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Displaying products alphabetically by name (P)

Product Name / Activity
4485P 22077

USP7 inhibitor


USP7 inhibitor


Protein disulfide isomerase (PDI) inhibitor


Potent Kir6 (KATP) channel opener


Potent antagonist of αvβ3-vitronectin interaction; antiangiogenic

1902[Ala92]-p16 (84-103)

Cyclin-dependent kinase inhibitor

2244p38 MAPK Inhibitor Tocriset™

Selection of 3 p38 MAPK inhibitors (Cat. Nos. 1264, 1202 and 1962)


Sialic acid analog; sialyltransferase inhibitor


NAMPT activator; also proneurogenic and neuroprotective

5463PA 1 dihydrochloride

Photoswitchable ENaC blocker

5086PA 452

RXR antagonist


Antagonist of neurosteroid potentiation and direct gating of GABAA

2581PAC 1

Activator of procaspase-3; pro-apoptotic

1183PACAP 1-27

Potent stimulator of adenylyl cyclase

1186PACAP 1-38

Potent stimulator of adenylyl cyclase

3236PACAP 6-38

Potent PAC1 receptor antagonist

5116PACMA 31

Irreversible protein disulfide isomerase (PDI) inhibitor


Phospholipase A2 inhibitor

2940PAF (C16)

Endogenous platelet-activating factor (PAF)


Endogenous lipid; potentiates effects of endovanilloids at TRPV1 receptors


Atypical antipsychotic; 5-HT2A and D2 antagonist

0609(±)-Palmitoylcarnitine chloride

Intermediate in fatty acid oxidation


Selective GPR55 agonist. FAAH and PAA substrate


Endogenous lipid; enhances activity of 2-arachidonylglycerol (Cat. No. 1298)


Inhibitor of FAAH


TLR2/6 agonist; induces TNF-α production

4638Pam2CSK4 Biotin

Biotinylated Pam2CSK4 (Cat. No. 4637)


TLR1/2 agonist; induces cytokine production

4636Pam3CSK4 Biotin

Biotinylated Pam3CSK4 (Cat. No. 4633)

4298Pamoic acid disodium salt

GPR35 agonist

1154Pancreatic Polypeptide (human)

NPY Y4 agonist; involved in gastrointestinal tract function

1365[cPP1-7,NPY19-23,Ala31,Aib32,Gln34] - hPancreatic Polypeptide

Potent, selective NPY Y5 agonist

0693Pancuronium dibromide

Nicotinic (neuromuscular) antagonist


Dopamine D2 receptor allosteric modulator


Reversible inhibitor of MKLP-2

3011Parathyroid hormone (1-34) (human)

Parathyroid hormone (PTH) receptor agonist


Analog of the active form of vitamin D2

2141Paroxetine maleate

Highly potent and selective 5-HT uptake inhibitor

3553Parstatin (human)

Peptide cleaved from PAR1 upon receptor activation

3554Parstatin (mouse)

Peptide cleaved from PAR1 upon receptor activation


5-HT release inhibitor


SERCA ATPase blocker. Also potent BKCa channel blocker

2562PB 28 dihydrochloride

High affinity σ2 agonist


JARID1 (Jumonji AT-Rich Interactive Domain 1) inhibitor

4611PBP 10

Selective FPR2 antagonist; cell permeable

5564PBS, 100 Tablets

PBS Tablets

0571PCA 4248

PAF receptor antagonist

5012PCI 29732

Potent BTK inhibitor

4643PCI 34051

Potent and selective HDAC8 inhibitor

5871pCPA methyl ester hydrochloride

Tryptophan hydroxylase inhibitor


Selective Epac activator; cell-permeable analog of 8CPT-2Me-cAMP (Cat. No. 1645)

