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Product Pages Catalogue Numbers 1901 - 2000

Cat. No.	Product Name & Pharmacological Action
1901	[Ala¹¹³]-MBP (104-118)
	Protein kinase C inhibitor
1902	[Ala⁹²]-p16 (84-103)
	Cyclin-dependent kinase inhibitor
1903	Peptide F9
	Inhibits laminin-mediated cell adhesion and migration
1904	PKA inhibitor fragment (6-22) amide
	Potent protein kinase A inhibitor
1905	VIP (6-28) (human, rat, porcine, bovine)
	VIP antagonist
1906	Atrial natriuretic factor (1-28) (human, porcine)
	Endogenous peptide regulating blood pressure
1907	Neuromedin N (rat, mouse, porcine, canine)
	Neurotensin-like peptide
1908	Neuromedin B (porcine)
	Mammalian bombesin-like peptide
1909	Neurotensin
	Endogenous neurotransmitter and endocrine modulator
1910	Oxytocin
	Involved in uterine contraction and lactation
1911	VIP (human, rat, mouse, rabbit, canine, porcine)
	Involved in neurotransmission, smooth muscle relaxation
1912	Atrial natriuretic factor (1-28) (rat)
	Endogenous peptide regulating blood pressure
1913	[D-Phe¹²]-Bombesin
	Bombesin receptor antagonist
1914	Eledoisin
	Potent tachykinin receptor ligand
1915	Kinetensin (human)
	Neurotensin-like peptide
1916	Litorin
	Amphibian bombesin-like peptide
1917	Neuromedin U (rat)
	Endogenous modulator of blood pressure and flow, gut ion transport, feeding and body temperature
1918	Secretin (human)
	Gastrointestinal peptide
1919	Secretin (rat)
	Gastrointestinal peptide
1920	Eledoisin-Related Peptide
	Tachykinin receptor ligand
1921	N-Formyl-Met-Leu-Phe
	Endogenous FPR agonist
1922	[D-Lys³]-GHRP-6
	GHS receptor antagonist
1923	pp60 c-src (521-533) (phosphorylated)
	Inhibits tyrosine kinase activity of pp60^c-src and pp60^v-src
1926	MLCK inhibitor peptide
	Myosin light chain kinase inhibitor
1927	N-Acetyl-O-phosphono-Tyr-Glu-Glu-Ile-Glu
	Phosphopeptide ligand for src SH2 domain
1928	Neuropeptide AF (human)
	Implicated in pain modulation, opioid function and metabolism
1929	Melanocyte stimulating hormone release inhibiting factor
	Inhibitor of α-MSH release; inhibits opioid effects in vivo
1930	N-Acetyl-O-phosphono-Tyr-Glu Dipentylamide
	Phosphopeptide ligand for src SH2 domain
1931	G-Protein antagonist peptide
	Inhibits G protein activation by GPCRs
1932	U 46619
	Potent, stable thromboxane A₂ (TP) receptor agonist
1933	Exendin-4
	Potent GLP-1 receptor agonist
1935	Caffeic acid-pYEEIE
	Phosphopeptide ligand for src SH2 domain
1937	NSC 693868
	Cdk inhibitor. Also inhibits GSK-3
1938	Amyloid β-Peptide (1-43) (human)
	Amyloid β-protein fragment
1939	C14TKL-1
	Endogenous NK₁ agonist
1941	m-3M3FBS
	Phospholipase C activator
1942	o-3M3FBS
	Inactive analogue of m-3M3FBS (Cat. No. 1941)
1944	Loratidine
	Peripheral H₁ antagonist; anti-allergic agent
1946	[D-Arg¹,D-Phe⁵,D-Trp^7,9,Leu¹¹]-Substance P
	Potent ghrelin receptor full inverse agonist. Also antagonist at other neuropeptide receptors. Anticancer in vitro
1947	PR 39 (porcine)
	IκBα inhibitor
1949	L-670,596
	Potent, selective thromboxane A₂/prostaglandin endoperoxide antagonist
1950	Gap 26
	Gap junction blocker; inhibits smooth muscle contraction and IP₃-mediated ATP release
1952	DCB
	Allosteric modulator at mGlu₅
1953	DMeOB
	Negative allosteric modulator at mGlu₅
1954	Antagonist G
	Broad spectrum neuropeptide receptor antagonist
1955	Ritanserin
	Potent 5-HT₂ antagonist
1956	Bestatin
	Aminopeptidase inhibitor
1957	GR 79236
	A₁ agonist
1958	GR 32191 hydrochloride
	Potent thromboxane A₂/TP receptor antagonist
1959	GW 311616 hydrochloride
	Potent, selective human neutrophil elastase inhibitor
1960	SB 334867
	Selective non-peptide OX₁ antagonist
1961	SB 258585 hydrochloride
	Potent, selective 5-ht₆ antagonist
1962	SB 239063
	Potent, selective p38 MAP kinase inhibitor; orally active
1963	SB 408124
	Selective non-peptide OX₁ antagonist
1964	Gossypol
	Anticancer, antifertility agent
1965	Simvastatin
	HMG-CoA reductase inhibitor
1966	UCM 707
	Potent anandamide transport inhibitor
1967	Ranitidine hydrochloride
	Selective H₂ antagonist
1968	AS 19
	Reported potent 5-HT₇ agonist
1969	SL 327
	Selective inhibitor of MEK1 and MEK2; brain penetrant
1970	Norketamine hydrochloride
	Potent, non-competitive NMDA antagonist
1971	(+)-Anabasine hydrochloride
	Neuronal nicotinic receptor agonist
1972	Tianeptine sodium salt
	Selective facilitator of 5-HT uptake; antidepressant
1974	SANT-1
	Inhibitor of hedgehog (hh) signalling; antagonises smoothened activity
1975	6-Iodonordihydrocapsaicin
	Potent, competitive vanilloid receptor antagonist
1979	L-803,087 trifluoroacetate
	Potent and selective sst₄ agonist
1980	L-817,818
	Potent and selective sst₅ agonist
1982	Reboxetine mesylate
	Potent, selective noradrenaline uptake inhibitor; orally active
1983	740 Y-P
	Cell-permeable PI 3-kinase activator
1984	Nogo-66 (1-40)
	Competitive antagonist for Nogo-66 receptor; promotes neuron regeneration
1985	PNU 142633
	Highly selective 5-HT_1D agonist
1987	Leptomycin B
	Inhibits nuclear export of proteins; antitumour
1989	c-JUN peptide
	Peptide inhibitor of JNK/c-Jun interaction
1990	(R,R)-THC
	Potent subtype selective ligand; ERα agonist/ERβ antagonist
1991	MPP dihydrochloride
	Highly selective ERα antagonist
1994	ZK 93423 hydrochloride
	Potent benzodiazepine agonist
1995	Ro 19-4603
	Benzodiazepine inverse agonist
1996	ZK 93426 hydrochloride
	Potent, competitive benzodiazepine antagonist
1997	Ro 15-4513
	Benzodiazepine partial inverse agonist
1998	JMV 449
	Potent neurotensin receptor agonist
1999	Linopirdine dihydrochloride
	KCNQ channel blocker
2000	XE 991 dihydrochloride
	Potent, selective KCNQ channel blocker; blocks M-current

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