All Products

Displaying products alphabetically by name (A)

Product Name / Activity
4431A 1070722

Highly potent, selective GSK-3 inhibitor

3793A 1120

High affinity retinol-binding protein 4 (RBP4) ligand

2524A 205804

Selective inhibitor of E-selectin and ICAM-1 expression

4228A 286982

Potent inhibitor of the LFA-1/ICAM-1 interaction

4697A 331440 dihydrochloride

Selective H3 antagonist

2753A 350619 hydrochloride

Soluble guanylyl cyclase (sGC) activator

5163A 366

Potent and selective G9a/GLP inhibitor

4552A 412997 dihydrochloride

Selective D4 agonist

3914A 419259 trihydrochloride

Inhibitor of Src family kinases

5781A 425619

Potent TRPV1 antagonist

2972A 438079 hydrochloride

Competitive P2X7 antagonist

4483A 484954

CaM kinase III (eEF-2 kinase) inhibitor

4341A 582941

Partial agonist at α7 nAChR

1052A 61603 hydrobromide

α1A agonist

1534A 68930 hydrochloride

Potent, selective D1-like agonist

3701A 740003

Potent and selective P2X7 antagonist

3336A 769662

Potent AMPK activator

1701A 77636 hydrochloride

Potent, selective D1-like agonist. Orally active

5937A 779

Selective Mas receptor (Ang-(1-7) receptor) antagonist

4319A 784168

Potent and selective TRPV1 antagonist

2976A 803467

Selective NaV1.8 channel blocker

2341A 80426 mesylate

High affinity α2 antagonist. Also 5-HT uptake inhibitor

4473A 804598

Potent and selective P2X7 antagonist

2939A 83-01

Selective inhibitor of TGF-βRI, ALK4 and ALK7

4232A 839977

Potent P2X7 antagonist

3060A 841720

Selective mGlu1 antagonist

4477A 844606

Selective α7 nAChR partial agonist

5017A 85380 dihydrochloride

High affinity and selective α4β2 agonist

4571A 867744

Positive allosteric modulator of α7 nAChR

4249A 887826

Potent voltage-dependent NaV1.8 channel blocker

3587A 922500

Potent DGAT-1 inhibitor

4845A 939572

Potent SCD-1 inhibitor

3753A 943931 dihydrochloride

Potent and selective H4 antagonist

4716A 967079

Selective TRPA1 channel blocker

5766A 971432

Potent and selective S1P5 agonist

3640A 987306

Potent and selective H4 receptor antagonist


High affinity Smurf1 inhibitor; enhances BMP signaling


Potent and selective polynucleotide kinase/phosphatase (PNKP) inhibitor

1234A23187, free acid

Calcium ionophore


ALDH1A1 inhibitor


Potent and selective PI 3-kinase p110α inhibitor

0378A-7 hydrochloride

Calmodulin antagonist


Potent and selective CCK1 agonist; suppresses feeding

3025AA 2414

Thromboxane A2 (TP) receptor antagonist

3972AA 29504

Positive allosteric modulator of GABAA receptors


Phospholipase A2 inhibitor


Selective Hsp90 inhibitor

5462AAQ chloride

Photoswitchable Kv channel blocker

4148Abacavir hemisulfate

Reverse transcriptase inhibitor; antiretroviral


Photo-crosslinking probe


Selective GPR55 agonist; neurobehaviorally inactive

5229ABP 688

High affinity human mGlu5 receptor antagonist


Cytochrome P450 inhibitor; inhibits 20-HETE synthesis

5079ABT 089 dihydrochloride

High affinity and selective α4β2 partial agonist

