1

5049TC-E 5001

Potent tankyrase inhibitor

5089TC-E 5002

Selective KDM2/7 inhibitor

5099TC-E 5003

Selective PRMT1 inhibitor

4572TC-E 5005

Potent and selective PDE10A inhibitor

4898TC-E 5006

γ-secretase modulator; reduces Aβ42 levels

5204TC-E 5007

Irreversible and selective dipeptidyl peptidase 8 and 9 (DPP-8/9) inhibitor

5244TC-E 5008

Selective mutant isocitrate dehydrogenase 1 (mIDH1) inhibitor; phenotypically lethal

4355TC-F 2

Potent, reversible and selective FAAH inhibitor

4624TC-FPR 43

Potent FPR2 agonist

5021TC-G 1000

Potent and selective α2D agonist

4879TC-G 1001

GPR35 agonist; more potent than zaprinast (Cat. No. 0947)

5080TC-G 1003

High affinity somatostatin sst2 receptor agonist

4407TC-G 1004

Potent and selective A2A antagonist

5129TC-G 1005

Potent and selective GPBA receptor (TGR5) agonist

4747TC-G 1006

Potent and selective sphingosine-1-phosphate receptor 1 (S1P1) agonist

5355TC-G 1008

Potent and selective GPR39 agonist

4353TC-G 24

Potent and selective GSK-3β inhibitor

4270TC-H 106

Class I histone deacetylase inhibitor

4527TC-I 15

Potent α2β1 inhibitor; displays antithrombotic activity in vivo

4632TC-I 2000

TRPM8 blocker

5410TC-I 2014

Potent TRPM8 antagonist


Selective ubiquitin C-terminal hydrolase-L3 (UCH-L3) inhibitor

4365TC-MCH 7c

Selective melanin-concentrating hormone receptor 1 (MCH1R) antagonist

4435TC-N 1752

NaV channel blocker

4154TCN 201

Selective NR1/NR2A receptor antagonist

4163TCN 213

NMDA antagonist; selective for NR2A over NR2B

4370TC-N 22A

Potent, selective mGlu4 positive allosteric modulator

4072TCN 237 dihydrochloride

Highly potent and selective NR2B antagonist

4259TCN 238

Positive allosteric modulator of mGlu4

4255TC-O 9311

Potent and selective GPR139 agonist

4386TC-P 262

Selective P2X3, P2X2/3 antagonist


Constitutive androstane receptor agonist

3818TCS 1102

Potent, dual orexin receptor antagonist

3942TCS 1105

GABAA α2 benzodiazepine receptor agonist

3941TCS 1205

Subtype-selective GABAA receptor agonist

2236TCS 183

Fragment 1-13 of GSK-3β sequence

2320TCS 184

Scrambled control peptide for use with TCS 183 (Cat. No. 2236)

