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Product Pages Catalogue Numbers 1101 - 1200

Cat. No. Product Name & Pharmacological Action
1101Cyclosporin A
Calcineurin inhibitor
1102Procaterol hydrochloride

Potent β2 agonist

1103Ketoconazole
Cytochrome P450c17 inhibitor
11042-Cl-IB-MECA
Highly selective A3 agonist
1105AF-DX 116

Selective M2 antagonist

1107ATPA
Selective, potent GluR5 agonist
1109GR 103691

Highly selective D3 antagonist

1110Genistein
EGFR-kinase, topoisomerase kinase inhibitor
1111ACPT-I
Group III mGlu agonist
1112ACPT-II
Competitive mGlu receptor antagonist
1114CGP 37157
Antagonist of mitochondrial Na+/Ca2+ exchange
1115AM 281

Potent, selective CB1 antagonist/inverse agonist

1116AM 404

Anandamide transport inhibitor

1117AM 251
Potent, selective CB1 antagonist/inverse agonist
1118Nocistatin (bovine)
Opposes action of nociceptin
1119NocII
Orphan neuropeptide
1120AM 630

CB2 selective antagonist/inverse agonist

1121(R)-(+)-Methanandamide

Potent and selective CB1 agonist

1122Telenzepine dihydrochloride

Potent selective M1 antagonist

1123(S)-(+)-Niguldipine hydrochloride
α1 antagonist, L-type Ca2+ channel blocker
1124(R)-(-)-Niguldipine hydrochloride
Less active enantiomer of Cat. No. 1123
1125Quercetin
Non-selective PI 3-kinase inhibitor
1126Dexamethasone
Anti-inflammatory glucocorticoid
1127Yohimbine hydrochloride

 α2-selective antagonist

1128Picrotoxin
GABAA receptor antagonist
1129BRL 54443
Potent 5-ht1E/F agonist
1130LY 294002 hydrochloride
Selective PI 3-kinase inhibitor
1131KU14R
Antagonist of pancreatic imidazoline receptor
1132Harmane
Putative endogenous imidazoline ligand. Also MAO inhibitor
1133BRL 44408 maleate

Selective α2A antagonist

1134CGP 12177 hydrochloride
β3 partial agonist. β1/β2 antagonist.
1135Spermine NONOate
Slow NO releasing agent
1136Okadaic acid
Protein phosphatase 1 and 2A inhibitor
1137Resiniferatoxin
Ultrapotent vanilloid receptor agonist
1138Thapsigargin
Potent inhibitor of SERCA ATPase
1139L-NIL hydrochloride
Selective iNOS inhibitor
11408-Bromo-cAMP, sodium salt
Cell-permeable cAMP analogue
1141Dibutyryl-cAMP, sodium salt
Cell-permeable cAMP analogue
1142Oxymetazoline hydrochloride
α1A agonist
1143Corynanthine hydrochloride
α1 antagonist
1144U0126
Potent, selective inhibitor of MEK1 and 2
1145L-733,060 hydrochloride
Potent NK1 antagonist
1147SKF 96365 hydrochloride
Receptor-operated calcium channel blocker
1148Siguazodan
PDE3 inhibitor
1149Bombesin
Involved in gastrointestinal tract function
1150CCK Octapeptide, non-sulfated
Non-sulfated form of CCK octapeptide
1151CRF (human, rat)
Stimulates ACTH release
1152Neurokinin A (porcine)
Endogenous tachykinin peptide
1153Neuropeptide Y (human, rat)
Influences feeding and sexual behaviour
1154Pancreatic Polypeptide (human)
NPY Y4 agonist; involved in gastrointestinal tract function
1155RR-src
Tyrosine kinase substrate peptide
1156Substance P
Sensory neuropeptide, inflammatory mediator
1157Somatostatin
Influences growth hormone release
1158Angiotensin II
Potent vasoconstrictor peptide
1159Calcitonin (salmon)
Affects bone formation and resorption
1160Endothelin 1 (human, porcine)
Potent vasoconstrictor peptide
1161CGRP (rat)
Potent vasodilator
1162Endothelin 3 (human, rat)
Potent vasoconstrictor
1163Saralasin
Non-selective angiotensin II antagonist
1164Endothelin 2 (human)
ETA/ETB agonist
1165Somatostatin 1-28
Somatostatin receptor agonist
1166CCK Octapeptide, sulfated
C-terminal octapeptide of CCK
1167Leupeptin hemisulfate
Inhibits trypsin-like/cysteine proteases
1168[Leu31,Pro34]-Neuropeptide Y (porcine)
Neuropeptide YY1 receptor agonist
1169CGRP 8-37 (rat)
CGRP1 receptor antagonist
1170DSLET
Selective δ agonist peptide
1171DAMGO
Selective μ agonist
1172[Ac-Tyr1,D-Phe2]GRF 1-29, amide (human)
VIP antagonist
1173Neuropeptide Y (porcine)
Influences feeding and sexual behaviour
1174Sarafotoxin S6b
Endothelin receptor agonist, non-selective
1175Sarafotoxin S6c
Selective ETB agonist
1176[Leu31,Pro34]-Neuropeptide Y (human, rat)
Neuropeptide YY1 receptor agonist
1177Neuropeptide Y 13-36 (porcine)
Y2 receptor agonist
1178[Sar9,Met(O2)11]-Substance P
Potent, selective NK1 agonist
1179Galanin (1-30) (human)
Modulator of neurotransmission
1180 [D-Ala2]-Deltorphin II
Selective δ agonist peptide
1181CGRP 8-37 (human)
CGRP1 receptor antagonist
1182VIP (guinea pig)
Involved in neurotransmission, smooth muscle relaxation
1183PACAP 1-27
Potent stimulator of adenylyl cyclase
1184α-helical CRF 9-41
CRF receptor antagonist
1185Thrombin Receptor Agonist Peptide
Causes platelet aggregation and secretion
1186PACAP 1-38
Potent stimulator of adenylyl cyclase
1187GRF (ovine)
Stimulates growth hormone release
1188BQ-123
Selective ETA antagonist
1189BQ-3020
Selective ETB agonist
1190Pepstatin A
Aspartic protease inhibitor
1191Amyloid β-Peptide (1-40) (human)
Amyloid β-protein fragment
1192Mastoparan
Activates Gi  and Go
1193Melittin
Inhibits Gs and stimulates Gi activity
1194MDL 29,913
Selective NK2 antagonist
1195IRL-1038
ETB antagonist
1196IRL-1620
Highly selective ETB agonist
1197[Ala1,3,11,15]-Endothelin
Selective ETB agonist
1198Nocistatin (human)
Human putative counterpart of nocistatin
1199NF 279
Potent selective P2X1 antagonist
1200Nω-Propyl-L-arginine
Highly selective inhibitor of nNOS
 
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