4192PD 0325901

Potent inhibitor of MEK1/2

4786PD 0332991 isethionate

Potent, selective Cdk4/6 inhibitor; brain penetrant

1671PD 102807

Selective M4 antagonist

2830PD 118057

Selective KV11.1 (hERG) channel activator

1361PD 123319 ditrifluoroacetate

Potent, selective non-peptide AT2 antagonist

1243(+)-PD 128907 hydrochloride

D3 agonist (D3 ≥ D2 > D4)

2608PD 135158

Potent and selective CCK2 antagonist

2606PD 144418 oxalate

High affinity, selective σ1 ligand

2850PD 146176

Selective 15-lipoxygenase inhibitor

1269PD 150606

Cell permeable calpain inhibitor

1037PD 153035 hydrochloride

EGFR-kinase inhibitor

2615PD 158780

Potent ErbB receptor family inhibitor

2200PD 160170

Selective non-peptide NPY Y1 receptor antagonist

3724PD 161570

Selective FGFR inhibitor

3785PD 166285 dihydrochloride

Potent Src inhibitor; also inhibits FGFR1, PDGFRβ and Wee1

2520PD 166793

Broad spectrum MMP inhibitor

1065PD 168077 maleate

High affinity, selective D4 agonist

3529PD 168568 dihydrochloride

Potent and selective D4 antagonist

3044PD 173074

FGFR1 and -3 inhibitor

3552PD 173212

Potent N-type Ca2+ channel blocker

2602PD 176252

GRP (BB2) and NMB (BB1) receptor antagonist

4965PD 180970

p210Bcr/Abl kinase inhibitor; also inhibits c-Src and KIT

4237PD 184352

Selective MEK inhibitor

2605PD 198306

Selective inhibitor of MEK1/2

4824PD 334581

MEK1 inhibitor

5124PD 404182

High affinity inhibitor of KDO 8-P synthase; also DDAH1 inhibitor

2694PD 407824

Selective inhibitor of Chk1 and Wee1

1363PD 81723

Allosteric potentiator of A1 receptors

5101PD 90780

Inhibits NGF binding to p75NTR

1213PD 98059

MEK inhibitor


Transportable EAAT1-4 inhibitor/non-transportable EAAT5 inhibitor


FAAH activator

2207PDZ1 Domain inhibitor peptide

Disrupts interaction between GluR6 and PSD-95 PDZ1 domain

4086PE 154

Fluorescent, potent AChE and BChE inhibitor

5018PEAQX tetrasodium salt

Potent NMDA receptor antagonist; NR2A selective


CNS stimulant, indirect monoamine agonist

4617Penitrem A

Potent and selective BKCa (KCa1.1) channel blocker

36924,4-Pentamethylenepiperidine hydrochloride

M2 proton channel blocker

3277Pentamidine isethionate

Antimicrobial that antagonizes NMDA receptors


κ-agonist; antinociceptive

4579Pentobarbital sodium salt

Enhances GABAergic activity


Adenosine deaminase inhibitor


PDE inhibitor


Fluorometric cytochrome P450 substrate


CNS stimulant

4054PEP 005

Protein kinase C activator


GluR1 subunit C-terminus peptide analog. Analog of Pep1-TGL (Cat. No. 1601)


GluR1 subunit C-terminus peptide analog


Peptide inhibitor of GluR2 subunit binding to PICK1


Peptide inhibitor of GluR2 subunit binding to PICK1


Peptide inhibitor of GluR2 subunit binding to NSF. Reduces AMPA currents

3801Pep2m, myristoylated

Myristoylated form of pep2m (Cat. No. 1595). Peptide inhibitor of GluR2 subunit binding to NSF


Inactive control peptide for pep2-SVKI (Cat. No. 1597)


Peptide inhibitor of GluR2 subunit binding to GRIP, ABP and PICK1. Increases AMPA current amplitude


Inactive control peptide for pep2m (Cat. No. 1595)


Allosteric potentiator of AMPA receptor desensitization

1190Pepstatin A

Aspartic protease inhibitor

1618Peptide YY (3-36)