3869TCS 2002

Potent GSK-3β inhibitor

4221TCS 21311

Potent JAK3 inhibitor. Also inhibits GSK-3β and PKC

3877TCS 2210

Inducer of neuronal differentiation in MSCs

3038TCS 2312

Potent Chk1 inhibitor

3900TCS 2314

α4β1 (VLA-4) antagonist

4069TCS 2510

Selective EP4 agonist

4244TCS 3035

GPR35 agonist

2591TCS 359

Potent FLT3 inhibitor

2754TCS 401

Selective inhibitor of PTP1B

2782TCS 46b

Orally active, subtype-selective NR1A/NR2B antagonist

3938TCS 5861528

TRPA1 blocker

4961TC-S 7001

Potent and highly selective ROCK inhibitor; orally active

3567TC-S 7003

Potent Lck inhibitor

5088TC-S 7004

Potent and selective DYRK1A/B inhibitor

4459TC-S 7005

Potent and selective PLK2 inhibitor

5240TC-S 7006

Potent and selective Tpl2 (Cot; MAP3K8) inhibitor

5243TC-S 7009

High affinity and selective HIF-2α inhibitor

5286TC-S 7010

Potent and selective Aurora kinase A inhibitor

4465TCS ERK 11e

Potent and selective ERK2 inhibitor

4805TCS HDAC6 20b

Selective HDAC6 inhibitor

2827TCS JNK 5a

Selective inhibitor of JNK2 and JNK3

3222TCS JNK 6o

Selective JNK inhibitor

3371TCS OX2 29

Potent and selective OX2 antagonist

2979TCS PIM-1 1

Selective, ATP-competitive Pim-1 kinase inhibitor

3714TCS PIM-1 4a

Selective, ATP-competitive Pim kinase inhibitor

3238TCS PrP Inhibitor 13

Antiprion agent; potently inhibits PrP-res accumulation

4363TC-SP 14

Potent S1P1 receptor agonist

5100TC-T 6000

Potent equilibrative nucleoside transporter 4 (ENT4) inhibitor


PAD4 inhibitor

6092TDZD 8

Selective non-ATP competitive inhibitor of GSK 3β


5-, 12-, 15-Lipoxygenase inhibitor

4613Tegaserod maleate

5-HT4 partial agonist

3664Teijin compound 1

Potent CCR2b antagonist

1122Telenzepine dihydrochloride

Potent, selective M1 antagonist


AT1 antagonist; PPARγ partial agonist


DNA-methylating antitumor agent


Superoxide scavenger; antioxidant


mTOR inhibitor; antitumor


NSAID, cyclooxygenase (COX-1) inhibitor. Also opener of KIR2.3


Reverse transcriptase inhibitor


Protects against MDM2-mediated p53 degradation

1506Terazosin hydrochloride

α1 and α2B antagonist (α1 > α2B). Orally active


H1 antagonist. Also KV11.1 (hERG) and Kir6 (KATP) channel blocker


Dihydroorotate dehydrogenase inhibitor

1405(-)-Terreic acid

Selective inhibitor of BTK

4339Tertiapin LQ

Selective Kir1.1 blocker; derivative of tertiapin-Q (Cat. No. 1316)


Selective blocker of inward-rectifier K+ channels


PPARα/γ agonist


Endogenous androgen receptor agonist


Potent inhibitor of vesicular monoamine transport

5537Tetrabenazine - d7

Deuterated tetrabenazine (Cat. No. 2175)

3068Tetraethylammonium chloride

Non-selective K+ channel blocker


Highly potent NMDA receptor agonist

0723Tetrindole mesylate

MAO-A inhibitor


Na+ channel blocker


Potent and selective Nav1.6 channel blocker

1069Tetrodotoxin citrate

Na+ channel blocker; citrate salt of tetrodotoxin (Cat. No. 1078)


High affinity EAAT1 and EAAT2 blocker

5108TFC 007

Potent hematopoietic prostaglandin D synthase (H-PGDS) inhibitor


PAR1-activating peptide


Selective androgen receptor modulator (SARM)

4336TG 003

Potent inhibitor of Clk-family kinases; also inhibits DYRK1A/B

4264TG 100713

PI 3-kinase inhibitor

5052TG 4-155

High affinity and selective EP2 receptor antagonist

5425TGN 020

Aquaporin 4 (AQP4) channel blocker

5832TGX 221

Potent and selective PI 3-kinase β inhibitor

6191TH 1020

Toll-like receptor (TLR) 5/Flagellin complex antagonist


Binds cereblon, inhibiting ubiquitin ligase activity; alsoTNF-a synthesis inhibitor