2372ABT 702 dihydrochloride

Adenosine kinase inhibitor; orally active

2214ABT 724 trihydrochloride

Potent, selective D4 partial agonist; proerectile

4138ABT 751

Inhibitor of microtubule polymerization; antimitotic and antitumor

5053AC 186

Potent and selective ERβ agonist; neuroprotective

3419AC 187

Potent and selective amylin receptor antagonist

4046AC 261066

RARβ2 agonist

3370AC 264613

PAR2 receptor agonist

5464AC 4

Photoswitchable TRPV1 channel blocker

3043AC 45594

SF-1 inverse agonist

5281AC 5216

Selective TSPO ligand

3369AC 55541

Potent and selective PAR2 agonist

2436AC 55649

Selective RARβ2 agonist

5013AC 710

Potent and selective PDGFR family inhibitor

2484(±)-AC 7954 hydrochloride

Non-peptide UT receptor agonist


Chloride transport inhibitor


Annexin/lipocortin 1-mimetic; inhibits leukocyte extravasation


Annexin/lipocortin 1-mimetic; inhibits leukocyte extravasation


Annexin I N-terminal peptide; acts as a FPR1 ligand

3618Acamprosate calcium

GABA agonist and glutamatergic modulator

5540Acamprosate - d6 calcium

Deuterated acamprosate (Cat. No. 3618)


Glucosidase α inhibitor (intestinal)


NMDA antagonist, acts at glycine site


Potent, selective L-glutamate uptake inhibitor

2254ACDPP hydrochloride

Selective mGlu5 receptor antagonist


Potent, highly selective CB1 agonist


High affinity angiotensin-converting enzyme (ACE) ligand


Anticholinesterase insecticide


Potent antagonist of GluR5-containing kainate receptors


Cyclooxygenase inhibitor; may be selective for COX-3

5852Acetyl Pepstatin

High affinity aspartic protease inhibitor; inhibits HIV-1/2 proteinases


Nitroxyl precursor

0355(±)-Acetylcarnitine chloride

Intermediate in lipid metabolism

2809Acetylcholine chloride

Endogenous neurotransmitter

5619N-Acetylcysteine amide

Glutathione (GSH) precursor; neuroprotective

03524-Acetyl-1,1-dimethylpiperazinium iodide

Nicotinic agonist

0395N-Acetylglycyl-D-glutamic acid

Potent convulsant


Cathepsin inhibitor

03511-Acetyl-4-methylpiperazine hydrochloride

Nicotinic agonist

1930N-Acetyl-O-phosphono-Tyr-Glu Dipentylamide

Phosphopeptide ligand for src SH2 domain


Phosphopeptide ligand for src SH2 domain


Downregulates SnoN and Ski protein expression; promotes TGF-β signaling


Substrate for serotonin N-acetyl transferase


Selective IKKα and IKKβ inhibitor


Hypolipidemic agent; agonist for the GPR109A (HM74A) and GPR109B receptors


Antilipolytic agent


Potent, selective CB1 agonist

1781ACPA (in Tocrisolve™ 100)

Potent, selective CB1 agonist (in water-soluble emulsion)


Group I/group II mGlu agonist


Potent NMDA agonist. Also group II mGluR agonist


Group I/group II mGlu agonist


Group III mGlu agonist


Competitive mGlu receptor antagonist

5092Acridine Orange hydrochloride

Nucleic acid binding dye


Artificial cerebrospinal fluid

4983ACT 335827

Potent and selective OX1 antagonist

5319ACT 462206

Potent, dual orexin receptor antagonist

3492ACTH (1-39)