Selective NPY Y2 receptor agonist

5166Perhexiline maleate

Carnitine palmitoyltransferase 1 and 2 (CPT1/2) inhibitor

4302Perindopril erbumine

Angiotensin-converting enzyme (ACE) inhibitor


Potent and selective hM3Dq DREADD agonist

4944Peroxy Orange 1

Fluorescent hydrogen peroxide indicator

3097Pertussis Toxin

Catalyzes ADP-ribosylation of Gi, Go and Gt


Activator of caspase-3

4821PF 03814735

Aurora kinase A and B inhibitor

4239PF 04217903 mesylate

Highly selective MET inhibitor

4818PF 04418948

Potent and selective EP2 receptor antagonist

4820PF 04691502

Potent and selective dual PI 3-K/mTOR inhibitor

4916PF 04885614

Potent and selective NaV1.8 channel blocker; active in vivo

5931PF 05089771

Potent and selective Nav1.7 channel blocker

6003PF 05105679

Selective TRPM8 blocker

5790PF 05175157

Acetyl-CoA carboxylase (ACC) 1 and 2 inhibitor

4823PF 05212384

Potent and selective dual PI 3-K/mTOR inhibitor

5752PF 06260933 dihydrochloride

MAP4K4 (HGK) inhibitor; also inhibits MINK and TNIK

6004PF 06281355

Selective myeloperoxidase (MPO) inhibitor

5716PF 06447475

Potent LRRK2 inhibitor; neuroprotective

5640PF 06463922

High affinity and selective ALK and ROS1 inhibitor

4710PF 06465469

Potent ITK inhibitor; also inhibits BTK

4238PF 184

Potent and selective IKKβ inhibitor

5751PF 3084014 hydrobromide

Potent γ-secretase inhibitor

4279PF 3644022

Potent MK2 inhibitor

4191PF 3716556

Selective H+,K+-ATPase inhibitor

4175PF 3845

Selective FAAH inhibitor

3354PF 429242

Competitive inhibitor of SREBP site 1 protease

4278PF 431396

Dual FAK/PYK2 inhibitor

4032PF 4708671

S6K1 inhibitor

4277PF 477736

Selective Chk1 inhibitor

4900PF 4778574

Positive allosteric modulator of AMPA receptors

4281PF 4800567 hydrochloride

Selective casein kinase 1ε inhibitor

4252PF 4981517

Selective CYP3A4 inhibitor

4362PF 5081090

Potent LpxC inhibitor

3676PF 514273

Potent and selective CB1 antagonist

5262PF 5274857 hydrochloride

High affinity and selective Smoothened (Smo) receptor antagonist

5754PF 543 hydrochloride

Potent and selective SphK1 inhibitor

3239PF 573228

Potent and selective FAK inhibitor

5939PF 6274484

High affinity and potent covalent EGFR kinase inhibitor

3316PF 670462

Potent and selective CK1ε and CK1δ inhibitor

3307PF 750

Selective FAAH inhibitor

4078PF 8380

Potent autotaxin inhibitor

3291PF 915275

Potent and selective 11β-hydroxysteroid dehydrogenase inhibitor

5917PF 9184

Potent microsomal prostaglandin E synthase 1 (mPGES-1) inhibitor

4419PF 945863

Macrolide antibiotic

3923PF 998425

Non-steroidal androgen receptor antagonist

5801PF CBP1

Selective CBP/p300 bromodomain inhibitor

4074PF9 tetrasodium salt

Potent GPR17 agonist

4445PFI 1

BET bromodomain inhibitor

4892(R)-PFI 2 hydrochloride

Potent and selective SETD7 inhibitor

5400(S)-PFI 2 hydrochloride

Negative control of (R)-PFI 2 hydrochloride (Cat. No. 4892)