Potent inhibitor of SERCA ATPase


Potent subtype-selective ligand; ERα agonist/ERβ antagonist


Glutamate receptor ligand


Adenosine receptor antagonist; bronchodilator

4390Thiamet G

Potent O-GlcNAcase inhibitor


Improves the efficiency of fibroblast reprogramming and induction of iPSCs


Anticancer and immunosuppressive agent


Bacterial RNA polymerase inhibitor


H3 antagonist and H4 inverse agonist

3070Thioridazine hydrochloride

Dopamine receptor antagonist; antipsychotic


Antibiotic, inhibits protein synthesis

32802-ThioUTP tetrasodium salt

Potent and selective P2Y2 agonist

0807THIP hydrochloride

GABAA agonist


Potent and selective MC4 receptor agonist

1185Thrombin Receptor Agonist Peptide

Causes platelet aggregation and secretion

3390Thymosin β4

Potent actin polymerization regulator

4256Tiagabine hydrochloride

GABA uptake inhibitor; anticonvulsant

1972Tianeptine sodium salt

Selective facilitator of 5-HT uptake; antidepressant

3931Ticlopidine hydrochloride

Selective P2Y12 antagonist


Potent and selective breast tumor kinase (Brk) inhibitor

0649(S)-Timolol maleate

β1 antagonist

0747Tin protoporphyrin IX dichloride

Heme oxygenase inhibitor


Potent, selective H2 antagonist

5902Tiotropium bromide

Potent muscarinic receptor antagonist


Plasminogen activator inhibitor-1 (PAI-1) inhibitor

3609Tizanidine hydrochloride

α2 agonist

3051TLQP 21

VGF-derived peptide

5769TM 5275 sodium salt

Plasminogen activator inhibitor-1 (PAI-1) inhibitor; orally bioavailable

6194TM 5441

Plasminogen activator inhibitor-1 (PAI-1) inhibitor


Dual-kinase inhibitor; inhibits CK2 and ERK8

5960TMI 1

Adam 17 (TACE) and MMP inhibitor; orally bioavailable

4152TMN 355

Cyclophilin A inhibitor

2438TMPH hydrochloride

Neuronal nicotinic receptor antagonist

4253TMPyP4 tosylate

Inhibitor of human telomerase


Cytochrome P450 1B1 inhibitor


Inhibitor of IP6K; also inhibits IP3K

2464TNP-ATP triethylammonium salt

Potent, selective P2X antagonist


Aminoglycoside antibiotic


Potent PDGFR and VEGFR inhibitor

2540Tocrifluor T1117

Fluorescent cannabinoid ligand; fluorescent form of AM 251 (Cat. No. 1117)

5268Tocriscreen Epigenetics Toolbox

80 Epigenetic modulators supplied pre-dissolved in DMSO (250 μL 10 mM solutions)

5933Tocriscreen Kinase Inhibitor Toolbox I

A library of 80 kinase inhibitor compounds (250 μL 10 mM DMSO solutions)

6268Tocriscreen Kinase Inhibitor Toolbox I & II

A library of 160 kinase inhibitor compounds (250 μL 10 mM DMSO solutions)

6225Tocriscreen Kinase Inhibitor Toolbox II

A library of 80 kinase inhibitor compounds (250 μL 10 mM DMSO solutions)

5932Tocriscreen Library of FDA-Approved Compounds

A library of 160 FDA-approved compounds (250 μL 10 mM DMSO solutions)

5840Tocriscreen Plus

A library of 1280 biologically active compounds (250 μL 10mM DMSO solutions)

5841Tocriscreen Plus Mini

A library of 1280 biologically active compounds (50 μL 10mM DMSO solutions)

5060Tocriscreen Stem Cell Toolbox

80 Stem Cell modulators supplied pre-dissolved in DMSO (250 μL 10 mM solutions)

1684Tocrisolve™ 100

Water-soluble emulsion; negative control for reagents in TocrisolveTM 100


COMT inhibitor; also inhibits transthyretin aggregation

3761Tolterodine L-tartrate

Potent, non-selective muscarinic receptor antagonist


Potent and selective vasopressin V2 receptor antagonist; renoprotective and orally active

5527Tomoxetine - d3 hydrochloride

Deuterated tomoxetine (Cat. No. 2011)

2011Tomoxetine hydrochloride

Potent, selective noradrenalin re-uptake inhibitor


GluR5 antagonist; inhibits carbonic anhydrase (CA) II and IV

5541Topiramate - d12

Deuterated topiramate (Cat. No. 3620)