Potent endogenous MC2 agonist

1229Actinomycin D

Inhibits RNA polymerase

3205ACV 1

α9α10-selective antagonist


Inhibits viral DNA polymerase; antiherpetic agent


RARβ and RARγ agonist


p210bcr/abl kinase inhibitor


HIF-prolyl hydroxylase-2 (PHD2) inhibitor; antioxidant


Adenine receptor agonist


Endogenous adenosine receptor agonist

3633Adenosine 5'-(α,β-methylene)diphosphate sodium salt

Ecto-5'-nucleotidase (CD73) inhibitor

5096AdipoRon hydrochloride

Orally active AdipoR1 and AdipoR2 agonist; antidiabetic


Selective, high affinity, non-competitive α1A adrenoceptor antagonist

4812ADWX 1

Potent and selective KV1.3 channel blocker

4416ADX 10059 hydrochloride

Negative allosteric modulator at mGlu5

5715(±)-ADX 71743

Negative allosteric modulator at mGlu7; brain penetrant


Broad spectrum, irreversible inhibitor of serine proteases

5318AEE 788

Potent EGFR and VEGFR inhibitor

2651AEG 3482

Inhibitor of JNK signaling

5330AEG 40730 dihydrochloride

IAP antagonist; induces apoptosis

1793AF 12198

Potent, selective human type I IL-1 receptor antagonist

1105AF-DX 116

Selective M2 antagonist

1345AF-DX 384

Potent M2/M4 antagonist

2730AG 045572

Selective GnRH receptor antagonist

1276AG 1478 hydrochloride

Highly potent EGFR-kinase inhibitor

0493AG 18

EGFR/PDGFR-kinase inhibitor

0414AG 490

EGFR-kinase inhibitor. Also JAK2, JAK3 inhibitor

0619AG 494

Potent EGFR-kinase inhibitor

0618AG 555

Potent EGFR-kinase inhibitor

0616AG 556

EGFR-kinase inhibitor

1555AG 825

Selective ErbB2 inhibitor

2617AG 879

TrkA inhibitor

0497AG 99

EGFR-kinase inhibitor

2799ω-Agatoxin IVA

Ca2+ channel blocker (P-type)

2802ω-Agatoxin TK

Ca2+ channel blocker (P/Q-type)

5195Agitoxin 2

Potent Shaker K+ channel blocker

3233AGK 2

Selective SIRT2 inhibitor

0842Agmatine sulfate

α2 ligand. Also imidazoline ligand

1072AGN 192403 hydrochloride

I1 selective ligand

0998AH 11110 hydrochloride

Subtype-selective α1B ligand

0671AH 6809

EP1 and EP2 receptor antagonist

5256AH 7614

Selective FFA4 (GPR120) antagonist


ARE activator; induces Nrf2-ARE-dependent transcription


AMPK activator


Potent, selective group I mGlu antagonist

4946AIM 100

Potent and selective Ack1 (TNK2) inhibitor

0678(+)-AJ 76 hydrochloride

Antagonist; preferential action at D2-like autoreceptors

4754AK 7

Selective SIRT2 inhibitor; brain penetrant

1353Akt/SKG Substrate Peptide

Akt/PKB substrate (synthetic)


Potent and selective dual Akt1 and 2 inhibitor


Akt/PKB substrate (synthetic)

4753AL 8697

Potent and selective p38α inhibitor


Stable form of L-glutamine; commonly used in cell culture


Endogenous glycine agonist, more selective than taurine (Cat. No. 0209)


Glycine receptor agonist


Antiproliferative; induces activin/Smad3 signaling

4005Alda 1

ALDH2 activator; cardioprotective

3979Alexidine dihydrochloride

Selective inhibitor of PTPMT1


Prodrug of vitamin D3 (Cat. No. 4156)

3305Alfuzosin hydrochloride

Uroselective α1 antagonist

5491Aliskiren hemifumarate

Potent renin inhibitor; antihypertensive


GABAA receptor positive allosteric modulator

5532Allopregnanolone - d5

Deuterated allopregnanolone (Cat. No. 3653)

1871α1-Adrenoceptor Tocriset™

Selection of 5 α1-adrenoceptor ligands (Cat. Nos. 1052, 0888, 1006, 0946 and 0623)

1872α2-Adrenoceptor Tocriset™

Selection of 5 α2-adrenoceptor ligands (Cat. Nos. 1030, 0425, 0928, 1133 and 0891)