5072PFI 3

Potent and selective SMARCA2/4 and polybromo 1 inhibitor

5576PFI 4

Potent and selective BRPF1 bromodomain inhibitor

5339PFK 15

Selective PFKFB3 inhibitor

3943PG 01

CFTR mutants potentiator

3887PG 01037 dihydrochloride

D3 receptor selective antagonist

4919PG 106

Selective MC3 receptor antagonist

5094PG 931

Potent and selective MC4 receptor agonist

0750PG-9 maleate

Presynaptic cholinergic modulator

5866PH 797804

Potent and selective p38α/β inhibitor

3092PHA 543613 hydrochloride

Potent and selective α7 nAChR agonist

3134PHA 568487

α7-selective agonist

2693PHA 665752

Potent and selective MET inhibitor

3140PHA 767491 hydrochloride

MK2 inhibitor; also inhibits cdc7/cdk9


Weak, selective GABAB antagonist


Promotes actin polymerization


Potent group I mGlu antagonist


Inhibits TRPP3-mediated currents; also inhibits epithelial Na+ channels


Selective TRPM4 blocker

2557Phencyclidine hydrochloride

Non-competitive NMDA receptor antagonist

4578Phenobarbital sodium salt

Enhances GABAergic activity


Cholinesterase inhibitor

09691-Phenylbiguanide hydrochloride

5-HT3 agonist

2682Sodium 4-Phenylbutyrate

Histone deacetylase inhibitor

2838(R)-(-)-Phenylephrine hydrochloride

α1 agonist


Potent melatonin agonist

07304-Phenyl-1,2,3,4-tetrahydroisoquinoline hydrochloride

DA release inhibitor

4326PhiKan 083

p53 stabilizing agent

2770Philanthotoxin 74

GluR1 and GluR3 AMPA receptor antagonist


Na+-glucose cotransporter (SGLT) inhibitor

2080PHM 27 (human)

Potent calcitonin receptor agonist; endogenous analog of human VIP

4153Phorbol 12,13-dibutyrate

Protein kinase C activator

1201Phorbol 12-myristate 13-acetate

Protein kinase C activator


Prodrug of the antitumor agent 5F 203

4325Phosphocreatine disodium salt

Phosphate reservoir

1881Phosphodiesterase Inhibitor Tocriset™

Selection of 5 phosphodiesterase inhibitors (Cat. Nos. 0915, 1504, 0415, 1349 and 1046)

1352Phospho-Glycogen Synthase Peptide-2 (substrate)

Glycogen synthase kinase-3 substrate (synthetic)

57782-Phospho-L-ascorbic acid trisodium salt

Ascorbic acid derivative; maintains differentiation potential in bone marrow-derived MSCs


Group III mGlu agonist

4466PHP 501 trifluoroacetate

Potent GABAA antagonist

4914Phrixotoxin 3

Potent blocker of NaV1.2, NaV1.3 and NaV1.5 channels

4598PHT 427

Dual Akt and PDK1 inhibitor; antitumor


Selective ERβ antagonist

0622Physostigmine hemisulfate

Cholinesterase inhibitor

2930PI 103 hydrochloride

Inhibitor of PI 3-kinase, mTOR and DNA-PK

2814PI 828

PI 3-kinase inhibitor, more potent than LY 294002 (Cat. No. 1130)


Inhibits TNF-induced NF-κB activation


Potent and selective PDE4 inhibitor


Selective IGF1R inhibitor


GABAA receptor antagonist

1267Pifithrin-α hydrobromide

p53 inhibitor. Also aryl hydrocarbon receptor agonist

3843Cyclic Pifithrin-α hydrobromide

p53 inhibitor


Inhibitor of p53-mitochondrial binding


Antibody recognizing PIKfyve

0694Pilocarpine hydrochloride

Muscarinic agonist

3589PIM-1 Inhibitor 2

Pim-1 kinase inhibitor


D2-like antagonist


β3 partial agonist


β3 partial agonist. More active enantiomer of pindolol (Cat. No. 0994)