4562Topotecan hydrochloride

DNA topoisomerase I inhibitor; Camptothecin (Cat. No. 1100) analog


Inhibitor of cholesteryl ester transfer protein (CETP)

4247Torin 1

Potent and selective mTOR inhibitor

4248Torin 2

Potent and selective mTOR inhibitor


Adenosine analog; antifungal antibiotic

4414TP 003

Functionally selective GABAA receptor (α3 subtype) partial agonist

6008TP 064

Potent and selective PRMT 4 inhibitor

6000TP 472

Potent BRD9/7 inhibitor

5999TP 472N

Negative control for TP 472 (Cat. No. 6000).


Potent, selective inhibitor of IKKβ


Cell-permeable Zn2+ chelator


Selective GABAA-ρ antagonist


High affinity PKC activator; also APP modulator


Potent soluble epoxide hydrolase inhibitor; orally bioavailable and brain penetrant


Positive allosteric modulator of α7 nAChRs

1558Tracazolate hydrochloride

Subtype-selective GABAA allosteric modulator

2946TRAM 34

Potent and highly selective KCa3.1 channel blocker

4952TRAM 39

Potent KCa3.1 blocker


Targets soluble Aβ to decrease amyloid plaque deposition. Also GABA analog


Antiallergic; inhibits inflammatory mediator release from mast cells

3852Tranylcypromine hydrochloride

Irreversible inhibitor of LSD1; also inhibits MAO

2508Trap 101

Potent and selective NOP antagonist; active in vivo


PAR1 peptide fragment (residues 42-47); acts as a PAR1 agonist


Potent and selective FP prostaglandin receptor agonist

4734TRC 051384

Inducer of heat shock protein Hsp70


Potent prostacyclin (PGI2) analog

2337Trequinsin hydrochloride

Extremely potent inhibitor of PDE3

2472Triacsin C

Inhibitor of acyl-CoA synthetase

1406Trichostatin A

Potent histone deacetylase inhibitor


Electrophoresis buffer


Thymidylate synthase inhibitor; induces DNA fragmentation


nNOS/iNOS inhibitor


Aryl hydrocarbon receptor antagonist

0662trans-Triprolidine hydrochloride

Standard H1 antagonist, highly potent


Inhibits RNAPII-mediated transcription; antitumor, anti-inflammatory and immunosuppressive

3163TRIS base

Commonly used laboratory reagent

3164TRIS hydrochloride

Commonly used laboratory reagent


Potent, selective inhibitor of mitotic kinesin Eg5

2906TRO 19622

Binds voltage-dependent anion channel (VDAC)


Selective PPARγ agonist; antidiabetic agent


Antioxidant vitamin E derivative


5-HT3 antagonist


Selective M4 muscarinic antagonist

2459Tropisetron hydrochloride

Potent 5-HT3 receptor antagonist; also partial agonist of α7 nAChR

3863Trovafloxacin mesylate

Antibiotic; inhibits bacterial DNA synthesis

4639TT 232

sst1/sst4 somatostatin receptor agonist


Retinoic acid analog; RAR agonist

4432TTP 22

High affinity, selective CK2 inhibitor


HDAC6 inhibitor; inhibits α-tubulin deacetylation

6270Tubastatin A hydrochloride

Potent HDAC6 inhibitor

2820(+)-Tubocurarine chloride

Nicotinic receptor antagonist

4601TUG 891

Potent and selective FFA4 (GPR120) agonist


Antibiotic; GlcNAc phosphotransferase inhibitor

4038TW 37

Bcl-2 inhibitor; induces apoptosis

3835TWS 119

GSK-3β inhibitor; induces neuronal differentiation in ESCs

5328TY 52156

S1P3 receptor antagonist

0578Tyrphostin B44, (-) enantiomer

EGFR-kinase inhibitor

0579Tyrphostin B44, (+) enantiomer

EGFR-kinase inhibitor

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