Direct activator and potentiator of GABAA

2806Alprenolol hydrochloride

β antagonist


Prostaglandin. Vasodilator and antiplatelet agent in vivo


Aldose reductase inhibitor

1809Altanserin hydrochloride

5-HT2A receptor antagonist

1757ALX 5407 hydrochloride

Selective non-transportable GlyT1 inhibitor


Amphibian bombesin-like peptide

2564AM 114

20S proteasome inhibitor

3381AM 1172

Anandamide uptake inhibitor; also FAAH inhibitor and CB receptor partial agonist

1117AM 251

Potent CB1 antagonist; also GPR55 agonist

1115AM 281

Potent, selective CB1 antagonist/inverse agonist

1116AM 404

Anandamide transport inhibitor

5789AM 4668

Potent FFA1 (GPR40) agonist

0760AM 580

Retinoic acid analog; RARα agonist

1120AM 630

CB2 selective antagonist/inverse agonist

5443AM 6545

High affinity and selective CB1 antagonist

3507AM 80

RARα agonist; anticancer

0876AM 92016 hydrochloride

KV channel blocker


Inhibitor of RNA polymerase II

0388Ambenonium dichloride

Cholinesterase inhibitor

2404Ambroxol hydrochloride

Na+ channel blocker

3299AMD 3100 octahydrochloride

Highly selective CXCR4 antagonist

4179AMD 3465 hexahydrobromide

Potent and selective CXCR4 antagonist

4330AMG 21629

Potent and selective TRPV1 antagonist

4487(±)-AMG 487

CXCR3 antagonist; inhibits cell migration and metastasis

3920AMG 548

Potent and selective p38α inhibitor

2316AMG 9810

Potent and selective, competitive antagonist of TRPV1

5517AMG PERK 44

Potent and selective PERK inhibitor; orally bioavailable


D2-like receptor antagonist

0890Amiloride hydrochloride

Na+ channel blocker; also I2 imidazoline ligand


Adenine receptor agonist


PARP inhibitor

0787Aminoguanidine hydrochloride

Irreversible iNOS inhibitor

55145-Aminolevulinic acid hydrochloride

Substrate for detection of δ-aminolevulinic acid dehydratase


H2 antagonist

2072Aminopurvalanol A

Cyclin-dependent kinase inhibitor


Non-selective KV channel blocker

4095Amiodarone hydrochloride

Broad spectrum ion channel blocker; antiarrhythmic


Selective D2/D3 receptor antagonist; atypical antipsychotic agent

4456Amitriptyline hydrochloride

5-HT and noradrenalin re-uptake inhibitor; also TrkA/B agonist


Inhibitor of TBK1 and IKKε; antiallergic agent

2571Amlodipine besylate

Ca2+ channel blocker (L-type)


KV4 channel blocker

2385AMN 082 dihydrochloride

The first selective mGlu7 agonist

1074(RS)-AMPA hydrobromide

Selective AMPA agonist. More water soluble form of (RS)-AMPA (Cat. No. 0169)

1822AMPA Receptor Tocriset™

Selection of 5 AMPA receptor ligands (Cat. Nos. 0254, 0306, 1044, 0713 and 1454)


Inactive isomer of (RS)-AMPA (Cat. No. 0169)


Selective AMPA agonist


Selective AMPA agonist. Active isomer of (RS)-AMPA (Cat. No. 0169)

2813D-Amphetamine sulfate

Induces dopamine, 5-HT and noradrenalin release

5503Ampicillin sodium salt

Antibiotic; selection reagent

1337cAMPS-Rp, triethylammonium salt

cAMP antagonist

1333cAMPS-Sp, triethylammonium salt

Cell-permeable cAMP analog

0871AMT hydrochloride

Potent, selective iNOS inhibitor

3989AMTB hydrochloride

TRPM8 blocker

0668Amthamine dihydrobromide

Highly selective standard H2 agonist


DNA polymerase λ and β inhibitor


Endogenous peptide agonist for amylin, calcitonin, CGRP and adrenomedullin receptors

3391Amyloid β-peptide (42-1) (human)

Inactive control peptide for amyloid β-peptide (1-42) (Cat. No. 1428)

1894Amyloid β-Peptide (12-28) (human)

Amyloid β-peptide; minimum required for binding to brain proteins

1191Amyloid β-Peptide (1-40) (human)

Amyloid β-protein fragment

2424Amyloid β-peptide (1-40) (rat)

Amyloid β-protein fragment

1428Amyloid β-Peptide (1-42) (human)