4124Pioglitazone hydrochloride

Selective PPARγ agonist; antidiabetic agent


σ1 selective ligand


Induces apoptosis; increases p53 and ROS levels in cancer cells


5-HT4 agonist. Also 5-HT3 antagonist

4212PIR 3.5

Negative control of IPA 3 (Cat. No. 3622)


Nootropic; modulates Na+-flux at AMPA receptors

1071Pirenzepine dihydrochloride

Selective M1 muscarinic antagonist


Antifibrotic agent; regulates cytokine levels in vivo

1031Piribedil dihydrochloride

Dopamine agonist

0724Pirlindole mesylate

MAO-A inhibitor


Cyclooxygenase-1 (COX-1) inhibitor


P2Y ligand; displays mixed antagonism/potentiation

4168PIT 1

Inhibits Akt signaling

4942Pitavastatin calcium

HMG-CoA reductase inhibitor

3255PJ 34 hydrochloride

Potent PARP inhibitor

0670PK 11195

Antagonist at peripheral benzodiazepine receptors

4145PK 44 phosphate

Potent and selective dipeptidyl peptidase IV (DPP-IV) inhibitor

1904PKA inhibitor fragment (6-22) amide

Potent protein kinase A inhibitor

1882PKA Tocriset™

Selection of 5 PKA modulators (Cat. Nos. 1337, 1140, 1099, 1288 and 1603)

4058PKC (19-36)

Pseudosubstrate peptide; inhibitor of PKC

4059[Glu27]-PKC (19-36)

Inactive control peptide for PKC (19-36) (Cat. No. 4058)

2992PKC 412

Protein kinase C inhibitor

1792PKC β pseudosubstrate

Selective cell-permeable PKC inhibitor peptide (attached to vector)

1791PKC ζ pseudosubstrate

PKC ζ inhibitor peptide (attached to cell-permeable vector)

2546PKI 14-22 amide, myristoylated

Cell-permeable protein kinase A inhibitor

4941PKI 166 hydrochloride

Potent EGFR-kinase inhibitor


Potent TASK-3 channel blocker

2024PL 017

Selective μ agonist

2567PLP (139-151)

Encephalitogenic myelin proteolipid fragment


Induces G2/M cell cycle arrest; anticancer


Dual ERK1/RasGAP inhibitor. Maintains ESC self-renewal

4847PluriSln 1

SCD-1 inhibitor

5102PLX 647 dihydrochloride

Potent dual Fms/KIT inhibitor

4034PM 102

Antagonist of heparin (Cat. No. 2812)


Potent, selective α1 antagonist

1380PMPA (NAALADase inhibitor)

GCP II inhibitor

2273PMPA (NMDA antagonist)

Competitive NMDA antagonist


Non-selective protease inhibitor; also blocks anandamide metabolism

5196PMX 205

Potent C5a receptor peptide antagonist

4996PMX 464

Putative inhibitor of the Trx-TrxR system; antiproliferative

5473PMX 53

Potent C5a receptor antagonist

5697PMX 53c

Negative control for PMX 53 (Cat. No. 5473)

