Tocris Bioscience

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Product Pages Catalogue Numbers 2001 - 2100

Cat. No. Product Name & Pharmacological Action
2001GS 39783
Positive modulator at GABAB receptors
2002Ro 31-8220 mesylate
Protein kinase inhibitor
2004Isradipine
Ca2+ channel blocker (L-type)
2005Ro 04-5595 hydrochloride
Selective NR2B antagonist
2006Paxilline
Potent blocker of BKCa channels
2007Fluticasone propionate
Selective high affinity glucocorticoid agonist
2008SKF 86002 dihydrochloride
p38 MAP kinase inhibitor; anti-inflammatory agent
2009PSB 1115 potassium salt
Selective human A2B receptor antagonist; water-soluble
2010PSB 10 hydrochloride
Potent, highly selective human A3 receptor antagonist/inverse agonist
2011Tomoxetine hydrochloride
Potent, selective noradrenaline re-uptake inhibitor
2012PSB 11 hydrochloride
Potent, selective human A3 receptor antagonist/inverse agonist
2013Guggulsterone
Broad spectrum steroid receptor ligand. Antagonises FXR and displays hypolipidaemic activity
2018Mirtazepine
Potent 5-HT2 antagonist. Also 5-HT3, H1 and α2-antagonist. Antidepressant
2019PSB 36
Potent, A1-selective antagonist
2020Ch 55
Potent retinoic acid receptor (RAR) agonist
2021LE 135
RARβ-selective antagonist
2022SR 202
Selective PPARγ antagonist; antidiabetic and antiobesity agent
2023Medetomidine hydrochloride
Potent, highly selective α2 agonist
2025Cinalukast
Potent, selective CysLT1 (LTD4) antagonist; orally active
2027Anti-mGlu2
Antibody recognising rat mGlu2 receptors
2029Anti-mGlu2/3
Antibody recognising human mGlu2 and mGlu3 receptors
2031Anti-mGlu7
Antibody recognising human mGlu7 receptors
2032Anti-mGlu5
Antibody recognising rat mGlu5 receptors
2033Pentostatin
Adenosine deaminase inhibitor
2034ROS 234 dioxalate
Potent H3 antagonist
2035BWX 46
Highly selective Y5 agonist
2037SDZ 205-557 hydrochloride
5-HT4/5-HT3 receptor antagonist
2038Iloprost
Prostacyclin (PGI2) analogue
2039CI 898 trihydrochloride
Dihydrofolate reductase inhibitor
2041Anti-phospho-GluR1 (Ser831)
Antibody recognising rat GluR1 subunits phosphorylated at Ser831
2046Anti-GluR4
Antibody recognising rat GluR4 subunits
2047Anti-GluR5
Antibody recognising rat GluR5 subunits
2048Anti-GluR6/7
Antibody recognising rat GluR6 and GluR7 subunits
2049Anti-glutamate receptor δ1/2
Antibody recognising rat glutamate receptor δ1 and δ2 subunits
2052Anti-phospho-NR1 (Ser896)
Antibody recognising rat NR1 subunits phosphorylated at Ser896
2053Anti-phospho-NR1 (Ser897)
Antibody recognising rat NR1 subunits phosphorylated at Ser897
2054Anti-NR1, alternative CT
Antibody recognising rat NR1 subunits with alternative C-terminus
2056Anti-phospho-NR2A (Ser1232)
Antibody recognising rat NR2A subunits phosphorylated at Ser1232
2059Anti-NR3A
Antibody recognising rat NR3A subunits
2060Anti-NR3B
Antibody recognising mouse NR3B subunits
2062Anti-KA2
Antibody recognising rat KA2 subunits
2063Anti-glutamate transporter GLT-1
Antibody recognising GLT-1
2064Anti-glutamate transporter GLAST
Antibody recognising GLAST
2066Anti-c-Fos
Antibody recognising c-Fos
2067187-1, N-WASP inhibitor
Inhibits actin assembly
2070K 41498
Highly selective and potent CRF2 antagonist
2071Antisauvagine-30
Potent, selective and competitive CRF2 antagonist
2072Aminopurvalanol A
Cyclin-dependent kinase inhibitor
2073(R)-(-)-Apomorphine hydrochloride
Dopamine agonist; non-subtype-selective
2074SKF 83959 hydrobromide

D1-like partial agonist

2075SKF 83822 hydrobromide
Selective D1-like agonist
2076Y-26763
KATP channel opener
2077Y-27152
Prodrug of KATP channel opener Y-26763; orally active in vivo
2078UBP 296
Selective, potent kainate antagonist; selective for GLUK5-containing receptors
2079UBP 302
Selective, potent kainate antagonist; active enantiomer of UBP 296 (Cat. No. 2078)
2080PHM 27 (human)
Potent calcitonin receptor agonist; endogenous analogue of human VIP
2081Exendin-3 (9-39) amide
Potent GLP-1 receptor antagonist
2082Glucagon-like peptide 1 (7-36) amide (human, rat, mouse)
Potent insulinotropic peptide
2084GIP (human)
Potent insulinotropic gut hormone
2085Galnon
Selective, non-peptide GalR1 agonist
2086GTP 14564
Class III receptor tyrosine kinase (RTK) inhibitor
2087NTR 368
p75NTR fragment; induces apoptosis
2088DMNB
DNA-dependent protein kinase inhibitor
2089RS 102895 hydrochloride
CCR2b chemokine receptor antagonist
2090CALP1
Cell-permeable calmodulin agonist
2092Ionomycin free acid
Calcium ionophore
2094Oxyntomodulin
Endogenous gut peptide; modulates feeding and metabolism
2095PNU 37883 hydrochloride
Vascular KATP channel blocker
2096DAU 5884 hydrochloride
M3 receptor antagonist
2097SKI II
Selective non-lipid inhibitor of sphingosine kinase; antitumour
2098Apoptosis Activator 2
Promotes apoptosome formation and activates caspase-9/caspase-3 pathway. Selectively induces tumour cell apoptosis
2100Anti-mGlu2 blocking peptide
Blocking peptide for anti-mGlu2 (Cat. No. 2027)
 
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