Predominant amyloid β-protein fragment

2425Amyloid β-peptide (1-42) (rat)

Predominant amyloid β-protein fragment

1938Amyloid β-Peptide (1-43) (human)

Amyloid β-protein fragment

1429Amyloid β-peptide (25-35) (human)

Human amyloid β-protein fragment functionally required for neurotoxicity

4781ANA 12

TrkB receptor antagonist

1971(+)-Anabasine hydrochloride

Neuronal nicotinic receptor partial agonist

3084Anacardic acid

Noncompetitive PCAF/p300 inhibitor

2432Anagrelide hydrochloride

Potent PDE3 inhibitor


Endogenous CB receptor agonist

1017Anandamide (in Tocrisolve™ 100)

Endogenous CB receptor agonist (in water-soluble emulsion)

3717Anandamide - d4

Deuterated anandamide


Potent aromatase (CYP19) inhibitor

0789(±)-Anatoxin A fumarate

Nicotinic agonist


Inhibits NFκB; blocks androgen receptor (AR) expression

1562Angiotensin (1-7)

Vasorelaxant peptide

5335Angiotensin A

Potent endogenous vasoconstrictor peptide - derivative of angiotensin II (Cat. No. 1158)

1563Angiotensin I (human, mouse, rat)

Endogenous precursor to angiotensin II (Cat. No. 1158)

1158Angiotensin II

Potent vasoconstrictor peptide


Desensitization inhibitor (AMPA > kainate)


JNK, SAPK and p38 activator

0703Anpirtoline hydrochloride

Highly potent 5-HT1B agonist. Also 5-HT3 antagonist

5074ANQ 11125

Selective motilin receptor antagonist

3937ANR 94

Adenosine A2A antagonist

1954Antagonist G

Broad spectrum neuropeptide receptor antagonist

2778Antalarmin hydrochloride

CRF1 antagonist

0791Antazoline hydrochloride

Imidazoline ligand


Potent, selective and competitive CRF2 antagonist

3296AP 18

Reversible TRPA1 channel blocker

4274AP 24534

Potent multi-kinase and pan-Bcr-Abl inhibitor

5498AP 811

High affinity, selective NPR3 antagonist


Group I mGlu antagonist

3699DL-AP4 Sodium salt

Broad spectrum EAA antagonist. Sodium salt of DL-AP4 (Cat. No. 0101)


Broad spectrum EAA antagonist


Broad spectrum EAA antagonist


Selective group III mGlu agonist

3693DL-AP5 Sodium salt

Sodium salt of DL-AP5 (Cat. No. 0105)


Potent, selective NMDA antagonist; more active form of DL-AP5 (Cat. No. 0105)


Potent, selective NMDA antagonist


Potent, selective NMDA antagonist. Less active form of DL-AP5 (Cat. No. 0105)


Selective agonist of the 'quis' effect


Specific NMDA antagonist


KCa2 channel blocker (small conductance)


IP3 receptor antagonist. Also TRP channel modulator

2511APC 366

Tryptase inhibitor


Cdc20 inhibitor; inhibits Cdc20-substrate interaction

3704APcK 110

KIT inhibitor


Highly selective group II agonist


Potent peptide agonist for APJ receptor

3007Apelin-17 (human, bovine)

Endogenous APJ receptor agonist

2426Apelin-36 (human)

Endogenous APJ receptor agonist

2427Apelin-36 (rat, mouse)

Endogenous APJ receptor agonist


ASIC3 channel blocker


DNA polymerase α, δ and ε inhibitor


Selective Akt/PKB inhibitor. Antitumor


Selective inhibitor of Akt/PKB signaling. Antitumor and antiviral


Selective group II antagonist


Potent histone deacetylase inhibitor


Protein kinase inhibitor


NADPH-oxidase inhibitor

2073(R)-(-)-Apomorphine hydrochloride

Dopamine agonist; non-subtype-selective

2098Apoptosis Activator 2

Promotes apoptosome formation and activates caspase-9/caspase-3 pathway. Selectively induces tumor cell apoptosis