2556PNU 109291

Potent and selective 5-HT1D agonist

2498PNU 120596

Positive allosteric modulator of α7 nAChR; active in vivo

1985PNU 142633

Highly selective 5-HT1D agonist

3355PNU 177864 hydrochloride

Highly selective D3 antagonist

2201PNU 22394 hydrochloride

5-HT2C agonist and 5-HT2A/2B partial agonist

2303PNU 282987

Selective α7 nAChR agonist

2095PNU 37883 hydrochloride

Vascular Kir6 (KATP) channel blocker

3534PNU 74654

β-catenin binder; inhibits Wnt signaling

2735PNU 96415E

D4 and 5-HT2A antagonist; antipsychotic


TLR3 agonist


TRPA1 channel activator; analgesic and antifungal

3165Polyoxyethylenesorbitan monolaurate

Detergent used for protein extraction

2689POM 1

Inhibitor of E-NTPDases


Slows neuronal Na+ channel inactivation

5225Ponceau S Staining Solution

Stain used to detect protein bands after Western blotting

3147Potassium Chloride

Commonly used laboratory reagent

3150Potassium phosphate monobasic

Commonly used in biological assay buffers

1397PP 1

Potent, selective Src family kinase inhibitor

3894PP 121

Dual kinase inhibitor; inhibits PI 3-K family kinases

1407PP 2

Potent, selective Src family kinase inhibitor

4257PP 242

Dual mTORC1/mTORC2 inhibitor

2794PP 3

Negative control for PP 2 (Cat. No. 1407)

1923pp60 c-src (521-533) (phosphorylated)

Inhibits tyrosine kinase activity of pp60c-src and pp60v-src

0625PPADS tetrasodium salt

P2 purinergic antagonist

0683iso-PPADS tetrasodium salt

P2X antagonist


Non-pungent vanilloid receptor agonist

06204-PPBP maleate

Specific σ ligand, NMDA antagonist

3870(±)-PPCC oxalate

Selective sigma (σ) agonist (σ1> σ2)


Subtype-selective NR2C/NR2D antagonist


MT2 antagonist


Potent, selective mGlu8 agonist


Potent, selective P2X1 antagonist


Competitive NR2A antagonist

4303PPQ 102

Potent, voltage-independent CFTR chloride channel inhibitor


Subtype-selective ERα agonist

4862PPTN hydrochloride

High affinity and selective P2Y14 antagonist

4730PPY A

Potent inhibitor of Abl T315l mutant and wild-type Abl kinases

2768PQ 401

IGF1R inhibitor

5351PQ 69

Potent and selective A1 antagonist/inverse agonist

1947PR 39 (porcine)

IκBα inhibitor

4482PR 619

Broad spectrum DUB inhibitor

4174Pramipexole dihydrochloride

Selective D3 agonist


Synthetic version of amylin (Cat. No. 3418)

2318Pravastatin sodium salt

HMG-CoA reductase inhibitor

0623Prazosin hydrochloride

α1 and α2B antagonist. MT3 antagonist

0589PRE-084 hydrochloride

Highly selective σ1 agonist


Anticonvulsant; selectively binds the α2δ subunit of voltage-sensitive calcium channels


GABAA receptor positive allosteric modulator

5376Pregnenolone sulfate sodium salt

NMDA Potentiator


Restores mutant p53 activity; induces apoptosis


Restores mutant p53 activity


Potentiates GABAA receptor function

3491Prion Protein 106-126 (human)

Prion protein fragment


Potent, reversible MAGL inhibitor


MRP inhibitor


Antioxidant, anti-inflammatory and hypocholesterolemic agent

1102Procaterol hydrochloride

Potent β2 agonist

3287Prochlorperazine dimaleate

D2 receptor antagonist. Also 5-HT3 and nAChR antagonist


Endogenous progesterone receptor agonist

1478Proglumide sodium salt

Non-selective CCK antagonist; orally active


DYRK1A/B inhibitor; prodrug of INDY (Cat. No. 4997)

0829Pronethalol hydrochloride

β antagonist

5135Propidium iodide

Red-fluorescent DNA stain; membrane impermeant to live cells

0611(±)-Propionylcarnitine chloride

Intermediate in lipid metabolism

0624Propranolol hydrochloride

β antagonist

0851Propranolol glycol

Propranolol (Cat. No. 0624) metabolite

0835(R)-(+)-Propranolol hydrochloride

β antagonist. Less active enantiomer of propranolol (Cat. No. 0624)

0834(S)-(-)-Propranolol hydrochloride

β antagonist. More active enantiomer of propranolol (Cat. No. 0624)

1200Nω-Propyl-L-arginine hydrochloride

Highly selective inhibitor of nNOS

5151Prosaptide TX14(A)