Competitive serine protease inhibitor

4865APY 29

Inhibits IRE1α autophosphorylation; activates IRE1α endoribonuclease activity


5-HT3 antagonist

2292AQ-RA 741

Selective, high affinity M2 antagonist

3966AR-A 014418

Selective GSK-3 inhibitor

2756Arachidonic acid (in Tocrisolve™100)

Endogenous free fatty acid (in water-soluble emulsion)

2836Arachidonyl serotonin

Dual FAAH inhibitor/TRPV1 antagonist


Inhibits pain in vivo


Endogenous cannabinoid agonist; potent GPR55 agonist


Endocannabinoid. Suppresses pain in vivo

3969AR-C 102222

Selective iNOS inhibitor

4890AR-C 118925XX

Selective, competitive P2Y2 receptor antagonist

0928ARC 239 dihydrochloride

α2B antagonist

3321AR-C 66096 tetrasodium salt

Potent and selective P2Y12 antagonist


MCT1 and MCT2 inhibitor; inhibits glycolysis in cancer cells

0389Arcaine sulfate

Competitive NMDA antagonist


Potent MEK1 inhibitor. Also inhibits IκBα phosphorylation

2457Arcyriaflavin A

Potent cdk4/cyclin D1 and CaM Kinase II inhibitor. Antiviral agent (anti-HCMV)

0383Arecaidine propargyl ester tosylate

Muscarinic agonist


Potent thrombin inhibitor


Endogenous substrate for NOS


High affinity D2 and 5-HT1A receptor partial agonist; also 5-HT2A antagonist

3319ARL 17477 dihydrochloride

Selective nNOS inhibitor

1283ARL 67156 trisodium salt

NTPDase inhibitor

4335AR-M 1000390 hydrochloride

Low-internalizing δ agonist

2699AR-M 1896

GAL2 agonist

4574ARN 272

FAAH-like anandamide transporter (FLAT) inhibitor

2621ARP 100

Selective inhibitor of MMP-2

2622ARP 101

Inhibitor of MMP-2

3964AR-R 17779 hydrochloride

α7-selective agonist

4676ARRY 520 trifluoroacetate

Potent and selective kinesin spindle protein (KSP) inhibitor; induces Mcl-1 degradation


Antimalarial; inhibits P-type ATPase (PfATP6) of P.falciparum


Potent CB1 and TRPV1 agonist. Also anandamide transport inhibitor

2446AS 101

Immunomodulator; inhibits IL-10 synthesis and potentiates IL-1α, IL-2 and TNF-α release

4177AS 1269574

GPR119 receptor agonist

4927AS 1892802

Potent ROCK inhibitor; orally bioavailable

1968AS 19

Potent 5-HT7 agonist

3718AS 1949490

SH2 domain-containing inositol 5'-phosphatase 2 (SHIP2) inhibitor

5035AS 2034178

Selective FFA1 (GPR40) agonist

5430AS 2444697

Potent and selective IRAK4 inhibitor

3671AS 252424

Selective inhibitor of PI 3-kinase γ

3578AS 605240

Potent and selective PI 3-kinase γ (PI 3-Kγ) inhibitor

6044AS 8351

Induces reprogramming of fibroblasts into functional cardiomyocytes


Calcineurin phosphatase inhibitor; analog of FK 506 (Cat. No. 3631)

4055L-Ascorbic acid

Enhances the generation of iPSCs; increases reprogramming efficiency

3737Asenapine maleate

Novel antipsychotic agent

5308ASP 2535

Potent and selective GlyT1 inhibitor

5310ASP 3026

Potent anaplastic lymphoma kinase (ALK) inhibitor; also potent ACK inhibitor

5178ASP 7663

Selective TRPA1 activator

0213D-Aspartic acid

NMDA agonist

0214L-Aspartic acid

NMDA agonist


Cyclooxygenase inhibitor; NSAID


Orally active, potent H1 antagonist. Also KV11.1 (hERG) channel blocker.