Potent GPR37 and GPR37L1 agonist

2296Prostaglandin E2

Major endogenous prostanoid

4214Prostaglandin F2α

Naturally-occurring prostanoid; potent vasoconstrictor

230615-deoxy-Δ-12,14-Prostaglandin J2

Endogenous PPARγ agonist


PKC activator; also NF-κB activator

5500Protease Inhibitor Cocktail I

Protease inhibitor cocktail for mammalian cells

4665ProTx I

CaV3.1 channel blocker; also inhibits NaV1.8 and KV2.1

4023ProTx II

Selective NaV1.7 channel blocker

5792ProTx III

Potent Nav1.7 blocker; analgesic

2477Proxyfan oxalate

High affinity H3 ligand

5047PRT 4165

Inhibitor of Bmi1/Ring1A; blocks histone H2A ubiquitination

4569PS 1145 dihydrochloride

Selective IKK inhibitor; orally active

5042Psalmotoxin 1

Potent and selective ASIC1a channel blocker

2715PSB 0474

Potent and selective P2Y6 agonist

2574PSB 06126

NTPDase 3 inhibitor

2573PSB 069

Non-selective NTPDase inhibitor

3983PSB 0739

Highly potent P2Y12 receptor antagonist

4334PSB 0777 ammonium salt

Potent adenosine A2A agonist

3199PSB 0788

Selective A2B antagonist

2010PSB 10 hydrochloride

Potent, highly selective hA3 receptor antagonist/inverse agonist

2012PSB 11 hydrochloride

Potent, selective hA3 receptor antagonist/inverse agonist

4333PSB 1114

Potent, selective P2Y2 agonist

2009PSB 1115

Selective human A2B receptor antagonist; water-soluble

2019PSB 36

Potent and selective A1 antagonist

3198PSB 603

Highly selective A2B antagonist

4042PSC 833

Inhibitor of P-gp-mediated MDR

1790Pseudo RACK1

Protein kinase C activator peptide (attached to cell permeable vector)


Proteasome inhibitor. Also prevents activation of NF-κB


Non-selective serotonin receptor agonist

3353PSN 375963 hydrochloride

GPR119 receptor agonist


CB1 receptor negative allosteric modulator

4367Psora 4

Potent KV1.3 channel blocker

4039PT 1

AMPK activator

4533PTAC oxalate

Muscarinic receptor ligand; exhibits partial agonist and antagonist activity at different subtypes

5191PTC 209

Bmi-1 inhibitor; antitumor


Potent MMP-3 expression inhibitor; neuroprotective

4700PU 02

Negative allosteric modulator of 5-HT3

3104PU H71

Potent Hsp90 inhibitor


O-GlcNAcase and β-hexosaminidase inhibitor


Smo receptor agonist

4089Puromycin dihydrochloride

Protein synthesis inhibitor

4922Purotoxin 1

Potent P2X3 modulator

1580Purvalanol A

Cyclin-dependent kinase inhibitor

1581Purvalanol B

Cyclin-dependent kinase inhibitor

2954PX 12

Thioredoxin-1 inhibitor

2978PYR 41

Ubiquitin-activating enzyme (E1) inhibitor


Selective TRPC3 blocker


High affinity, partial agonist of α4β2 receptors

4763Pyridostatin pentahydrochloride

Stabilizes G-quadruplexes; induces DNA damage and cell cycle arrest

24782-Pyridylethylamine dihydrochloride

H1 receptor agonist


Potent inhibitor of multidrug and toxin extrusion (MATE) transporters; also DHFR and STAT3 inhibitor


Enhances survival of human ESCs following enzymatic dissociation


Histone deacetylase inhibitor

0727Pyrrolidinedithiocarbamate ammonium

Inhibits NF-κB, prevents increase in NOS mRNA

4994PYZD 4409

Ubiquitin-activating enzyme (E1) inhibitor

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