Potent CRF receptor antagonist

2391Astressin 2B

Selective CRF2 antagonist

3367AT 101

Downregulates Bcl-2 and Mcl-1; pro-apoptotic

4468AT 1015

Long-acting 5-HT2A antagonist

3531AT 56

L-PGDS inhibitor

3359ATC 0065

Potent and selective MCH1 antagonist

3346ATC 0175 hydrochloride

MCH1 antagonist; also 5-HT2B antagonist and 5-HT1A partial agonist


β1 antagonist


β1-antagonist. Active isomer of atenolol (Cat. No. 0387)

5795ATI 2341

CXCR4 allosteric agonist

2937Atipamezole hydrochloride

Selective α2 antagonist

4580Atiprimod dihydrochloride

JAK2 inhibitor

3776Atorvastatin hemicalcium salt

Potent HMG-CoA reductase inhibitor

3245ATP disodium salt

P2 agonist


Selective, potent GluR5 agonist

4080ATPγS tetralithium salt

P2 agonist; ATP (Cat. No. 3245) analog

1912Atrial natriuretic factor (1-28) (rat)

Endogenous peptide regulating blood pressure

1906Atrial natriuretic factor (1-28) (human, porcine)

Endogenous peptide regulating blood pressure


Thioredoxin reductase inhibitor; induces MPT

1688Autocamtide-2-related inhibitory peptide

Selective CaM kinase II inhibitor

5959Autocamtide-2-related inhibitory peptide, myristoylated

CaM kinase II inhibitor; enhanced cell permeable derivative of Autocamtide-2-related inhibitory peptide

4397AV 412

Potent inhibitor of EGFR, ErbB2 and Abl receptor tyrosine kinases


Potent and selective human V1B agonist


Potent VEGFR-1, -2 and -3 inhibitor

1639AY 9944 dihydrochloride

Inhibitor of Hedgehog (Hh) signaling. Inhibits Δ7-dehydrocholesterol reductase


Selective PAR4 agonist

2172AZ 10417808

Selective non-peptide caspase-3 inhibitor

3323AZ 10606120 dihydrochloride

Potent P2X7 receptor antagonist

3317AZ 11645373

Potent and selective human P2X7 antagonist

4838AZ 12080282 dihydrochloride

Inhibitor of Hedgehog (Hh) signaling

4832AZ 12216052

Positive allosteric modulator at mGlu8

5232AZ 191

Potent DYRK1B inhibitor

5198AZ 20

Potent and selective ATR kinase inhibitor; antitumor

3994AZ 3146

Potent and selective Mps1 kinase inhibitor

5775AZ 6102

Potent TNKS1/2 inhibitor

4836AZ 628

Potent Raf kinase inhibitor

5742AZ PFKFB3 67

Potent and selective PFKFB3 inhibitor


DNA methyltransferase inhibitor


Purine analog; prodrug of 6-mercaptopurine (Cat. No. 4103)

5617AZD 1480

Potent and selective JAK2 inhibitor; antiangiogenic

5614AZD 2066

mGlu5 antagonist; orally bioavailable and brain penetrant

5615AZD 3147

Potent and selective dual mTORC1 and 2 inhibitor; orally bioavailable

4837AZD 3988

Potent and selective DGAT-1 inhibitor

3968AZD 5438

Potent cyclin-dependent kinase (cdk) 1, 2 and 9 inhibitor

5141AZD 5582 dihydrochloride

Dimeric Smac mimetic; potent IAP inhibitor

4839AZD 6482

Potent and selective PI 3-Kβ inhibitor

5199AZD 7762 hydrochloride

Potent and selective ATP-competitive inhibitor of Chk1 and Chk2

5613AZD 9272

Potent and selective mGlu5 antagonist; brain penetrant


Click-activated fluorescent probe


Selective reverse transcriptase inhibitor; antiretroviral


Potent AT1 receptor inverse agonist; antihypertensive


Antibiotic; inhibits 50S ribosomal subunit formation and elongation at transpeptidation

3963AZM 475271

Src tyrosine kinase inhibitor


Unfolded protein response (UPR) modulator

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